Literature DB >> 30612205

NS5A-P32 deletion as a factor involved in virologic failure in patients receiving glecaprevir and pibrentasvir.

Hayato Uemura1, Yoshihito Uchida1, Jun-Ichi Kouyama1, Kayoko Naiki1, Shohei Tsuji1, Kayoko Sugawara1, Masamitsu Nakao1, Daisuke Motoya1, Nobuaki Nakayama1, Yukinori Imai1, Tomoaki Tomiya1, Satoshi Mochida2.   

Abstract

BACKGROUND: This study sought to clarify the factors involved in virologic failure in patients with HCV receiving retreatment with glecaprevir/pibrentasvir (GLE/PIB) in real-world practice.
METHODS: Forty-two patients who had previously received direct-acting antivirals (DAAs) therapies consisting of 35, 3, 3, and 1 patient(s) with genotype (GT)-1b, GT-2a, GT-2b, and GT-3b HCV, respectively, received GLE/PIB for 12 weeks. Resistance-associated substitutions (RASs) at baseline were evaluated, and the dynamics of NS5A-RASs were assessed by deep sequencing in patients showing virologic failure.
RESULTS: Baseline NS5A-RASs were found in all the patients with GT-1b HCV including 16 patients with NS3-RASs. In contrast, both NS5A-RASs and NS3-RASs were absent in 3 and 2 patients with GT-2a and GT-2b HCV, respectively. Virologic failure occurred in 3 patients with GT-1b HCV with NS5A-P32del, while a sustained virologic response (SVR) was achieved in the remaining 39 patients including those with GT-1b HCV carrying NS5A-L31V + Y93H and NS5A-A92K. Virologic failure even occurred in a patient in whom the NS5A-P32del HCV strains had become undetectable by direct sequencing, and the percentage of such strains relative to the total HCV strains was 10%, as determined by deep sequencing. In the other patient with GT-1b HCV with NS5A-P32del, NS3-A156A/V/S were found at 4 weeks after GLE/PIB therapy, but had disappeared at 11 weeks, as determined by direct sequencing.
CONCLUSIONS: GLE/PIB was effective for patients with HCV who failed to achieve an SVR after prior DAA therapies except in those with GT-1b HCV carrying NS5A-P32del even when such strains became undetectable by direct sequencing.

Entities:  

Keywords:  DAA retreatment; Glecaprevir; NS5A-P32 deletion; Pibrentasvir

Mesh:

Substances:

Year:  2019        PMID: 30612205     DOI: 10.1007/s00535-018-01543-9

Source DB:  PubMed          Journal:  J Gastroenterol        ISSN: 0944-1174            Impact factor:   6.772


  26 in total

1.  Chronic hepatitis caused by hepatitis C virus showing a discrepancy between serogroup and genotype because of intergenotypic 2b/1b recombination: A pitfall in antiviral therapy with direct-acting antivirals.

Authors:  Hayato Kurata; Yoshihito Uchida; Jun-Ichi Kouyama; Kayoko Naiki; Manabu Nakazawa; Satsuki Ando; Masamitsu Nakao; Daisuke Motoya; Kayoko Sugawara; Mie Inao; Yukinori Imai; Nobuaki Nakayama; Tomoaki Tomiya; Satoshi Mochida
Journal:  Hepatol Res       Date:  2017-09-25       Impact factor: 4.288

2.  Sofosbuvir-velpatasvir with ribavirin for 24 weeks in hepatitis C virus patients previously treated with a direct-acting antiviral regimen.

Authors:  Edward J Gane; Mitchell L Shiffman; Kyle Etzkorn; Giuseppe Morelli; Catherine A M Stedman; Mitchell N Davis; Federico Hinestrosa; Hadas Dvory-Sobol; K C Huang; Anu Osinusi; John McNally; Diana M Brainard; John G McHutchison; Alex J Thompson; Mark S Sulkowski
Journal:  Hepatology       Date:  2017-08-26       Impact factor: 17.425

3.  Development of rare resistance-associated variants that are extremely tolerant against NS5A inhibitors during daclatasvir/asunaprevir therapy by a two-hit mechanism.

