Literature DB >> 30418321

Eplerenone improves endothelial function and arterial stiffness and inhibits Rho-associated kinase activity in patients with idiopathic hyperaldosteronism: a pilot study.

Shinji Kishimoto1, Kenji Oki2, Tatsuya Maruhashi3, Masato Kajikawa4, Shogo Matsui3, Haruki Hashimoto3, Yuji Takaeko3, Yasuki Kihara3, Kazuaki Chayama5, Chikara Goto6, Yoshiki Aibara1, Farina Mohamad Yusoff1, Ayumu Nakashima1, Kensuke Noma1, James K Liao7, Yukihito Higashi1,4.   

Abstract

OBJECTIVE: Primary aldosteronism is one of the most common cause of secondary hypertension. It is well known that the incidence of cardiovascular events is higher in patients with primary aldosteronism than in patients with essential hypertension. In a previous study, we showed that aldosterone-producing adenoma is associated with vascular function and structure. The aim of this study was to evaluate the effects of eplerenone on vascular function in the macrovasculature and microvasculature, arterial stiffness and Rho-associated kinase (ROCK) activity in patients with idiopathic hyperaldosteronism (IHA).
METHODS: Vascular function, including reactive hyperemia index (RHI), flow-mediated vasodilation (FMD) and nitroglycerine-induced vasodilation (NID), arterial stiffness including brachial-ankle pulse wave velocity (baPWV) and brachial intima-media thickness (IMT) and ROCK activity in peripheral leukocytes were measured before and after 12 weeks of treatment with eplerenone in 50 patients with IHA.
RESULTS: After 12 weeks, eplerenone decreased the aldosterone renin ratio but did not alter SBP and DBP. Eplerenone treatment increased log RHI from 0.56 ± 0.25 to 0.69 ± 0.25 (P < 0.01) and NID from 12.8 ± 5.8 to 14.9 ± 6.9% (P = 0.02) and it decreased baPWV from 1540 ± 263 to 1505 ± 281 (P = 0.04) and ROCK activity from 1.20 ± 0.54 to 0.89 ± 0.42 (P < 0.01), whereas there was no significant change in FMD (increase from 4.6 ± 3.4 to 4.6 ± 3.6%, P = 0.99) or brachial IMT (decrease from 0.28 ± 0.07 to 0.28 ± 0.04 mm, P = 0.14).
CONCLUSION: Eplerenone improves microvascular endothelial function, vascular smooth muscle function, arterial stiffness and ROCK activity in patients with IHA. CLINICAL TRIAL REGISTRATION INFORMATION: URL for Clinical Trial: http://UMIN; Registration Number for Clinical Trial: UMIN000003409.

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Year:  2019        PMID: 30418321      PMCID: PMC6467648          DOI: 10.1097/HJH.0000000000001989

Source DB:  PubMed          Journal:  J Hypertens        ISSN: 0263-6352            Impact factor:   4.844


  44 in total

Review 1.  From bedside to bench to bedside: role of renin-angiotensin-aldosterone system in remodeling of resistance arteries in hypertension.

Authors:  Ernesto L Schiffrin; Rhian M Touyz
Journal:  Am J Physiol Heart Circ Physiol       Date:  2004-08       Impact factor: 4.733

2.  Possible involvement of Rho-kinase in the pathogenesis of hypertension in humans.

Authors:  A Masumoto; Y Hirooka; H Shimokawa; K Hironaga; S Setoguchi; A Takeshita
Journal:  Hypertension       Date:  2001-12-01       Impact factor: 10.190

3.  Increased expression and activity of RhoA are associated with increased DNA synthesis and reduced p27(Kip1) expression in the vasculature of hypertensive rats.

Authors:  T M Seasholtz; T Zhang; M R Morissette; A L Howes; A H Yang; J H Brown
Journal:  Circ Res       Date:  2001-09-14       Impact factor: 17.367

4.  Inhibition of rho-associated kinase results in suppression of neointimal formation of balloon-injured arteries.

Authors:  N Sawada; H Itoh; K Ueyama; J Yamashita; K Doi; T H Chun; M Inoue; K Masatsugu; T Saito; Y Fukunaga; S Sakaguchi; H Arai; N Ohno; M Komeda; K Nakao
Journal:  Circulation       Date:  2000-05-02       Impact factor: 29.690

5.  Primary aldosteronism: factors associated with normalization of blood pressure after surgery.

Authors:  A M Sawka; W F Young; G B Thompson; C S Grant; D R Farley; C Leibson; J A van Heerden
Journal:  Ann Intern Med       Date:  2001-08-21       Impact factor: 25.391

6.  Effect of nifedipine and cerivastatin on coronary endothelial function in patients with coronary artery disease: the ENCORE I Study (Evaluation of Nifedipine and Cerivastatin On Recovery of coronary Endothelial function).

Authors: 
Journal:  Circulation       Date:  2003-01-28       Impact factor: 29.690

7.  Impaired endothelium-dependent flow-mediated vasodilation in hypertensive subjects with hyperaldosteronism.

Authors:  Mari K Nishizaka; M Amin Zaman; Sharon A Green; Kerry Y Renfroe; David A Calhoun
Journal:  Circulation       Date:  2004-06-01       Impact factor: 29.690

8.  Preferential stiffening of central over peripheral arteries in type 2 diabetes.

Authors:  Eiji Kimoto; Tetsuo Shoji; Kayo Shinohara; Masaaki Inaba; Yasuhisa Okuno; Takami Miki; Hidenori Koyama; Masanori Emoto; Yoshiki Nishizawa
Journal:  Diabetes       Date:  2003-02       Impact factor: 9.461

9.  Aldosterone administration to mice stimulates macrophage NADPH oxidase and increases atherosclerosis development: a possible role for angiotensin-converting enzyme and the receptors for angiotensin II and aldosterone.

Authors:  Shlomo Keidar; Marielle Kaplan; Elsa Pavlotzky; Raymond Coleman; Tony Hayek; Shadi Hamoud; Michael Aviram
Journal:  Circulation       Date:  2004-05-03       Impact factor: 29.690

10.  Rho/Rho kinase and phosphoinositide 3-kinase are parallel pathways in the development of spontaneous arterial tone in deoxycorticosterone acetate-salt hypertension.

Authors:  Erica A Wehrwein; Carrie A Northcott; Robert D Loberg; Stephanie W Watts
Journal:  J Pharmacol Exp Ther       Date:  2004-02-24       Impact factor: 4.030

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  2 in total

Review 1.  Endothelial Dysfunction in Primary Aldosteronism.

Authors:  Zheng-Wei Chen; Cheng-Hsuan Tsai; Chien-Ting Pan; Chia-Hung Chou; Che-Wei Liao; Chi-Sheng Hung; Vin-Cent Wu; Yen-Hung Lin
Journal:  Int J Mol Sci       Date:  2019-10-21       Impact factor: 5.923

2.  Relationship between plasma aldosterone levels and arterial stiffness parameters in hypertensive patients with subclinical vascular damage.

Authors:  L Petramala; A Concistrè; M Mezzadri; F Sarlo; F Circosta; M Schina; M Soldini; G Iannucci; C Letizia
Journal:  Int J Cardiol Cardiovasc Risk Prev       Date:  2022-06-06
  2 in total

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