Literature DB >> 30056318

Effects of gap junctions blockers on fast ripples and connexin in rat hippocampi after status epilepticus.

Xiao Ran1, Jing Xiang2, Pan-Pan Song3, Li Jiang4, Ben-Ke Liu5, Yue Hu6.   

Abstract

OBJECTIVE: To assess the dynamic changes in the average and peak spectral power of fast ripples (FRs) in the hippocampi after interventions with valproate sodium (VPA), carbenoxolone (CBX) and quinine (QUIN).
METHOD: Adult rats were used to establish a lithium-pilocarpine (pilo) epileptic model, and were assigned to a lithium-pilocarpine (PILO), VPA + PILO, QUIN + PILO or CBX + PILO group. Intracranial electroencephalography was performed before and after status epilepticus (SE). The hippocampal connexin (CX) 43, CX32 and CX36 expressions were analyzed via western blotting.
RESULTS: The time required for the disappearance of SE after chloral hydrate injection was lower in the intervention groups than in the PILO group (p < 0.05). Seizures induced CX43 expression, but had no significant effects on CX36 or CX32 expressions. Pretreatment with VPA, QUIN and CBX inhibited CX43, CX36 and CX32 expression after SE. The average spectral power of the FRs was significantly lower in the VPA + PILO and QUIN + PILO groups than in the PILO group at 10 min after SE, 10 min before chloral hydrate injection, and 10 min after chloral hydrate injection (p < 0.05). The average spectral power of FRs was lower in the CBX + PILO group than in the PILO group at 10 min after SE (p < 0.05). The average spectral power of FRs in the 3 intervention groups recovered to the baseline level at 10 min after chloral hydrate injection and persisted for 3 days after SE. The dynamic changes in the average and peak spectral power of FRs were similar. SIGNIFICANCE: After SE, CX may participate in pathological FR generation by establishing abnormal electrical synaptic transmission. Gap junction blockers can inhibit various CX expressions, and thus decrease FR energy and alleviate the degree of seizure. These findings could contribute to the development of new anti-epileptic drugs with novel mechanistic targets.
Copyright © 2018 Elsevier B.V. All rights reserved.

Entities:  

Keywords:  Carbenoxolone; Epilepsy; Fast ripples; Gap junction; Quinine

Mesh:

Substances:

Year:  2018        PMID: 30056318     DOI: 10.1016/j.eplepsyres.2018.07.010

Source DB:  PubMed          Journal:  Epilepsy Res        ISSN: 0920-1211            Impact factor:   3.045


  5 in total

1.  Anticonvulsant Effect of Carbenoxolone on Chronic Epileptic Rats and Its Mechanism Related to Connexin and High-Frequency Oscillations.

Authors:  Benke Liu; Xiao Ran; Yanjun Yi; Xinyu Zhang; Hengsheng Chen; Yue Hu
Journal:  Front Mol Neurosci       Date:  2022-05-09       Impact factor: 6.261

2.  The protective effect of carbenoxolone on gap junction damage in the hippocampal CA1 area of a temporal lobe epilepsy rat model.

Authors:  Yi Shu; Can Zhu; Min Zeng; Qiong Zhan; Zhiping Hu; Xiaomei Wu
Journal:  Ann Transl Med       Date:  2019-11

Review 3.  Astrocytes as Guardians of Neuronal Excitability: Mechanisms Underlying Epileptogenesis.

Authors:  Quirijn P Verhoog; Linda Holtman; Eleonora Aronica; Erwin A van Vliet
Journal:  Front Neurol       Date:  2020-11-26       Impact factor: 4.003

Review 4.  Connexins-Based Hemichannels/Channels and Their Relationship with Inflammation, Seizures and Epilepsy.

Authors:  Laura Medina-Ceja; Juan C Salazar-Sánchez; Jorge Ortega-Ibarra; Alberto Morales-Villagrán
Journal:  Int J Mol Sci       Date:  2019-11-27       Impact factor: 5.923

5.  The Anti-Epileptic Effects of Carbenoxolone In Vitro and In Vivo.

Authors:  Anna Volnova; Vassiliy Tsytsarev; Olga Ganina; Grace E Vélez-Crespo; Janaina M Alves; Alla Ignashchenkova; Mikhail Inyushin
Journal:  Int J Mol Sci       Date:  2022-01-08       Impact factor: 5.923

  5 in total

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