Authors:  Yoshihito Uchida; Jun-Ichi Kouyama; Kayoko Naiki; Kayoko Sugawara; Mie Inao; Yukinori Imai; Nobuaki Nakayama; Satoshi Mochida
Journal:  Hepatol Res       Date:  2016-03-30       Impact factor: 4.288

4.  In vitro and in vivo antiviral activity and resistance profile of ombitasvir, an inhibitor of hepatitis C virus NS5A.

Authors:  Preethi Krishnan; Jill Beyer; Neeta Mistry; Gennadiy Koev; Thomas Reisch; David DeGoey; Warren Kati; Andrew Campbell; Laura Williams; Wangang Xie; Carolyn Setze; Akhteruzzaman Molla; Christine Collins; Tami Pilot-Matias
Journal:  Antimicrob Agents Chemother       Date:  2014-12-01       Impact factor: 5.191

5.  Real-world efficacy of glecaprevir plus pibrentasvir for chronic hepatitis C patient with previous direct-acting antiviral therapy failures.

Authors:  Mitsutaka Osawa; Michio Imamura; Yuji Teraoka; Takuro Uchida; Kei Morio; Hatsue Fujino; Takashi Nakahara; Atsushi Ono; Eisuke Murakami; Tomokazu Kawaoka; Daiki Miki; Masataka Tsuge; Akira Hiramatsu; Hiroshi Aikata; C Nelson Hayes; Kazuaki Chayama
Journal:  J Gastroenterol       Date:  2018-10-17       Impact factor: 7.527

6.  Prevalence of NS5A resistance associated variants in NS5A inhibitor treatment failures and an effective treatment for NS5A-P32 deleted hepatitis C virus in humanized mice.

Authors:  Yuji Teraoka; Takuro Uchida; Michio Imamura; Mitsutaka Osawa; Masataka Tsuge; Hiromi Abe-Chayama; C Nelson Hayes; Grace Naswa Makokha; Hiroshi Aikata; Daiki Miki; Hidenori Ochi; Yuji Ishida; Chise Tateno; Kazuaki Chayama
Journal:  Biochem Biophys Res Commun       Date:  2018-04-13       Impact factor: 3.575

7.  Complex Pattern of Resistance-Associated Substitutions of Hepatitis C Virus after Daclatasvir/Asunaprevir Treatment Failure.

Authors:  Jun Itakura; Masayuki Kurosaki; Chitomi Hasebe; Yukio Osaki; Kouji Joko; Hitoshi Yagisawa; Shinya Sakita; Hiroaki Okushin; Takashi Satou; Hiroyuki Hisai; Takehiko Abe; Keiji Tsuji; Takashi Tamada; Haruhiko Kobashi; Akeri Mitsuda; Yasushi Ide; Chikara Ogawa; Syotaro Tsuruta; Kouichi Takaguchi; Miyako Murakawa; Yasuhiro Asahina; Nobuyuki Enomoto; Namiki Izumi
Journal:  PLoS One       Date:  2016-10-24       Impact factor: 3.240

8.  Integrated Resistance Analysis of CERTAIN-1 and CERTAIN-2 Studies in Hepatitis C Virus-Infected Patients Receiving Glecaprevir and Pibrentasvir in Japan.

Authors:  Preethi Krishnan; Gretja Schnell; Rakesh Tripathi; Jill Beyer; Thomas Reisch; Tatyana Dekhtyar; Michelle Irvin; Wangang Xie; Bo Fu; Margaret Burroughs; Rebecca Redman; Hiromitsu Kumada; Kazuaki Chayama; Christine Collins; Tami Pilot-Matias
Journal:  Antimicrob Agents Chemother       Date:  2018-01-25       Impact factor: 5.191

9.  In Vitro Antiviral Activity and Resistance Profile of the Next-Generation Hepatitis C Virus NS3/4A Protease Inhibitor Glecaprevir.

