Literature DB >> 30309721

A phase II evaluation of elesclomol sodium and weekly paclitaxel in the treatment of recurrent or persistent platinum-resistant ovarian, fallopian tube or primary peritoneal cancer: An NRG oncology/gynecologic oncology group study.

Bradley J Monk1, James T Kauderer2, Katherine M Moxley3, Albert J Bonebrake4, Summer B Dewdney5, Angeles Alvarez Secord6, Frederick R Ueland7, Carolyn M Johnston8, Carol Aghajanian9.   

Abstract

OBJECTIVE: Preclinical data suggest elesclomol increases oxidative stress and enhances sensitivity to cytotoxic agents. The objective of this prospective multicenter phase 2 trial was to estimate the activity of IV elesclomol plus weekly paclitaxel in patients with platinum-resistant recurrent ovarian, tubal or peritoneal cancer through the frequency of objective tumor responses (ORR).
METHODS: Patients with measurable disease, acceptable organ function, performance status ≤ 2, and one prior platinum containing regimen were eligible. A two-stage design was utilized with a target sample size of 22 and 30 subjects, respectively. Prior Gynecologic Oncology Group studies within the same population involving single agent taxanes showed an ORR of approximately (20%) and served as a historical control for direct comparison. The present study was designed to determine if the regimen had an ORR of ≥40% with 90% power.
RESULTS: Fifty-eight patients were enrolled, of whom 2 received no study treatment and were inevaluable. The median number of cycles was 3 (268 total cycles, range 1-18). The number of patients responding was 11 (19.6%; 90% CI 11.4% to 30.4%) with one complete response. The median progression-free survival and overall survival was 3.6 months and 13.3 months, respectively. The median ORR duration was 9.2 months. Percentages of subjects with grade 3 toxicity included: Neutropenia 9%; anemia 5%; metabolic 5%; nausea 4%; infection 4%; neurologic (mostly neuropathy) 4%; and vascular (mostly thromboembolism) 4%. There were no grade 4 toxicities reported.
CONCLUSIONS: This combination was well tolerated but is unworthy of further investigation based on the proportion responding [ClinicalTrials.gov Identifier: NCT00888615].
Copyright © 2018. Published by Elsevier Inc.

Entities:  

Keywords:  Clinical trial; Elesclomol; Ovarian cancer

Mesh:

Substances:

Year:  2018        PMID: 30309721      PMCID: PMC6392076          DOI: 10.1016/j.ygyno.2018.10.001

Source DB:  PubMed          Journal:  Gynecol Oncol        ISSN: 0090-8258            Impact factor:   5.482


  9 in total

1.  Copper ionophore elesclomol selectively targets GNAQ/11-mutant uveal melanoma.

Authors:  Yongyun Li; Jie Yang; Qianqian Zhang; Shiqiong Xu; Wei Sun; Shengfang Ge; Xiaowei Xu; Martine J Jager; Renbing Jia; Jianming Zhang; Xianqun Fan
Journal:  Oncogene       Date:  2022-06-13       Impact factor: 8.756

2.  Onvansertib and paclitaxel combined in platinum-resistant ovarian carcinomas.

Authors:  Roberta Affatato; Michela Chiappa; Federica Guffanti; Francesca Ricci; Laura Formenti; Robert Fruscio; Marta Jaconi; Maya Ridinger; Mark Erlander; Giovanna Damia
Journal:  Ther Adv Med Oncol       Date:  2022-05-31       Impact factor: 5.485

Review 3.  Interplay Between MicroRNAs and Oxidative Stress in Ovarian Conditions with a Focus on Ovarian Cancer and Endometriosis.

Authors:  Josep Marí-Alexandre; Antonio Pellín Carcelén; Cristina Agababyan; Andrea Moreno-Manuel; Javier García-Oms; Silvia Calabuig-Fariñas; Juan Gilabert-Estellés
Journal:  Int J Mol Sci       Date:  2019-10-25       Impact factor: 5.923

Review 4.  Selective Targeting of Cancer Cells by Copper Ionophores: An Overview.

Authors:  Valentina Oliveri
Journal:  Front Mol Biosci       Date:  2022-03-04

5.  A novel cuproptosis-related gene signature for predicting prognosis in cervical cancer.

Authors:  Lei Lei; Liao Tan; Long Sui
Journal:  Front Genet       Date:  2022-08-25       Impact factor: 4.772

Review 6.  Elesclomol: a copper ionophore targeting mitochondrial metabolism for cancer therapy.

Authors:  Peijie Zheng; Chuntao Zhou; Liuyi Lu; Bin Liu; Yuemin Ding
Journal:  J Exp Clin Cancer Res       Date:  2022-09-12

7.  Cuproptosis status affects treatment options about immunotherapy and targeted therapy for patients with kidney renal clear cell carcinoma.

Authors:  Ganghua Zhang; Xinyu Chen; Jianing Fang; Panpan Tai; Aiyan Chen; Ke Cao
Journal:  Front Immunol       Date:  2022-08-19       Impact factor: 8.786

8.  Pan-cancer analysis of cuproptosis regulation patterns and identification of mTOR-target responder in clear cell renal cell carcinoma.

Authors:  Shichao Long; Ya Wang; Yuqiao Chen; Tianshu Fang; Yuanbing Yao; Kai Fu
Journal:  Biol Direct       Date:  2022-10-08       Impact factor: 7.173

Review 9.  Metallo-Drugs in Cancer Therapy: Past, Present and Future.

Authors:  Roxana Liana Lucaciu; Adriana Corina Hangan; Bogdan Sevastre; Luminița Simona Oprean
Journal:  Molecules       Date:  2022-10-01       Impact factor: 4.927

  9 in total

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