Literature DB >> 30413631

Safety, tolerability, and efficacy of fluoxetine as an antiviral for acute flaccid myelitis.

Kevin Messacar1, Stefan Sillau2, Sarah E Hopkins2, Catherine Otten2, Molly Wilson-Murphy2, Brian Wong2, Jonathan D Santoro2, Andrew Treister2, Harlori K Bains2, Alcy Torres2, Luke Zabrocki2, Julia R Glanternik2, Amanda L Hurst2, Jan A Martin2, Teri Schreiner2, Naila Makhani2, Roberta L DeBiasi2, Michael C Kruer2, Adriana H Tremoulet2, Keith Van Haren2, Jay Desai2, Leslie A Benson2, Mark P Gorman2, Mark J Abzug2, Kenneth L Tyler2, Samuel R Dominguez2.   

Abstract

OBJECTIVE: To determine the safety, tolerability, and efficacy of fluoxetine for proven or presumptive enterovirus (EV) D68-associated acute flaccid myelitis (AFM).
METHODS: A multicenter cohort study of US patients with AFM in 2015-2016 compared serious adverse events (SAEs), adverse effects, and outcomes between fluoxetine-treated patients and untreated controls. Fluoxetine was administered at the discretion of treating providers with data gathered retrospectively. The primary outcome was change in summative limb strength score (SLSS; sum of Medical Research Council strength in all 4 limbs, ranging from 20 [normal strength] to 0 [complete quadriparesis]) between initial examination and latest follow-up, with increased SLSS reflecting improvement and decreased SLSS reflecting worsened strength.
RESULTS: Fifty-six patients with AFM from 12 centers met study criteria. Among 30 patients exposed to fluoxetine, no SAEs were reported and adverse effect rates were similar to unexposed patients (47% vs 65%, p = 0.16). The 28 patients treated with >1 dose of fluoxetine were more likely to have EV-D68 identified (57.1% vs 14.3%, p < 0.001). Their SLSS was similar at initial examination (mean SLSS 12.9 vs 14.3, p = 0.31) but lower at nadir (mean SLSS 9.25 vs 12.82, p = 0.02) and latest follow-up (mean SLSS 12.5 vs 16.4, p = 0.005) compared with the 28 patients receiving 1 (n = 2) or no (n = 26) doses. In propensity-adjusted analysis, SLSS from initial examination to latest follow-up decreased by 0.2 (95% confidence interval [CI] -1.8 to +1.4) in fluoxetine-treated patients and increased by 2.5 (95% CI +0.7 to +4.4) in untreated patients (p = 0.015).
CONCLUSION: Fluoxetine was well-tolerated. Fluoxetine was preferentially given to patients with AFM with EV-D68 identified and more severe paralysis at nadir, who ultimately had poorer long-term outcomes. CLASSIFICATION OF EVIDENCE: This study provides Class IV evidence that for patients with EV-D68-associated AFM, fluoxetine is well-tolerated and not associated with improved neurologic outcomes.
© 2018 American Academy of Neurology.

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Year:  2018        PMID: 30413631      PMCID: PMC6512883          DOI: 10.1212/WNL.0000000000006670

Source DB:  PubMed          Journal:  Neurology        ISSN: 0028-3878            Impact factor:   9.910


  22 in total

1.  Enterovirus 71 infection-associated acute flaccid paralysis: a case series of long-term neurologic follow-up.

Authors:  Hsiu-Fen Lee; Ching-Shiang Chi
Journal:  J Child Neurol       Date:  2014-01-21       Impact factor: 1.987

2.  Treatment of Chronic Enterovirus Encephalitis With Fluoxetine in a Patient With X-Linked Agammaglobulinemia.

Authors:  Jacqueline Gofshteyn; Ana María Cárdenas; David Bearden
Journal:  Pediatr Neurol       Date:  2016-06-25       Impact factor: 3.372

3.  Fluoxetine pharmacokinetics in pediatric patients.

Authors:  Timothy E Wilens; Louise Cohen; Joseph Biederman; Annah Abrams; Debarah Neft; Nagy Faird; Vikram Sinha
Journal:  J Clin Psychopharmacol       Date:  2002-12       Impact factor: 3.153

4.  Rationale for the evaluation of fluoxetine in the treatment of enterovirus D68-associated acute flaccid myelitis.

Authors:  Kenneth L Tyler
Journal:  JAMA Neurol       Date:  2015-05       Impact factor: 18.302

5.  Selective serotonin reuptake inhibitor fluoxetine inhibits replication of human enteroviruses B and D by targeting viral protein 2C.

Authors:  Rachel Ulferts; Lonneke van der Linden; Hendrik Jan Thibaut; Kjerstin H W Lanke; Pieter Leyssen; Bruno Coutard; Armando M De Palma; Bruno Canard; Johan Neyts; Frank J M van Kuppeveld
Journal:  Antimicrob Agents Chemother       Date:  2013-01-18       Impact factor: 5.191

6.  Susceptibilities of enterovirus D68, enterovirus 71, and rhinovirus 87 strains to various antiviral compounds.

Authors:  Donald F Smee; W Joseph Evans; K C Nicolaou; E Bart Tarbet; Craig W Day
Journal:  Antiviral Res       Date:  2016-04-07       Impact factor: 5.970

Review 7.  Acute flaccid myelitis: A clinical review of US cases 2012-2015.

