Literature DB >> 30577988

PI3K inhibitor provides durable response in metastatic metaplastic carcinoma of the breast: A hidden gem in the BELLE-4 study.

Ming-Han Yang1, I-Chun Chen2, Yen-Shen Lu3.   

Abstract

PURPOSE: Metaplastic carcinoma of the breast (MCB) is a rare cancer characterized by the histologic presence of two or more histological cell types originating from epithelial and mesenchymal stem cells. Patients with metastatic MCB have a low response rate to conventional chemotherapy and poor survival. Optimal treatment strategies for metastatic MCB are urgently needed.
METHODS: We retrospectively reviewed a patient who had enrolled in the phase II/III seamless study, BELLE-4 (NCT01572727). The patient's response to the study drug assessed by an investigator per protocol and clinical course were examined and compared with those of the main cohorts in the BELLE-4 study.
RESULTS: Our patient exhibited metastatic MCB and received systemic chemotherapy, paclitaxel (70 mg/m2/week) and buparlisib (80 mg/day), a pan-class I phosphatidylinositol-3 kinase (PI3K) inhibitor. The optimal response was a confirmed partial response for 17 months in total. During the compassionated use program period, the tumor regrew when buparlisib was stop because of toxicity, and responded to the treatment again after resumed the buparlisib treatment. The overall survival of the patient after the development of metastatic MCB was 42 months. She experienced grade 3 hyperglycemia similar to that observed in the main cohort.
CONCLUSION: Buparlisib plus weekly paclitaxel might be a new treatment option for patients with metastatic MCB harboring a PIK3CA mutation. Additional prospective studies for investigating the efficacy of the proposed combination are warranted.
Copyright © 2018 Formosan Medical Association. Published by Elsevier B.V. All rights reserved.

Entities:  

Keywords:  BELLE-4; Buparlisib; Metaplastic breast cancer; Phosphatidylinositol 3-kinases inhibitor; Triple-negative breast cancer

Mesh:

Substances:

Year:  2018        PMID: 30577988     DOI: 10.1016/j.jfma.2018.12.004

Source DB:  PubMed          Journal:  J Formos Med Assoc        ISSN: 0929-6646            Impact factor:   3.282


  7 in total

1.  Case Reports on Metaplastic Squamous Cell Carcinoma of the Breast and Treatment Dilemma.

Authors:  Anita Pandey; Kishor Joshi; Harry Moussouris; Gardith Joseph
Journal:  Case Rep Oncol Med       Date:  2019-09-18

2.  Complete Response of Chemo-Refractory Metastatic Metaplastic Breast Cancer to Paclitaxel-Immunotherapy Combination.

Authors:  Adher D Al Sayed; Mahmoud A Elshenawy; Asma Tulbah; Taher Al-Tweigeri; Hazem Ghebeh
Journal:  Am J Case Rep       Date:  2019-11-06

Review 3.  An Update on the Molecular Pathology of Metaplastic Breast Cancer.

Authors:  Amy E McCart Reed; Emarene M Kalaw; Sunil R Lakhani
Journal:  Breast Cancer (Dove Med Press)       Date:  2021-02-26

4.  TERT promoter hotspot mutations and gene amplification in metaplastic breast cancer.

Authors:  Edaise M da Silva; Pier Selenica; Mahsa Vahdatinia; Fresia Pareja; Arnaud Da Cruz Paula; Lorenzo Ferrando; Andrea M Gazzo; Higinio Dopeso; Dara S Ross; Ariya Bakhteri; Nadeem Riaz; Sarat Chandarlapaty; Pedram Razavi; Larry Norton; Hannah Y Wen; Edi Brogi; Britta Weigelt; Hong Zhang; Jorge S Reis-Filho
Journal:  NPJ Breast Cancer       Date:  2021-04-16

5.  The role of radiotherapy in metaplastic breast cancer: a propensity score-matched analysis of the SEER database.

Authors:  Yongfeng Li; Meng Chen; Barbara Pardini; Mihnea P Dragomir; Anthony Lucci; George A Calin
Journal:  J Transl Med       Date:  2019-09-23       Impact factor: 5.531

6.  Combination of PI3K and MEK inhibitors yields durable remission in PDX models of PIK3CA-mutated metaplastic breast cancers.

Authors:  F Coussy; R El Botty; M Lavigne; C Gu; L Fuhrmann; A Briaux; L de Koning; A Dahmani; E Montaudon; L Morisset; L Huguet; L Sourd; P Painsec; S Chateau-Joubert; T Larcher; S Vacher; S Melaabi; A Vincent Salomon; E Marangoni; I Bieche
Journal:  J Hematol Oncol       Date:  2020-02-22       Impact factor: 17.388

Review 7.  A comprehensive overview of metaplastic breast cancer: clinical features and molecular aberrations.

Authors:  Tejaswini P Reddy; Roberto R Rosato; Xiaoxian Li; Stacy Moulder; Helen Piwnica-Worms; Jenny C Chang
Journal:  Breast Cancer Res       Date:  2020-11-04       Impact factor: 6.466

  7 in total

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