Literature DB >> 30927159

A double-blind randomized placebo controlled study assessing safety, tolerability and efficacy of palmitoylethanolamide for symptoms of knee osteoarthritis.

Elizabeth Steels1,2, Ruchitha Venkatesh3, Eleanor Steels4, Gemma Vitetta5, Luis Vitetta6,5.   

Abstract

BACKGROUND: The aim of the study was to assess the safety, tolerability and efficacy of palmitoylethanolamide (PEA) when dosed at 300 mg and 600 mg per day on symptoms of knee osteoarthritis.
METHODS: This was a single site, comparative, double-blind placebo controlled study in adults with mild to moderate knee osteoarthritis with 111 participants randomized to receive 300 mg PEA, 600 mg PEA or placebo each day, in divided doses b.i.d, for 8 weeks. The primary outcome was the Western Ontario and McMaster Universities Osteoarthritis Index (WOMAC). The secondary outcomes were the Numerical Rating Scales (NRS) for pain, the Depression Anxiety Stress Scale (DASS), the Perceived Stress Scale (PSS), the Pittsburg Sleep Quality Index (PSQI), the Short Form Health Survey (SF-36), the use of rescue pain medication and clinical safety assessment.
RESULTS: There was a significant reduction in the total WOMAC score in the 300 mg PEA (p = 0.0372) and the 600 mg PEA (p = 0.0012) groups, the WOMAC pain score (300 mg PEA, p = 0.0074; 600 mg PEA, p =  < 0.001), the WOMAC stiffness score (PEA 300 mg, p < 0.0490; 600 mg PEA, p = 0.001) and in the WOMAC function score in the 600 mg PEA group (p = 0.033) compared to placebo. The NRS pain evaluations for "worst pain" and "least pain" were significantly reduced in the 300 mg PEA group (p < 0.001, p = 0.005) and the 600 mg PEA group (p < 0.001, p < 0.001) compared to placebo. There was a significant reduction in anxiety (DASS) in both active treatment groups (300 mg PEA, p = 0.042; 600 mg PEA group (p = 0.043) compared to placebo. There were no changes in the clinical markers and the product was well tolerated.
CONCLUSIONS: The study demonstrated that palmitoylethanolamide may be a novel treatment for attenuating pain and reducing other associated symptoms of knee osteoarthritis. Further studies on the pharmacological basis of this anti-inflammatory effect are now required.

Entities:  

Keywords:  Inflammation; N-acylethanolamines; Osteoarthritis; Pain; Palmitoylethanolamide

Mesh:

Substances:

Year:  2019        PMID: 30927159     DOI: 10.1007/s10787-019-00582-9

Source DB:  PubMed          Journal:  Inflammopharmacology        ISSN: 0925-4692            Impact factor:   4.473


  12 in total

1.  Anti-arthritic effects of Schisandra chinensis extract in monosodium iodoacetate-induced osteoarthritis rats.

Authors:  You-Suk Lee; Sung-Min Kim; Eun-Jung Park; Hae-Jeung Lee
Journal:  Inflammopharmacology       Date:  2022-09-05       Impact factor: 5.093

2.  Inflammatory and Immune Protein Pathways Possible Mechanisms for Pain Following Walking in Knee Osteoarthritis.

Authors:  N Jennifer Klinedinst; Weiliang Huang; Amy K Nelson; Barbara Resnick; Cynthia Renn; Maureen A Kane; Susan G Dorsey
Journal:  Nurs Res       Date:  2022-03-18       Impact factor: 2.364

3.  Safety and efficacy of a new micronized formulation of the ALIAmide palmitoylglucosamine in preclinical models of inflammation and osteoarthritis pain.

Authors:  Marika Cordaro; Rosalba Siracusa; Daniela Impellizzeri; Ramona D' Amico; Alessio Filippo Peritore; Rosalia Crupi; Enrico Gugliandolo; Roberta Fusco; Rosanna Di Paola; Carlo Schievano; Salvatore Cuzzocrea
Journal:  Arthritis Res Ther       Date:  2019-11-28       Impact factor: 5.156

4.  Palmitoylethanolamide: Prenatal Developmental Toxicity Study in Rats.

Authors:  Narendra S Deshmukh; Shailesh Gumaste; Silma Subah; Nathasha Omal Bogoda
Journal:  Int J Toxicol       Date:  2021-02-12       Impact factor: 2.032

5.  Anti-inflammatory activity of palmitoylethanolamide ameliorates osteoarthritis induced by monosodium iodoacetate in Sprague-Dawley rats.

Authors:  Jae In Jung; Hyun Sook Lee; Young Eun Jeon; So Mi Kim; Su Hee Hong; Joo Myung Moon; Cho Young Lim; Yoon Hee Kim; Eun Ji Kim
Journal:  Inflammopharmacology       Date:  2021-09-01       Impact factor: 4.473

Review 6.  Effects of Palmitoylethanolamide (PEA) on Nociceptive, Musculoskeletal and Neuropathic Pain: Systematic Review and Meta-Analysis of Clinical Evidence.

Authors:  Damiana Scuteri; Francesca Guida; Serena Boccella; Enza Palazzo; Sabatino Maione; Juan Francisco Rodríguez-Landa; Lucia Martínez-Mota; Paolo Tonin; Giacinto Bagetta; Maria Tiziana Corasaniti
Journal:  Pharmaceutics       Date:  2022-08-11       Impact factor: 6.525

Review 7.  Palmitoylethanolamide: A Natural Compound for Health Management.

Authors:  Paul Clayton; Mariko Hill; Nathasha Bogoda; Silma Subah; Ruchitha Venkatesh
Journal:  Int J Mol Sci       Date:  2021-05-18       Impact factor: 5.923

8.  Relative Deficiency of Anti-Inflammatory N-Acylethanolamines Compared to Prostaglandins in Oral Lichen Planus.

Authors:  Linda Rankin; Sandra Gouveia-Figueira; Karin P Danielsson; Christopher J Fowler
Journal:  Biomedicines       Date:  2020-11-06

Review 9.  The Basal Pharmacology of Palmitoylethanolamide.

Authors:  Linda Rankin; Christopher J Fowler
Journal:  Int J Mol Sci       Date:  2020-10-26       Impact factor: 5.923

Review 10.  Chronic Pain in Dogs and Cats: Is There Place for Dietary Intervention with Micro-Palmitoylethanolamide?

Authors:  Giorgia Della Rocca; Davide Gamba
Journal:  Animals (Basel)       Date:  2021-03-29       Impact factor: 2.752

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