Authors:  Kevin Messacar; Teri L Schreiner; Keith Van Haren; Michele Yang; Carol A Glaser; Kenneth L Tyler; Samuel R Dominguez
Journal:  Ann Neurol       Date:  2016-08-04       Impact factor: 10.422

8.  Evaluating Treatment Efficacy in a Mouse Model of Enterovirus D68-Associated Paralytic Myelitis.

Authors:  Alison M Hixon; Penny Clarke; Kenneth L Tyler
Journal:  J Infect Dis       Date:  2017-12-05       Impact factor: 5.226

9.  Acute Flaccid Myelitis in the United States, August-December 2014: Results of Nationwide Surveillance.

Authors:  James J Sejvar; Adriana S Lopez; Margaret M Cortese; Eyal Leshem; Daniel M Pastula; Lisa Miller; Carol Glaser; Anita Kambhampati; Kayoko Shioda; Negar Aliabadi; Marc Fischer; Nicole Gregoricus; Robert Lanciotti; W Allan Nix; Senthilkumar K Sakthivel; D Scott Schmid; Jane F Seward; Suxiang Tong; M Steven Oberste; Mark Pallansch; Daniel Feikin
Journal:  Clin Infect Dis       Date:  2016-06-17       Impact factor: 9.079

Review 10.  The association between acute flaccid myelitis (AFM) and Enterovirus D68 (EV-D68) - what is the evidence for causation?

Authors:  Amalie Dyda; Sacha Stelzer-Braid; Dillon Adam; Abrar A Chughtai; C Raina MacIntyre
Journal:  Euro Surveill       Date:  2018-01
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  16 in total

1.  Enterovirus D68 Antivirals: Past, Present, and Future.

Authors:  Yanmei Hu; Rami Musharrafieh; Madeleine Zheng; Jun Wang
Journal:  ACS Infect Dis       Date:  2020-05-14       Impact factor: 5.084

2.  Validating Enterovirus D68-2Apro as an Antiviral Drug Target and the Discovery of Telaprevir as a Potent D68-2Apro Inhibitor.

Authors:  Rami Musharrafieh; Chunlong Ma; Jiantao Zhang; Yanmei Hu; Jessica M Diesing; Michael T Marty; Jun Wang
Journal:  J Virol       Date:  2019-03-21       Impact factor: 5.103

3.  A Novel Capsid Binding Inhibitor Displays Potent Antiviral Activity against Enterovirus D68.

Authors:  Chunlong Ma; Yanmei Hu; Jiantao Zhang; Rami Musharrafieh; Jun Wang
Journal:  ACS Infect Dis       Date:  2019-09-18       Impact factor: 5.084

4.  Enterovirus A71 antivirals: Past, present, and future.

Authors:  Jun Wang; Yanmei Hu; Madeleine Zheng
Journal:  Acta Pharm Sin B       Date:  2021-08-20       Impact factor: 14.903

5.  Pharmacological Characterization of the Mechanism of Action of R523062, a Promising Antiviral for Enterovirus D68.

Authors:  Chunlong Ma; Yanmei Hu; Jiantao Zhang; Jun Wang
Journal:  ACS Infect Dis       Date:  2020-08-05       Impact factor: 5.084

Review 6.  Acute flaccid myelitis: cause, diagnosis, and management.

Authors:  Olwen C Murphy; Kevin Messacar; Leslie Benson; Riley Bove; Jessica L Carpenter; Thomas Crawford; Janet Dean; Roberta DeBiasi; Jay Desai; Matthew J Elrick; Raquel Farias-Moeller; Grace Y Gombolay; Benjamin Greenberg; Matthew Harmelink; Sue Hong; Sarah E Hopkins; Joyce Oleszek; Catherine Otten; Cristina L Sadowsky; Teri L Schreiner; Kiran T Thakur; Keith Van Haren; Carolina M Carballo; Pin Fee Chong; Amary Fall; Vykuntaraju K Gowda; Jelte Helfferich; Ryutaro Kira; Ming Lim; Eduardo L Lopez; Elizabeth M Wells; E Ann Yeh; Carlos A Pardo
Journal:  Lancet       Date:  2020-12-23       Impact factor: 79.321

7.  Discovery of Potent and Broad-Spectrum Pyrazolopyridine-Containing Antivirals against Enteroviruses D68, A71, and Coxsackievirus B3 by Targeting the Viral 2C Protein.

Authors:  Yanmei Hu; Naoya Kitamura; Rami Musharrafieh; Jun Wang
Journal:  J Med Chem       Date:  2021-06-04       Impact factor: 8.039

8.  Fluoxetine Inhibits Enterovirus Replication by Targeting the Viral 2C Protein in a Stereospecific Manner.

Authors:  Lisa Bauer; Roberto Manganaro; Birgit Zonsics; Jeroen R P M Strating; Priscila El Kazzi; Moira Lorenzo Lopez; Rachel Ulferts; Clara van Hoey; Maria J Maté; Thierry Langer; Bruno Coutard; Andrea Brancale; Frank J M van Kuppeveld
Journal:  ACS Infect Dis       Date:  2019-07-31       Impact factor: 5.084

Review 9.  Current Understanding of Human Enterovirus D68.

Authors:  Jing Sun; Xiao-Yi Hu; Xiao-Fang Yu
Journal:  Viruses       Date:  2019-05-29       Impact factor: 5.048

Review 10.  Acute flaccid myelitis and enterovirus D68: lessons from the past and present.

Authors:  Jelte Helfferich; Marjolein Knoester; Coretta C Van Leer-Buter; Rinze F Neuteboom; Linda C Meiners; Hubert G Niesters; Oebele F Brouwer
Journal:  Eur J Pediatr       Date:  2019-07-23       Impact factor: 3.183

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