Literature DB >> 30638399

A Phase II study of the safety and efficacy of lenvatinib in patients with advanced thyroid cancer.

Shunji Takahashi1, Naomi Kiyota2, Tomoko Yamazaki3, Naoko Chayahara2, Kenji Nakano1, Lina Inagaki1, Kazuhisa Toda4, Tomohiro Enokida5, Hironobu Minami2, Yoshinori Imamura2, Naoki Fukuda1, Tatsuya Sasaki6, Takuya Suzuki6, Hiroki Ikezawa6, Corina E Dutcus7, Makoto Tahara5.   

Abstract

AIM: To investigate the safety and efficacy of lenvatinib in advanced thyroid cancer. PATIENTS/
METHODS: In this Phase II study, 51 Japanese patients with radioiodine-refractory differentiated thyroid cancer (RR-DTC), medullary thyroid cancer (MTC) or anaplastic thyroid cancer (ATC) received once-daily lenvatinib 24 mg. The primary end point was safety.
RESULTS: All patients experienced ≥1 adverse event (AE); only one patient experienced an AE leading to discontinuation. The most common any-grade AEs were hypertension, decreased appetite, palmar-plantar erythrodysesthesia, fatigue and proteinuria. Response rates for RR-DTC: 68%; MTC: 22%; ATC: 24%. Median progression-free survival for RR-DTC: 25.8 months; MTC: 9.2 months; ATC: 7.4 months.
CONCLUSION: Lenvatinib demonstrated a manageable safety profile, proven antitumor activity in RR-DTC and promising efficacy in MTC and ATC. CLINICAL TRIAL REGISTRATION: clinicaltrials.gov NCT01728623.

Entities:  

Keywords:  anaplastic; lenvatinib; medullary; radioiodine-refractory differentiated thyroid cancer; thyroid carcinoma

Mesh:

Substances:

Year:  2019        PMID: 30638399     DOI: 10.2217/fon-2018-0557

Source DB:  PubMed          Journal:  Future Oncol        ISSN: 1479-6694            Impact factor:   3.404


  34 in total

Review 1.  Novel treatments for anaplastic thyroid carcinoma.

Authors:  Silvia Martina Ferrari; Giusy Elia; Francesca Ragusa; Ilaria Ruffilli; Concettina La Motta; Sabrina Rosaria Paparo; Armando Patrizio; Roberto Vita; Salvatore Benvenga; Gabriele Materazzi; Poupak Fallahi; Alessandro Antonelli
Journal:  Gland Surg       Date:  2020-01

2.  Prognostic Significance of Neutrophil-to-Lymphocyte Ratio in Differentiated Thyroid Carcinoma Having Distant Metastasis: A Comparison With Thyroglobulin-doubling Rate and Tumor Volume-doubling Rate.

Authors:  Yasuhiro Ito; Naoyoshi Onoda; Minoru Kihara; Akihiro Miya; Akira Miyauchi
Journal:  In Vivo       Date:  2021 Mar-Apr       Impact factor: 2.155

3.  Effect of Kinase Inhibitors on the Technetium-99m Uptake into Thyroid Carcinoma Cells In Vitro.

Authors:  Anna Anschlag; Brandon H Greene; Lorianna KÖnneker; Markus Luster; James Nagarajah; Sabine WÄchter; Annette Wunderlich; Andreas Pfestroff
Journal:  In Vivo       Date:  2021 Mar-Apr       Impact factor: 2.155

Review 4.  Immunotherapy for advanced thyroid cancers - rationale, current advances and future strategies.

Authors:  Jena D French
Journal:  Nat Rev Endocrinol       Date:  2020-08-24       Impact factor: 43.330

5.  Neutrophil-to-Lymphocyte Ratio as a Prognostic Marker for Anaplastic Thyroid Cancer Treated With Lenvatinib.

Authors:  Naoki Fukuda; Kazuhisa Toda; Y U Fujiwara; Xiaofei Wang; Akihiro Ohmoto; Tetsuya Urasaki; Naomi Hayashi; Yasuyoshi Sato; Kenji Nakano; Mayu Yunokawa; Makiko Ono; Junichi Tomomatsu; Hiroki Mitani; Shunji Takahashi
Journal:  In Vivo       Date:  2020 Sep-Oct       Impact factor: 2.155

6.  Inflammatory biomarkers and dynamics of neutrophil-to-lymphocyte ratio in lenvatinib treatment for anaplastic thyroid carcinoma.

Authors:  Haruhiko Yamazaki; Hiroyuki Iwasaki; Nobuyasu Suganuma; Soji Toda; Katsuhiko Masudo; Hirotaka Nakayama; Yasushi Rino; Munetaka Masuda
Journal:  Gland Surg       Date:  2021-03

7.  Lenvatinib as a salvage therapy for advanced metastatic medullary thyroid cancer.

Authors:  A Matrone; A Prete; A Nervo; A Ragni; L Agate; E Molinaro; C Giani; L Valerio; E Minaldi; A Piovesan; R Elisei
Journal:  J Endocrinol Invest       Date:  2021-02-17       Impact factor: 4.256

Review 8.  Anaplastic Thyroid Carcinoma: Current Issues in Genomics and Therapeutics.

Authors:  Ichiro Abe; Alfred King-Yin Lam
Journal:  Curr Oncol Rep       Date:  2021-02-13       Impact factor: 5.075

9.  2021 American Thyroid Association Guidelines for Management of Patients with Anaplastic Thyroid Cancer.

Authors:  Keith C Bible; Electron Kebebew; James Brierley; Juan P Brito; Maria E Cabanillas; Thomas J Clark; Antonio Di Cristofano; Robert Foote; Thomas Giordano; Jan Kasperbauer; Kate Newbold; Yuri E Nikiforov; Gregory Randolph; M Sara Rosenthal; Anna M Sawka; Manisha Shah; Ashok Shaha; Robert Smallridge; Carol K Wong-Clark
Journal:  Thyroid       Date:  2021-03       Impact factor: 6.568

Review 10.  Clinical Indications for Treatment with Multi-Kinase Inhibitors in Patients with Radioiodine-Refractory Differentiated Thyroid Cancer.

Authors:  Naoki Fukuda; Shunji Takahashi
Journal:  Cancers (Basel)       Date:  2021-05-10       Impact factor: 6.639

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