Literature DB >> 30679329

The Bruton tyrosine kinase inhibitor zanubrutinib (BGB-3111) demonstrated synergies with other anti-lymphoma targeted agents.

Chiara Tarantelli1, Lu Zhang2,3, Elisabetta Curti1, Eugenio Gaudio1, Filippo Spriano1, Valdemar Priebe1, Luciano Cascione1, Alberto J Arribas1, Emanuele Zucca2, Davide Rossi1,2, Anastasios Stathis2, Francesco Bertoni4.   

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Year:  2019        PMID: 30679329      PMCID: PMC6601092          DOI: 10.3324/haematol.2018.214759

Source DB:  PubMed          Journal:  Haematologica        ISSN: 0390-6078            Impact factor:   9.941


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  5 in total

1.  The Bruton tyrosine kinase inhibitor CC-292 shows activity in mantle cell lymphoma and synergizes with lenalidomide and NIK inhibitors depending on nuclear factor-κB mutational status.

Authors:  Anna Vidal-Crespo; Vanina Rodriguez; Alba Matas-Cespedes; Eriong Lee; Alfredo Rivas-Delgado; Eva Giné; Alba Navarro; Sílvia Beà; Elias Campo; Armando López-Guillermo; Monica Lopez-Guerra; Gaël Roué; Dolors Colomer; Patricia Pérez-Galán
Journal:  Haematologica       Date:  2017-08-24       Impact factor: 9.941

2.  PQR309 Is a Novel Dual PI3K/mTOR Inhibitor with Preclinical Antitumor Activity in Lymphomas as a Single Agent and in Combination Therapy.

Authors:  Chiara Tarantelli; Eugenio Gaudio; Alberto J Arribas; Ivo Kwee; Petra Hillmann; Andrea Rinaldi; Luciano Cascione; Filippo Spriano; Elena Bernasconi; Francesca Guidetti; Laura Carrassa; Roberta Bordone Pittau; Florent Beaufils; Reto Ritschard; Denise Rageot; Alexander Sele; Barbara Dossena; Francesca Maria Rossi; Antonella Zucchetto; Monica Taborelli; Valter Gattei; Davide Rossi; Anastasios Stathis; Georg Stussi; Massimo Broggini; Matthias P Wymann; Andreas Wicki; Emanuele Zucca; Vladimir Cmiljanovic; Doriano Fabbro; Francesco Bertoni
Journal:  Clin Cancer Res       Date:  2017-10-24       Impact factor: 12.531

3.  Acalabrutinib (ACP-196) in Relapsed Chronic Lymphocytic Leukemia.

Authors:  John C Byrd; Bonnie Harrington; Susan O'Brien; Jeffrey A Jones; Anna Schuh; Steve Devereux; Jorge Chaves; William G Wierda; Farrukh T Awan; Jennifer R Brown; Peter Hillmen; Deborah M Stephens; Paolo Ghia; Jacqueline C Barrientos; John M Pagel; Jennifer Woyach; Dave Johnson; Jane Huang; Xiaolin Wang; Allard Kaptein; Brian J Lannutti; Todd Covey; Maria Fardis; Jesse McGreivy; Ahmed Hamdy; Wayne Rothbaum; Raquel Izumi; Thomas G Diacovo; Amy J Johnson; Richard R Furman
Journal:  N Engl J Med       Date:  2015-12-07       Impact factor: 91.245

4.  Acalabrutinib in relapsed or refractory mantle cell lymphoma (ACE-LY-004): a single-arm, multicentre, phase 2 trial.

Authors:  Michael Wang; Simon Rule; Pier Luigi Zinzani; Andre Goy; Olivier Casasnovas; Stephen D Smith; Gandhi Damaj; Jeanette Doorduijn; Thierry Lamy; Franck Morschhauser; Carlos Panizo; Bijal Shah; Andrew Davies; Richard Eek; Jehan Dupuis; Eric Jacobsen; Arnon P Kater; Steven Le Gouill; Lucie Oberic; Taduesz Robak; Todd Covey; Richa Dua; Ahmed Hamdy; Xin Huang; Raquel Izumi; Priti Patel; Wayne Rothbaum; J Greg Slatter; Wojciech Jurczak
Journal:  Lancet       Date:  2017-12-11       Impact factor: 79.321

Review 5.  Role of Bruton's tyrosine kinase in B cells and malignancies.

Authors:  Simar Pal Singh; Floris Dammeijer; Rudi W Hendriks
Journal:  Mol Cancer       Date:  2018-02-19       Impact factor: 27.401

  5 in total
  4 in total

Review 1.  Zanubrutinib: First Approval.

Authors:  Yahiya Y Syed
Journal:  Drugs       Date:  2020-01       Impact factor: 9.546

Review 2.  Recent Research Progress of Chiral Small Molecular Antitumor-Targeted Drugs Approved by the FDA From 2011 to 2019.

Authors:  Xuetong Chu; Yizhi Bu; Xiaoping Yang
Journal:  Front Oncol       Date:  2021-12-17       Impact factor: 6.244

3.  Preliminary Evaluation of Zanubrutinib-Containing Regimens in DLBCL and the Cerebrospinal Fluid Distribution of Zanubrutinib: A 13-Case Series.

Authors:  Yan Zhang; Yanan Li; Zhe Zhuang; Wei Wang; Chong Wei; Danqing Zhao; Daobin Zhou; Wei Zhang
Journal:  Front Oncol       Date:  2021-12-24       Impact factor: 6.244

Review 4.  Regulation of B-Cell Receptor Signaling and Its Therapeutic Relevance in Aggressive B-Cell Lymphomas.

Authors:  Núria Profitós-Pelejà; Juliana Carvalho Santos; Ana Marín-Niebla; Gaël Roué; Marcelo Lima Ribeiro
Journal:  Cancers (Basel)       Date:  2022-02-09       Impact factor: 6.639

  4 in total

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