Literature DB >> 29976087

Sildenafil and calcitonin gene-related peptide dilate intradural arteries: A 3T MR angiography study in healthy volunteers.

Casper Emil Christensen1, Faisal Mohammad Amin1, Samaira Younis1, Ulrich Lindberg2, Patrick de Koning3, Esben Thade Petersen4, Olaf Bjarne Paulson5, Henrik Bo Wiberg Larsson2, Messoud Ashina1.   

Abstract

BACKGROUND: Sildenafil and calcitonin gene-related peptide are vasoactive substances that induce migraine attacks in patients. The intradural arteries are thought to be involved, but these have never been examined in vivo. Sildenafil is the only migraine-inducing compound for which cephalic, extracranial artery dilation is not reported. Here, we investigate the effects of sildenafil and calcitonin gene-related peptide on the extracranial and intradural parts of the middle meningeal artery.
METHODS: In a double-blind, randomized, three-way crossover, placebo-controlled head-to-head comparison study, MR-angiography was recorded in healthy volunteers at baseline and twice after study drug (sildenafil/ calcitonin gene-related peptide/saline) administration. Circumferences of extracranial and intradural middle meningeal artery segments were measured using semi-automated analysis software. The area under the curve for circumference change was compared using paired t-tests between study days.
RESULTS: Twelve healthy volunteers completed the study. The area under the curveBaseline-120min was significantly larger on both the sildenafil and the calcitonin gene-related peptide day in the intradural middle meningeal artery (calcitonin gene-related peptide, p = 0.013; sildenafil, p = 0.027) and the extracranial middle meningeal artery (calcitonin gene-related peptide, p = 0.0003; sildenafil, p = 0.021), compared to placebo. Peak intradural middle meningeal artery dilation was 9.9% (95% CI [2.9-16.9]) after sildenafil (T30min) and 12.5% (95% CI [8.1-16.8]) after calcitonin gene-related peptide (T30min). Peak dilation of the extracranial middle meningeal artery after calcitonin gene-related peptide (T30min) was 15.7% (95% CI [11.2-20.1]) and 18.9% (95% CI [12.8-24.9]) after sildenafil (T120min).
CONCLUSION: An important novel finding is that both sildenafil and calcitonin gene-related peptide dilate intradural arteries, supporting the notion that all known pharmacological migraine triggers dilate cephalic vessels. We suggest that intradural artery dilation is associated with headache induced by calcitonin gene-related peptide and sildenafil.

Entities:  

Keywords:  Neuroimaging; human migraine models; middle meningeal artery

Mesh:

Substances:

Year:  2018        PMID: 29976087     DOI: 10.1177/0333102418787336

Source DB:  PubMed          Journal:  Cephalalgia        ISSN: 0333-1024            Impact factor:   6.292


  6 in total

1.  New discoveries in migraine mechanisms and therapeutic targets.

Authors:  Greg Dussor
Journal:  Curr Opin Physiol       Date:  2019-10-18

2.  Cerebrovascular effects of glibenclamide investigated using high-resolution magnetic resonance imaging in healthy volunteers.

Authors:  Mohammad Al-Mahdi Al-Karagholi; Hashmat Ghanizada; Cherie Amalie Waldorff Nielsen; Assan Ansari; Christian Gram; Samaria Younis; Mark B Vestergaard; Henrik Bw Larsson; Lene Theil Skovgaard; Faisal Mohammad Amin; Messoud Ashina
Journal:  J Cereb Blood Flow Metab       Date:  2020-10-07       Impact factor: 6.200

Review 3.  Why is the therapeutic effect of acute antimigraine drugs delayed? A review of controlled trials and hypotheses about the delay of effect.

Authors:  Peer Tfelt-Hansen; Karl Messlinger
Journal:  Br J Clin Pharmacol       Date:  2019-09-04       Impact factor: 4.335

4.  Ultra-high field MR angiography in human migraine models: a 3.0 T/7.0 T comparison study.

Authors:  Casper Emil Christensen; Samaira Younis; Ulrich Lindberg; Vincent Oltman Boer; Patrick de Koning; Esben Thade Petersen; Olaf Bjarne Paulson; Henrik Bo Wiberg Larsson; Faisal Mohammad Amin; Messoud Ashina
Journal:  J Headache Pain       Date:  2019-05-06       Impact factor: 7.277

5.  Vascular actions of peripheral CGRP in migraine-like photophobia in mice.

Authors:  Bianca N Mason; Anne-Sophie Wattiez; Louis K Balcziak; Adisa Kuburas; William J Kutschke; Andrew F Russo
Journal:  Cephalalgia       Date:  2020-08-18       Impact factor: 6.292

6.  Cerebrovascular Reactivity Measures Are Associated With Post-traumatic Headache Severity in Chronic TBI; A Retrospective Analysis.

Authors:  Franck Amyot; Cillian E Lynch; John Ollinger; J Kent Werner; E Silverman; Carol Moore; Cora Davis; L Christine Turtzo; Ramon Diaz-Arrastia; Kimbra Kenney
Journal:  Front Physiol       Date:  2021-05-13       Impact factor: 4.566

  6 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.