Literature DB >> 30284134

Pharmacological Treatment of Opioid-Induced Constipation Is Effective but Choice of Endpoints Affects the Therapeutic Gain.

Salman Nusrat1, Taseen Syed2, Rabia Saleem2, Shari Clifton3,4, Klaus Bielefeldt5.   

Abstract

BACKGROUND: Widespread opioid use has led to increase in opioid-related adverse effects like constipation. We examined the impact of study endpoints on reported treatment benefits.
METHODS: Using MEDLINE, EMBASE, and ClinicalTrials.gov, we searched for randomized control trials targeting chronic opioid-induced constipation (OIC) and subjected them to meta-analysis. Data are given with 95% confidence intervals.
RESULTS: Thirty trials met our inclusion criteria. Combining all dichotomous definitions of responders, active drugs were consistently more effective than placebo, with an odds ratio (OR): 2.30 [2.01-2.63; 15 studies], independent of the underlying drug mechanism. The choice of endpoints significantly affected the therapeutic gain. When time from drug administration to defecation was used, the OR decreased from 4.74 [2.71-4.74] at 6 h or less to 2.46 [1.80-3.30] at 24 h (P < 0.05). Using other response definitions, the relative benefit over placebo was 2.10 [1.77-2.50; 12 studies] for weekly bowel frequency, 2.03 [1.39-2.95; 9 studies] for symptom scores, 2.21 [1.25-3.90; 4 studies] for global assessment scales, and 1.27 [0.79-2.03; 7 studies] for rescue laxative use.
CONCLUSION: While treatment of OIC with active drugs is more effective than placebo, the relative gain depends on the choice of endpoints. The commonly used time-dependent response definition is associated with the highest response rate but is of questionable relevance in a chronic disorder. The limited data do not clearly demonstrate a unique advantage of the peripherally restricted opioid antagonists, suggesting that treatment with often cheaper agents should be optimized before shifting to these novel expensive agents.

Entities:  

Keywords:  Laxative use; Methylnaltrexone; Naloxegol; Opioid antagonists; Opioid-induced constipation

Mesh:

Substances:

Year:  2018        PMID: 30284134     DOI: 10.1007/s10620-018-5308-9

Source DB:  PubMed          Journal:  Dig Dis Sci        ISSN: 0163-2116            Impact factor:   3.199


  47 in total

1.  Both Urgency and Balance Needed in Addressing Opioid Epidemic: A Report From the National Academies of Sciences, Engineering, and Medicine.

Authors:  Richard J Bonnie; Aaron S Kesselheim; David J Clark
Journal:  JAMA       Date:  2017-08-01       Impact factor: 56.272

2.  Subcutaneous methylnaltrexone for treatment of opioid-induced constipation in patients with chronic, nonmalignant pain: a randomized controlled study.

Authors:  Edward Michna; E Richard Blonsky; Seth Schulman; Evan Tzanis; Amy Manley; Haiying Zhang; Shrividya Iyer; Bruce Randazzo
Journal:  J Pain       Date:  2011-03-22       Impact factor: 5.820

3.  A randomized, placebo-controlled phase 3 trial (Study SB-767905/013) of alvimopan for opioid-induced bowel dysfunction in patients with non-cancer pain.

Authors:  Gordon Irving; Janos Pénzes; Brian Ramjattan; Michael Cousins; Richard Rauck; Egilius L H Spierings; Christi S Kleoudis; Jerry W Snidow; Amy Pierce; John Wurzelmann; Eric R Mortensen
Journal:  J Pain       Date:  2011-02       Impact factor: 5.820

4.  Efficacy and safety of prucalopride in patients with chronic noncancer pain suffering from opioid-induced constipation.

Authors:  Cornelius E J Sloots; An Rykx; Marina Cools; Rene Kerstens; Martine De Pauw
Journal:  Dig Dis Sci       Date:  2010-04-30       Impact factor: 3.199

5.  Efficacy of Treatments for Opioid-Induced Constipation: Systematic Review and Meta-analysis.

Authors:  Judy Nee; Mohammed Zakari; Michael A Sugarman; Julia Whelan; William Hirsch; Shahnaz Sultan; Sarah Ballou; Johanna Iturrino; Anthony Lembo
Journal:  Clin Gastroenterol Hepatol       Date:  2018-01-31       Impact factor: 11.382

6.  Methylnaltrexone for treatment of opioid-induced constipation in advanced illness patients.

Authors:  Neal Slatkin; Jay Thomas; Arthur G Lipman; George Wilson; Michelle L Boatwright; Charles Wellman; Donna S Zhukovsky; Richard Stephenson; Russell Portenoy; Nancy Stambler; Robert Israel
Journal:  J Support Oncol       Date:  2009 Jan-Feb

7.  Methylnaltrexone for opioid-induced constipation in advanced illness.

Authors:  Jay Thomas; Sloan Karver; Gail Austin Cooney; Bruce H Chamberlain; Charles Kevin Watt; Neal E Slatkin; Nancy Stambler; Alton B Kremer; Robert J Israel
Journal:  N Engl J Med       Date:  2008-05-29       Impact factor: 91.245

8.  Phase IIb, Randomized, Double-Blind, Placebo-Controlled Study of Naldemedine for the Treatment of Opioid-Induced Constipation in Patients With Cancer.

Authors:  Nobuyuki Katakami; Koji Oda; Katsunori Tauchi; Ken Nakata; Katsunori Shinozaki; Takaaki Yokota; Yura Suzuki; Masaru Narabayashi; Narikazu Boku
Journal:  J Clin Oncol       Date:  2017-04-26       Impact factor: 50.717

9.  Fixed-Dose Subcutaneous Methylnaltrexone in Patients with Advanced Illness and Opioid-Induced Constipation: Results of a Randomized, Placebo-Controlled Study and Open-Label Extension.

Authors:  Janet Bull; Charles V Wellman; Robert J Israel; Andrew C Barrett; Craig Paterson; William P Forbes
Journal:  J Palliat Med       Date:  2015-05-14       Impact factor: 2.947

10.  Prescription Opioid Use, Misuse, and Use Disorders in U.S. Adults: 2015 National Survey on Drug Use and Health.

Authors:  Beth Han; Wilson M Compton; Carlos Blanco; Elizabeth Crane; Jinhee Lee; Christopher M Jones
Journal:  Ann Intern Med       Date:  2017-08-01       Impact factor: 25.391

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