Literature DB >> 30836094

Real-Time Targeted Genome Profile Analysis of Pancreatic Ductal Adenocarcinomas Identifies Genetic Alterations That Might Be Targeted With Existing Drugs or Used as Biomarkers.

Aatur D Singhi1, Ben George2, Joel R Greenbowe3, Jon Chung3, James Suh3, Anirban Maitra4, Samuel J Klempner5, Andrew Hendifar6, Javle M Milind4, Talia Golan7, Randall E Brand8, Amer H Zureikat9, Somak Roy10, Alexa B Schrock3, Vincent A Miller3, Jeffrey S Ross3, Siraj M Ali3, Nathan Bahary8.   

Abstract

BACKGROUND & AIMS: It has been a challenge to select treatment for patients with pancreatic ductal adenocarcinomas (PDACs) based on genome alterations. We performed targeted genomic profile analyses of a large number of PDACs to assess the full spectrum of actionable genomic alterations.
METHODS: We performed targeted genomic profile analyses of 3594 PDAC samples from an international cohort, including capture-based targeted genomic profiling of as many as 315 cancer-associated genes and intron regions of 28 genes that are rearranged in cancer cells. Tumor mutation burden (TMB) and microsatellite instability (MSI) status were also assessed. TMB was calculated across a 1.14-megabase region; TMB-high was defined as ≥20 mutations/megabase. MSI-high status was assigned based on analysis of 114 intron homopolymer loci.
RESULTS: KRAS, TP53, CDKN2A, and SMAD4 were the most frequently altered genes in PDAC. We found KRAS mutations in 88% of samples. Among PDACs without mutations in KRAS, we found alterations in genes whose products are in the mitogen-activated protein kinase signaling pathway and are candidate drug targets (actionable targets, n = 132; 4%), as well as gene fusions (n = 51), gene amplifications (n = 35), genes with missense mutations (n = 30), and genes that contain deletions (n = 16). Many of these encode proteins in receptor tyrosine kinase, RAS, or mitogen-activated protein kinase signaling pathways. Aside from TP53, alterations in genes encoding DNA damage repair proteins (BRCA and FANC) were detected in 14% of PDACs. Among PDACs evaluated for MSI (n = 2563) and TMB (n = 1021), MSI-high and/or TMB-high phenotypes were detected in 0.5% of samples. Alterations in FGF23, CCND2, PIK3CA, and FGF6 were more commonly detected in intraductal papillary mucinous neoplasm-associated PDACs.
CONCLUSIONS: In targeted genomic profile analyses of 3594 PDACs, we found 17% to contain genomic alterations that might make the tumor cells susceptible to currently used anticancer agents. We identified mutations in genes that could contribute to progression of intraductal papillary mucinous neoplasms into malignancies. These alterations might be used as biomarkers for early detection.
Copyright © 2019 AGA Institute. Published by Elsevier Inc. All rights reserved.

Entities:  

Keywords:  IPMN; Locally Advanced; MAPK; Metastatic

Mesh:

Substances:

Year:  2019        PMID: 30836094     DOI: 10.1053/j.gastro.2019.02.037

Source DB:  PubMed          Journal:  Gastroenterology        ISSN: 0016-5085            Impact factor:   22.682


  73 in total

1.  Ras Variant Biology and Contributions to Human Disease.

Authors:  Ian Prior
Journal:  Methods Mol Biol       Date:  2021

Review 2.  The Impact of Recent Advances in Endoscopic Ultrasound-Guided Tissue Acquisition on the Management of Pancreatic Cancer.

Authors:  Susana Marques; Miguel Bispo; Ricardo Rio-Tinto; Paulo Fidalgo; Jacques Devière
Journal:  GE Port J Gastroenterol       Date:  2020-10-23

3.  Precision Medicine in Pancreatic Disease-Knowledge Gaps and Research Opportunities: Summary of a National Institute of Diabetes and Digestive and Kidney Diseases Workshop.

Authors:  Mark E Lowe; Dana K Andersen; Richard M Caprioli; Jyoti Choudhary; Zobeida Cruz-Monserrate; Anil K Dasyam; Christopher E Forsmark; Fred S Gorelick; Joe W Gray; Mark Haupt; Kimberly A Kelly; Kenneth P Olive; Sylvia K Plevritis; Noa Rappaport; Holger R Roth; Hanno Steen; S Joshua Swamidass; Temel Tirkes; Aliye Uc; Kirill Veselkov; David C Whitcomb; Aida Habtezion
Journal:  Pancreas       Date:  2019 Nov/Dec       Impact factor: 3.327

Review 4.  [Medicinal treatment of pancreatic cancer : Still a domain of chemotherapy?]

Authors:  Georg Feldmann
Journal:  Internist (Berl)       Date:  2020-02       Impact factor: 0.743

Review 5.  The Role of Endoscopic Ultrasound in Pancreatic Cancer Staging in the Era of Neoadjuvant Therapy and Personalised Medicine.

Authors:  Miguel Bispo; Susana Marques; Ricardo Rio-Tinto; Paulo Fidalgo; Jacques Devière
Journal:  GE Port J Gastroenterol       Date:  2020-09-07

Review 6.  Transportome Malfunctions and the Hallmarks of Pancreatic Cancer.

Authors:  Qi Ling; Holger Kalthoff
Journal:  Rev Physiol Biochem Pharmacol       Date:  2021       Impact factor: 5.545

7.  Prolonged response to liposomal irinotecan in a patient with stage IV pancreatic/bile duct cancer previously treated with FOLFIRINOX and gemcitabine plus nab-paclitaxel.

Authors:  A Surinach; T Phung; O Abdul-Rahim; M Khushman
Journal:  Curr Oncol       Date:  2020-05-01       Impact factor: 3.677

Review 8.  The Frequency of Ras Mutations in Cancer.

Authors:  Ian A Prior; Fiona E Hood; James L Hartley
Journal:  Cancer Res       Date:  2020-03-24       Impact factor: 12.701

9.  Identification of Targetable Gene Fusions and Structural Rearrangements to Foster Precision Medicine in KRAS Wild-Type Pancreatic Cancer.

Authors:  Michael J Fusco; Daryoush Saeed-Vafa; Estrella M Carballido; Theresa A Boyle; Mokenge Malafa; Kirsten L Blue; Jamie K Teer; Christine M Walko; Howard L McLeod; J Kevin Hicks; Martine Extermann; Jason B Fleming; Todd C Knepper; Dae Won Kim
Journal:  JCO Precis Oncol       Date:  2021-01-11

Review 10.  First international workshop of the ATM and cancer risk group (4-5 December 2019).

Authors:  Fabienne Lesueur; Douglas F Easton; Anne-Laure Renault; Sean V Tavtigian; Jonine L Bernstein; Zsofia Kote-Jarai; Rosalind A Eeles; Dijana Plaseska-Karanfia; Lidia Feliubadaló; Banu Arun; Natalie Herold; Beatrix Versmold; Rita Katharina Schmutzler; Tú Nguyen-Dumont; Melissa C Southey; Leila Dorling; Alison M Dunning; Paola Ghiorzo; Bruna Samia Dalmasso; Eve Cavaciuti; Dorothée Le Gal; Nicholas J Roberts; Mev Dominguez-Valentin; Matti Rookus; Alexander M R Taylor; Alisa M Goldstein; David E Goldgar; Dominique Stoppa-Lyonnet; Nadine Andrieu
Journal:  Fam Cancer       Date:  2021-06-14       Impact factor: 2.375

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