Literature DB >> 30850503

Effect of External Cooling on 177Lu-PSMA Uptake by the Parotid Glands.

Burcak Yilmaz1, Serap Nisli2, Nurhan Ergul2, Riza Umar Gursu3, Ozgur Acikgoz4, Tevfik Fikret Çermik2.   

Abstract

Recent years have seen the start of treatment of metastatic castration-resistant prostate cancer with prostate-specific membrane antigen (PSMA)-targeted radioligand therapy (PRLT), especially 177Lu-PSMA-617. However, PRLT has side effects on the salivary glands that limit the safety of the treatment. The current study aimed to show the effect of external cooling with ice packs on 177Lu-PSMA-617 uptake by the parotid glands (PGs).
Methods: The study included 19 patients (mean age, 72.9 y) with metastatic castration-resistant prostate cancer who had been referred for the first time for 177Lu-PSMA-617 treatment and underwent pretreatment 68Ga-PSMA-11 PET/CT. Before the initiation of PRLT, the SUVmax and SUVmean of the right and left PGs were measured on 68Ga-PSMA PET/CT. Frozen ice packs were then affixed over the right PG of each patient for approximately 5 h; 1 h after they were affixed, PRLT was administered. At 4 h after PRLT, head-and-neck SPECT/CT was performed, and at both 4 and 24 h after PRLT, whole-body planar scintigraphy was performed. Regions and volumes of interest were applied for the right and left PGs, and the counts and volumes were determined.
Results: Before PRLT, 68Ga-PSMA-11 PET/CT showed no significant difference in SUVmax or SUVmean between the right and left PGs (P > 0.05). At 4 and 24 h after PRLT, planar imaging showed no significant difference in counts between the cooled and noncooled PGs (P > 0.05). Furthermore, at 4 h after PRLT, SPECT/CT showed no significant difference in counts or volumes between the cooled and noncooled PGs (P > 0.05).
Conclusion: External cooling does not reduce uptake of 177Lu-PSMA-617 by the PGs.
© 2019 by the Society of Nuclear Medicine and Molecular Imaging.

Entities:  

Keywords:  177Lu; PSMA; ice-pack; parotid; prostate cancer

Mesh:

Substances:

Year:  2019        PMID: 30850503     DOI: 10.2967/jnumed.119.226449

Source DB:  PubMed          Journal:  J Nucl Med        ISSN: 0161-5505            Impact factor:   10.057


  11 in total

1.  Sublingual Atropine Administration as a Tool to Decrease Salivary Glands' PSMA-Ligand Uptake: A Preclinical Proof of Concept Study Using [68Ga]Ga-PSMA-11.

Authors:  Vincent Nail; Béatrice Louis; Anaïs Moyon; Adrien Chabert; Laure Balasse; Samantha Fernandez; Guillaume Hache; Philippe Garrigue; David Taïeb; Benjamin Guillet
Journal:  Pharmaceutics       Date:  2022-06-16       Impact factor: 6.525

2.  Advances in PSMA theranostics.

Authors:  Thomas M Jeitner; John W Babich; James M Kelly
Journal:  Transl Oncol       Date:  2022-05-18       Impact factor: 4.803

3.  68Ga-PSMA PET/CT: effect of external cooling on salivary gland uptake.

Authors:  Matheus Zanelatto Junqueira; Nelisa Helena Rocha; Marcelo Tatit Sapienza
Journal:  Radiol Bras       Date:  2021 May-Jun

4.  The Impact of Monosodium Glutamate on 68Ga-PSMA-11 Biodistribution in Men with Prostate Cancer: A Prospective Randomized, Controlled Imaging Study.

Authors:  Wesley R Armstrong; Andrei Gafita; Shaojun Zhu; Pan Thin; Kathleen Nguyen; Rejah Alano; Stephanie Lira; Kiara Booker; Linda Gardner; Tristan Grogan; David Elashoff; Martin Allen-Auerbach; Magnus Dahlbom; Johannes Czernin; Jeremie Calais
Journal:  J Nucl Med       Date:  2021-01-28       Impact factor: 11.082

5.  A simple strategy to reduce the salivary gland and kidney uptake of PSMA-targeting small molecule radiopharmaceuticals.

Authors:  Teja Muralidhar Kalidindi; Sang-Gyu Lee; Katerina Jou; Goutam Chakraborty; Myrto Skafida; Scott T Tagawa; Neil H Bander; Heiko Schoder; Lisa Bodei; Neeta Pandit-Taskar; Jason S Lewis; Steven M Larson; Joseph R Osborne; Naga Vara Kishore Pillarsetty
Journal:  Eur J Nucl Med Mol Imaging       Date:  2021-01-25       Impact factor: 10.057

6.  The 68Ga/177Lu-theragnostic concept in PSMA-targeting of metastatic castration-resistant prostate cancer: impact of post-therapeutic whole-body scintigraphy in the follow-up.

Authors:  Johanna Maffey-Steffan; Lorenza Scarpa; Anna Svirydenka; Bernhard Nilica; Christian Mair; Sabine Buxbaum; Jasmin Bektic; Elisabeth von Guggenberg; Christian Uprimny; Wolfgang Horninger; Irene Virgolini
Journal:  Eur J Nucl Med Mol Imaging       Date:  2019-11-27       Impact factor: 9.236

7.  Design of PSMA ligands with modifications at the inhibitor part: an approach to reduce the salivary gland uptake of radiolabeled PSMA inhibitors?

Authors:  Veronika Barbara Felber; Manuel Amando Valentin; Hans-Jürgen Wester
Journal:  EJNMMI Radiopharm Chem       Date:  2021-02-26

8.  Muscarinic inhibition of salivary glands with glycopyrronium bromide does not reduce the uptake of PSMA-ligands or radioiodine.

Authors:  V Mohan; N M Bruin; M E T Tesselaar; J P de Boer; E Vegt; J J M A Hendrikx; A Al-Mamgani; J B van de Kamer; J-J Sonke; W V Vogel
Journal:  EJNMMI Res       Date:  2021-03-12       Impact factor: 3.138

9.  Safety of PSMA-Targeted Molecular Radioligand Therapy with 177Lu-PSMA-617: Results from the Prospective Multicenter Phase 2 Trial RESIST-PC (NCT03042312).

Authors:  Jeremie Calais; Johannes Czernin; Pan Thin; Jeannine Gartmann; Kathleen Nguyen; Wesley R Armstrong; Martin Allen-Auerbach; Andrew Quon; Shadfar Bahri; Pawan Gupta; Linda Gardner; Magnus Dahlbom; Beilei He; Rouzbeh Esfandiari; David Ranganathan; Ken Herrmann; Matthias Eiber; Wolfgang P Fendler; Ebrahim Delpassand
Journal:  J Nucl Med       Date:  2021-07-16       Impact factor: 10.057

Review 10.  Global experience with PSMA-based alpha therapy in prostate cancer.

Authors:  Mike M Sathekge; Frank Bruchertseifer; Mariza Vorster; Alfred Morgenstern; Ismaheel O Lawal
Journal:  Eur J Nucl Med Mol Imaging       Date:  2021-06-26       Impact factor: 9.236

View more

北京卡尤迪生物科技股份有限公司 © 2022-2023.