Authors:  Teresa I Ng; Rakesh Tripathi; Thomas Reisch; Liangjun Lu; Timothy Middleton; Todd A Hopkins; Ron Pithawalla; Michelle Irvin; Tatyana Dekhtyar; Preethi Krishnan; Gretja Schnell; Jill Beyer; Keith F McDaniel; Jun Ma; Guoqiang Wang; Li-Juan Jiang; Yat Sun Or; Dale Kempf; Tami Pilot-Matias; Christine Collins
Journal:  Antimicrob Agents Chemother       Date:  2017-12-21       Impact factor: 5.191

10.  Sofosbuvir, Velpatasvir, and Voxilaprevir for Previously Treated HCV Infection.

Authors:  Marc Bourlière; Stuart C Gordon; Steven L Flamm; Curtis L Cooper; Alnoor Ramji; Myron Tong; Natarajan Ravendhran; John M Vierling; Tram T Tran; Stephen Pianko; Meena B Bansal; Victor de Lédinghen; Robert H Hyland; Luisa M Stamm; Hadas Dvory-Sobol; Evguenia Svarovskaia; Jie Zhang; K C Huang; G Mani Subramanian; Diana M Brainard; John G McHutchison; Elizabeth C Verna; Peter Buggisch; Charles S Landis; Ziad H Younes; Michael P Curry; Simone I Strasser; Eugene R Schiff; K Rajender Reddy; Michael P Manns; Kris V Kowdley; Stefan Zeuzem
Journal:  N Engl J Med       Date:  2017-06-01       Impact factor: 91.245

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  10 in total

1.  The effectiveness and safety of glecaprevir/pibrentasvir in chronic hepatitis C patients with refractory factors in the real world: a comprehensive analysis of a prospective multicenter study.

Authors:  Akito Nozaki; Masanori Atsukawa; Chisa Kondo; Hidenori Toyoda; Makoto Chuma; Makoto Nakamuta; Haruki Uojima; Koichi Takaguchi; Hiroki Ikeda; Tsunamasa Watanabe; Shintaro Ogawa; Norio Itokawa; Taeang Arai; Atsushi Hiraoka; Toru Asano; Shinichi Fujioka; Tadashi Ikegami; Toshihide Shima; Chikara Ogawa; Takehiro Akahane; Noritomo Shimada; Shinya Fukunishi; Hiroshi Abe; Akihito Tsubota; Takuya Genda; Hironao Okubo; Shigeru Mikami; Asahiro Morishita; Akio Moriya; Joji Tani; Yoshihiko Tachi; Naoki Hotta; Toru Ishikawa; Takeshi Okanoue; Yasuhito Tanaka; Takashi Kumada; Katsuhiko Iwakiri; Shin Maeda
Journal:  Hepatol Int       Date:  2020-03-03       Impact factor: 6.047

2.  Features of resistance-associated substitutions after failure of multiple direct-acting antiviral regimens for hepatitis C.

Authors:  Jun Itakura; Masayuki Kurosaki; Satoru Kakizaki; Keisuke Amano; Nobuaki Nakayama; Jun Inoue; Tetsu Endo; Hiroyuki Marusawa; Chitomi Hasebe; Kouji Joko; Shuichi Wada; Takehiro Akahane; Youhei Koushima; Chikara Ogawa; Tatsuya Kanto; Masashi Mizokami; Namiki Izumi
Journal:  JHEP Rep       Date:  2020-06-18

3.  Mutational spectrum of hepatitis C virus in patients with chronic hepatitis C determined by single molecule real-time sequencing.

