Literature DB >> 30830724

Safety and efficacy of ertugliflozin in Asian patients with type 2 diabetes mellitus inadequately controlled with metformin monotherapy: VERTIS Asia.

Linong Ji1, Yanmei Liu2, Heng Miao3, Yongli Xie4, Ming Yang5, Wei Wang5, Yuting Mu5, Ping Yan5, Sharon Pan6, Brett Lauring7, Shu Liu8, Susan Huyck7, Yanping Qiu8, Steven G Terra9.   

Abstract

AIM: Phase III, randomized, double-blind study evaluating the efficacy and safety of ertugliflozin in Asian patients with type 2 diabetes mellitus (T2DM) inadequately controlled on metformin, including evaluation in the China subpopulation.
MATERIALS AND METHODS: A 26-week, double-blind study of 506 Asian patients (80.2% from mainland China), randomized 1:1:1 to placebo, ertugliflozin 5- or 15 mg, was performed. Primary endpoint was change from baseline in HbA1c at week 26. Secondary endpoints were change from baseline at week 26 in fasting plasma glucose (FPG), body weight (BW), systolic/diastolic blood pressure (SBP/DBP), and proportion of patients with HbA1c <7.0%. Hypotheses for the primary endpoint and FPG and BW secondary endpoints were tested in the China subpopulation.
RESULTS: At week 26, least squares mean (95% CI) change from baseline HbA1c was significantly greater with ertugliflozin 5- and 15 mg versus placebo: -1.0% (-1.1, -0.9), -0.9% (-1.0, -0.8), -0.2% (-0.3, -0.1), respectively. Ertugliflozin significantly reduced FPG, BW and SBP. Reductions in DBP with ertugliflozin were not significant. At week 26, 16.2%, 38.2% and 40.8% of patients had HbA1c <7.0% with placebo, ertugliflozin 5- and 15 mg, respectively. 59.3%, 56.5% and 53.3% of patients experienced adverse events with placebo, ertugliflozin 5- and 15 mg, respectively. Incidence of symptomatic hypoglycaemia was higher for ertugliflozin 15 mg vs placebo. Results in the China subpopulation were consistent.
CONCLUSIONS: Ertugliflozin significantly improved glycaemic control and reduced BW and SBP in Asian patients with T2DM. Ertugliflozin was generally well-tolerated. Results in the China subpopulation were consistent with the overall population. ClinicalTrials.gov: NCT02630706.
© 2019 John Wiley & Sons Ltd.

Entities:  

Keywords:  Asia; SGLT2 inhibitor; ertugliflozin; type 2 diabetes mellitus

Mesh:

Substances:

Year:  2019        PMID: 30830724     DOI: 10.1111/dom.13681

Source DB:  PubMed          Journal:  Diabetes Obes Metab        ISSN: 1462-8902            Impact factor:   6.577


  23 in total

1.  Comparative Effects of Sodium-Glucose Cotransporter 2 Inhibitors on Serum Electrolyte Levels in Patients with Type 2 Diabetes: A Pairwise and Network Meta-Analysis of Randomized Controlled Trials.

Authors:  Jingjing Zhang; Yonghong Huan; Mark Leibensperger; Bojung Seo; Yiqing Song
Journal:  Kidney360       Date:  2022-01-19

Review 2.  Effect of ertugliflozin on glycemic levels, blood pressure and body weight of patients with type 2 diabetes mellitus: a systematic review and meta-analysis.

Authors:  Maryam Zaman; Roha Saeed Memon; Arooba Amjad; Tehlil Rizwan; Jai Kumar; Ibtehaj Ul Haque; Syed Saad Ali; Lin Li; Muhammad Shariq Usman
Journal:  J Diabetes Metab Disord       Date:  2020-09-03

Review 3.  End-to-end application of model-informed drug development for ertugliflozin, a novel sodium-glucose cotransporter 2 inhibitor.

Authors:  Daryl J Fediuk; Gianluca Nucci; Vikas K Dawra; Ernesto Callegari; Susan Zhou; Cynthia J Musante; Yali Liang; Kevin Sweeney; Vaishali Sahasrabudhe
Journal:  CPT Pharmacometrics Syst Pharmacol       Date:  2021-05-15

4.  Pharmacokinetic Properties of Single and Multiple Doses of Ertugliflozin, a Selective Inhibitor of SGLT2, in Healthy Chinese Subjects.

Authors:  Yinhua Li; Yuting Mu; Haihong Shi; Yali Liang; Zeyuan Liu; Kyle Matschke; Anne Hickman; Rajesh Krishna; Vaishali Sahasrabudhe
Journal:  Clin Pharmacol Drug Dev       Date:  2019-04-01

5.  Risk of any hypoglycaemia with newer antihyperglycaemic agents in patients with type 2 diabetes: A systematic review and meta-analysis.

Authors:  Sanaz Kamalinia; Robert G Josse; Patrick J Donio; Lindsay Leduc; Baiju R Shah; Sheldon W Tobe
Journal:  Endocrinol Diabetes Metab       Date:  2019-11-13

6.  Bioequivalence of Metformin in Ertugliflozin/Metformin Fixed-Dose Combination Tablets to Canadian-Sourced Metformin Coadministered With Ertugliflozin Under Fasted and Fed States.

Authors:  Vikas Kumar Dawra; Kathleen Pelletier; Kyle Matschke; Haihong Shi; Anne Hickman; Susan Zhou; Rajesh Krishna; Vaishali Sahasrabudhe
Journal:  Clin Pharmacol Drug Dev       Date:  2020-11-02

7.  SGLT-2i and Risk of Malignancy in Type 2 Diabetes: A Meta-Analysis of Randomized Controlled Trials.

Authors:  Nanjing Shi; Yetan Shi; Jingsi Xu; Yuexiu Si; Tong Yang; Mengting Zhang; Derry Minyao Ng; Xiangyuan Li; Fei Xie
Journal:  Front Public Health       Date:  2021-06-07

8.  Population Pharmacokinetic Analyses of Ertugliflozin in Select Ethnic Populations.

Authors:  Daryl J Fediuk; Vaishali Sahasrabudhe; Vikas Kumar Dawra; Susan Zhou; Kevin Sweeney
Journal:  Clin Pharmacol Drug Dev       Date:  2021-07-02

9.  Effect of Hemoglobin A1c Reduction or Weight Reduction on Blood Pressure in Glucagon-Like Peptide-1 Receptor Agonist and Sodium-Glucose Cotransporter-2 Inhibitor Treatment in Type 2 Diabetes Mellitus: A Meta-Analysis.

Authors:  Mengdie Hu; Xiaoling Cai; Wenjia Yang; Simin Zhang; Lin Nie; Linong Ji
Journal:  J Am Heart Assoc       Date:  2020-03-30       Impact factor: 5.501

10.  Efficacy and safety of ertugliflozin in East/Southeast Asian patients with type 2 diabetes mellitus.

Authors:  Jie Liu; Shrita Patel; Nilo B Cater; Larry Wu; Susan Huyck; Steven G Terra; Anne Hickman; Amanda Darekar; Annpey Pong; Ira Gantz
Journal:  Diabetes Obes Metab       Date:  2020-01-03       Impact factor: 6.577

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