Literature DB >> 30547193

Low dosage of apatinib monotherapy as rescue treatment in advanced lung squamous cell carcinoma.

Da-Xiong Zeng1, Wei Lei1, Chang-Guo Wang1, Jian-An Huang1, Jun-Hong Jiang2.   

Abstract

PURPOSE: Platinum-based doublet chemotherapy and radiotherapy are the standard treatment option in advanced squamous cell carcinoma patients. However, few agents could be selected for subsequent post-second-line treatment. As a small molecule inhibitor of vascular endothelial growth factor receptor-2 tyrosine kinase, apatinib had been proved in advanced gastric cancer. Here, we showed its efficacy and safety in lung squamous cell carcinoma.
METHODS: In this retrospective study, 13 advanced lung squamous cell carcinoma patients were enrolled. They received doublet chemotherapy or docetaxel as the first-line treatment. After disease progressed, all patients were administrated apatinib monotherapy (250-425 mg/day) for second-line or fourth-line therapy.
RESULTS: After apatinib monotherapy, two patients achieved partial response, four patients achieved stable disease, and seven patients achieved progression disease. The medium PFS was 3.1 months. The median OS had not yet been reached. The objective remission rate was 15.4% (2/13). The total disease control rate was 46.2% (6/13). The main advert effects were vomiting and hypertension.
CONCLUSION: Apatinib might be an option as rescue treatment in advanced lung squamous cell carcinoma.

Entities:  

Keywords:  Apatinib; Squamous cell carcinoma; VEGFR-2

Mesh:

Substances:

Year:  2018        PMID: 30547193     DOI: 10.1007/s00280-018-3743-0

Source DB:  PubMed          Journal:  Cancer Chemother Pharmacol        ISSN: 0344-5704            Impact factor:   3.333


  5 in total

1.  Safety and Efficacy of Low-Dosage Apatinib Monotherapy in Advanced Lung Squamous-Cell Carcinoma: A Prospective Cohort Study.

Authors:  Qian Geng; Hua Shen; Wenyu Zhu; Yingzhi Lu; Mengjie Wang; Hua Jiang; Dongqing Li
Journal:  Onco Targets Ther       Date:  2020-11-10       Impact factor: 4.147

2.  Safety and effectiveness of apatinib in patients with previously treated metastatic gastric cancer: a sub-analysis from the real-world study of apatinib for gastric cancer treatment (AHEAD-G202).

Authors:  Xiang Wang; Junyan Yu; Mudan Yang; Likun Liu; Jinghua Gao; Yuchuan Ren; Ruixing Zhang; Diansheng Zhong; Nan Du; Zhanzhao Fu; Junmei Jia; Qingshan Li; Jianfeng Diao; Junping Zhang; Jun Guo; Xiaomei Li; Xiang Song; Yan Zhang; Zhonghe Yu; Liwen Ma; Zaiwen Fan; Zheng Liu; Guozhong Li; Feng Liang; Huaqing Wang; Yunge Gao; Ping Yang; Chunmei Bai; Aimin Zang; Xiubao Ren
Journal:  Am J Cancer Res       Date:  2020-03-01       Impact factor: 6.166

3.  Continuous Low-Dose Apatinib Combined With WBRT Significantly Reduces Peritumoral Edema and Enhances the Efficacy of Symptomatic Multiple Brain Metastases in NSCLC.

Authors:  Yue Ren; Shan-Bing Wang; Lin Zhou; Si-Qiao Liu; Lei-Ya Du; Ting Li; Mao-Qiong Jiang; Kai-Jian Lei; Bang-Xian Tan; Yu-Ming Jia
Journal:  Technol Cancer Res Treat       Date:  2021 Jan-Dec

4.  Efficacy and safety of low-dose apatinib in ovarian cancer patients with platinum-resistance or platinum-refractoriness: A single-center retrospective study.

Authors:  Wei Chen; Ziting Li; Zhong Zheng; Xiaohua Wu
Journal:  Cancer Med       Date:  2020-07-06       Impact factor: 4.452

5.  Apatinib ameliorates doxorubicin-induced migration and cancer stemness of osteosarcoma cells by inhibiting Sox2 via STAT3 signalling.

Authors:  Zhi C Tian; Jia Q Wang; Hong Ge
Journal:  J Orthop Translat       Date:  2019-08-07       Impact factor: 5.191

  5 in total

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