Literature DB >> 30638082

Pathophysiology of idiopathic gastroparesis and implications for therapy.

Mattis Bekkelund1,2, Dag A Sangnes2,3,4, Jan Gunnar Hatlebakk2,3,4, Lars Aabakken1,5.   

Abstract

OBJECTIVES: Idiopathic gastroparesis is a gastric motility disorder characterized by chronic upper gastrointestinal symptoms and delayed gastric emptying without an identifiable underlying condition. This review summarizes recent understanding of the pathophysiology and treatment of idiopathic gastroparesis.
MATERIALS AND METHODS: Structured literature search in the PubMed, Embase and ClinicalTrials.gov databases.
RESULTS: Idiopathic gastroparesis involves several alterations in gastric motility and sensation, including delayed gastric emptying, altered myoelectrical activity, impaired fundic accommodation, visceral hypersensitivity and disturbances in antropyloroduodenal motility and coordination. Multiple cellular changes have been identified, including depletion of interstitial cells of Cajal (ICC) and enteric nerves, as well as stromal fibrosis. The underlying cause of these changes is not fully understood but may be an immune imbalance, including loss of anti-inflammatory heme-oxygenase-1 positive (HO-1) macrophages. There is currently no causal therapy for idiopathic gastroparesis. The treatment ladder consists of dietary measures, prokinetic and antiemetic medications, and varying surgical or endoscopic interventions, including promising pyloric therapies. There are ongoing trials with several novel medications, raising hopes for future treatment.
CONCLUSIONS: Patients with idiopathic gastroparesis present several pathophysiological alterations in the stomach, where depletion of ICC is of special importance. Treatment is currently focused on alleviating symptoms through dietary adjustments, medication or surgical or endoscopic interventions.

Entities:  

Keywords:  Gastroparesis; gastric accommodation; gastric dysrhythmia; gastric emptying; idiopathic gastroparesis; interstitial cells of Cajal

Mesh:

Substances:

Year:  2019        PMID: 30638082     DOI: 10.1080/00365521.2018.1558280

Source DB:  PubMed          Journal:  Scand J Gastroenterol        ISSN: 0036-5521            Impact factor:   2.423


  8 in total

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Authors:  Bin Liu; Jun Dong; Shasha Wang; Haining Yu; Zhongchao Li; Pengfei Sun; Lei Zhao
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4.  Gastroparesis Symptoms Associated with Intestinal Hypomotility: An Explorative Study Using Wireless Motility Capsule.

Authors:  Mattis Bekkelund; Dag A Sangnes; Eirik Søfteland; Lars Aabakken; Martin Biermann; Elisabeth K Steinsvik; Trygve Hausken; Georg Dimcevski; Jan Gunnar Hatlebakk
Journal:  Clin Exp Gastroenterol       Date:  2021-04-28

5.  Non-Clinical Safety Pharmacology Evaluations of Trazpiroben (TAK-906), a Novel Dopamine D2/D3 Selective Receptor Antagonist for the Management of Gastroparesis.

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6.  Evaluating the Safety, Tolerability, and Disposition of Trazpiroben, a D2 /D3 Receptor Antagonist: Phase I Single- and Multiple-Ascending Dose Studies in Healthy Japanese Participants.

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7.  A Clinical Randomized Controlled Trial of Acupuncture Treatment of Gastroparesis Using Different Acupoints.

Authors:  Wu Xuefen; Li Ping; Liu Li; Chen Xiaoli; Zenghui Yue
Journal:  Pain Res Manag       Date:  2020-04-25       Impact factor: 3.037

8.  Safety, Pharmacokinetics, and Pharmacodynamics of Trazpiroben (TAK-906), a Novel Selective D2 /D3 Receptor Antagonist: A Phase 1 Randomized, Placebo-Controlled Single- and Multiple-Dose Escalation Study in Healthy Participants.

Authors:  Roger L Whiting; Borje Darpo; Chunlin Chen; Margaret Fletcher; Dan Combs; Hongqi Xue; Randall R Stoltz
Journal:  Clin Pharmacol Drug Dev       Date:  2021-01-18
  8 in total

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