Literature DB >> 30349694

Onset of analgesia by a topically administered flurbiprofen lozenge: a randomised controlled trial using the double stopwatch method.

Bernard Schachtel1,2, Sue Aspley3, Adrian Shephard3, Emily Schachtel1, Mary Beth Lorton1, Tim Shea4.   

Abstract

BACKGROUND: The double stopwatch (DSW) method for determining the onset of analgesic activity has been implemented extensively by investigators studying orally administered drugs.
OBJECTIVE: The aim of this randomised, placebo-controlled trial was to use the DSW method to determine the time to onset of analgesia of a single dose of a topically administered non-steroidal anti-inflammatory drug, flurbiprofen 8.75 mg lozenge.
METHODS: Adults with acute sore throat (n = 122) were examined to confirm the presence of tonsillopharyngitis (Tonsillo-Pharyngitis Assessment) and sore throat pain of at least moderate intensity (≥6 on a 0-10 Sore Throat Scale). Lozenges containing flurbiprofen 8.75 mg or inert ingredients (identically flavoured) were administered under double-blind conditions in the clinic while patients assessed pain and pain relief over 3 hours. Onset of analgesia was determined using the DSW method and reported as the Kaplan-Meier median time to meaningful relief. The median time to first perceived relief was also documented.
RESULTS: About 78% of flurbiprofen-treated patients reported meaningful pain relief compared with 48% of placebo-treated patients (p < 0.01); median time to meaningful relief for flurbiprofen-treated patients was 43 minutes (placebo-treated patients were right-censored due to non-responsivity; p = 0.01). Median time to first perceived pain relief was 11 minutes for flurbiprofen-treated patients and 19 minutes for placebo-treated patients (p = 0.03). Flurbiprofen lozenge was well tolerated, with no serious adverse events occurring and no patient discontinuing due to an adverse event.
CONCLUSION: These results indicate that the DSW method can be successfully applied to the evaluation of the onset of action of a locally administered analgesic in patients with acute sore throat, demonstrating that the onset of action (time to meaningful pain relief) of flurbiprofen lozenge was <45 minutes.

Entities:  

Keywords:  Double stopwatch method; flurbiprofen; onset of action; pharyngitis; sore throat; topical analgesia

Year:  2018        PMID: 30349694      PMCID: PMC6194974          DOI: 10.1177/2049463718756152

Source DB:  PubMed          Journal:  Br J Pain        ISSN: 2049-4637


  26 in total

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Journal:  Can Fam Physician       Date:  2007-11       Impact factor: 3.275

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3.  Demonstration of dose response of flurbiprofen lozenges with the sore throat pain model.

Authors:  Bernard P Schachtel; Harvey D Homan; Iain A Gibb; Jenny Christian
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4.  Clinical practice guideline for the diagnosis and management of group A streptococcal pharyngitis: 2012 update by the Infectious Diseases Society of America.

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Authors:  A W van der Velden; J Bell; A Sessa; M Duerden; A Altiner
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8.  Utility of the sore throat pain model in a multiple-dose assessment of the acute analgesic flurbiprofen: a randomized controlled study.

Authors:  Bernard Schachtel; Sue Aspley; Adrian Shephard; Timothy Shea; Gary Smith; Emily Schachtel
Journal:  Trials       Date:  2014-07-03       Impact factor: 2.279

9.  Continued high rates of antibiotic prescribing to adults with respiratory tract infection: survey of 568 UK general practices.

Authors:  Martin C Gulliford; Alex Dregan; Michael V Moore; Mark Ashworth; Tjeerd van Staa; Gerard McCann; Judith Charlton; Lucy Yardley; Paul Little; Lisa McDermott
Journal:  BMJ Open       Date:  2014-10-27       Impact factor: 2.692

10.  Efficacy of disintegrating aspirin in two different models for acute mild-to-moderate pain: sore throat pain and dental pain.

Authors:  M Voelker; B P Schachtel; S A Cooper; S C Gatoulis
Journal:  Inflammopharmacology       Date:  2015-11-24       Impact factor: 4.473

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  5 in total

1.  Determination of the Permeation and Penetration of Flurbiprofen into Cadaveric Human Pharynx Tissue.

Authors:  Rob Turner; Sean Robert Wevrett; Suzanne Edmunds; Marc B Brown; Robert Atkinson; Oluwajoba Adegoke; Anuradha Kulasekaran; Tim Shea
Journal:  Clin Pharmacol       Date:  2020-03-24

Review 2.  Locally Delivered Flurbiprofen 8.75 mg for Treatment and Prevention of Sore Throat: A Narrative Review of Clinical Studies.

Authors:  Ferdinandus de Looze; Adrian Shephard; Adam B Smith
Journal:  J Pain Res       Date:  2019-12-27       Impact factor: 3.133

3.  Penetration of Flurbiprofen from a Locally Applied Sore Throat Lozenge and Spray into Cadaveric Human Pharynx Tissue: A Novel ex vivo Model and Microautoradiography Method.

Authors:  Rob Turner; Sean Robert Wevrett; Suzanne Edmunds; Marc Brown; Anuradha Kulasekaran; Oluwajoba Adegoke; John Farrah
Journal:  Clin Pharmacol       Date:  2021-01-19

4.  Evaluation on immediate analgesic efficacy and safety of Kai-Hou-Jian spray (children's type) in treating sore throat caused by acute pharyngitis and tonsillitis in children: study protocol for a randomized controlled trial.

Authors:  Yan-Ning Ma; Cheng-Liang Zhong; Si-Yuan Hu; Qiu-Han Cai; Sheng-Xuan Guo
Journal:  Trials       Date:  2021-03-18       Impact factor: 2.279

5.  Validation of an analytical method to quantify the permeation and penetration of flurbiprofen into human pharynx tissue.

Authors:  Rob Turner; Sean Robert Wevrett; Suzanne Edmunds; Marc Brown; Robert Atkinson; Tim Shea
Journal:  Biomed Chromatogr       Date:  2019-05-06       Impact factor: 1.902

  5 in total

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