Authors:  Fumiyasu Nakamura; Haruhiko Takeda; Yoshihide Ueda; Atsushi Takai; Ken Takahashi; Yuji Eso; Soichi Arasawa; Eriko Iguchi; Takahiro Shimizu; Masako Mishima; Ken Kumagai; Taiki Yamashita; Shinji Uemoto; Nobuyuki Kato; Hiroyuki Marusawa; Akihiro Sekine; Hiroshi Seno
Journal:  Sci Rep       Date:  2022-04-30       Impact factor: 4.996

Review 4.  Glecaprevir/pibrentasvir for the treatment of chronic hepatitis C: design, development, and place in therapy.

Authors:  Thomas G Cotter; Donald M Jensen
Journal:  Drug Des Devel Ther       Date:  2019-07-29       Impact factor: 4.162

Review 5.  Efficacy and Safety of Glecaprevir/Pibrentasvir in Patients with Chronic HCV Infection.

Authors:  Xiaoqing Liu; Peng Hu
Journal:  J Clin Transl Hepatol       Date:  2021-01-18

6.  Efficacy of Glecaprevir/Pibrentasvir for Real-World HCV Infected Patients in the Northern Part of Tokyo, Japan.

Authors:  Yoichiro Yamana; Tatsuo Kanda; Naoki Matsumoto; Masayuki Honda; Mariko Kumagawa; Reina Sasaki; Shini Kanezawa; Taku Mizutani; Hiroaki Yamagami; Ryota Masuzaki; Tomotaka Ishii; Kazushige Nirei; Mitsuhiko Moriyama
Journal:  J Clin Med       Date:  2021-11-26       Impact factor: 4.241

7.  Effectiveness of Glecaprevir/Pibrentasvir for Hepatitis C: Real-World Experience and Clinical Features of Retreatment Cases.

Authors:  Ayumi Sugiura; Satoru Joshita; Yuki Yamashita; Tomoo Yamazaki; Naoyuki Fujimori; Takefumi Kimura; Akihiro Matsumoto; Shuichi Wada; Hiromitsu Mori; Soichiro Shibata; Kaname Yoshizawa; Susumu Morita; Kiyoshi Furuta; Atsushi Kamijo; Akihiro Iijima; Satoko Kako; Atsushi Maruyama; Masakazu Kobayashi; Michiharu Komatsu; Makiko Matsumura; Chiharu Miyabayashi; Tetsuya Ichijo; Aki Takeuchi; Yuriko Koike; Yukio Gibo; Toshihisa Tsukadaira; Hiroyuki Inada; Yoshiyuki Nakano; Seiichi Usuda; Kendo Kiyosawa; Eiji Tanaka; Takeji Umemura
Journal:  Biomedicines       Date:  2020-04-03

8.  Single-molecular real-time deep sequencing reveals the dynamics of multi-drug resistant haplotypes and structural variations in the hepatitis C virus genome.

Authors:  Taiki Yamashita; Haruhiko Takeda; Atsushi Takai; Soichi Arasawa; Fumiyasu Nakamura; Yoichi Mashimo; Miyuki Hozan; Shigeru Ohtsuru; Hiroshi Seno; Yoshihide Ueda; Akihiro Sekine
Journal:  Sci Rep       Date:  2020-02-14       Impact factor: 4.379

9.  Insights into the unique characteristics of hepatitis C virus genotype 3 revealed by development of a robust sub-genomic DBN3a replicon.

Authors:  Joseph C Ward; Sebastian Bowyer; Shucheng Chen; Guilherme Rodrigues Fernandes Campos; Santseharay Ramirez; Jens Bukh; Mark Harris
Journal:  J Gen Virol       Date:  2020-11       Impact factor: 3.891

10.  HCV genome-wide analysis for development of efficient culture systems and unravelling of antiviral resistance in genotype 4.

Authors:  Long V Pham; Martin Schou Pedersen; Ulrik Fahnøe; Carlota Fernandez-Antunez; Daryl Humes; Kristian Schønning; Santseharay Ramirez; Jens Bukh
Journal:  Gut       Date:  2021-04-08       Impact factor: 23.059

  10 in total

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