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Literature DB >> 2988419

Affinity labels for opioid receptors.

A E Takemori, P S Portoghese.

Abstract

Mesh：

Substances：

Year: 1985 PMID： 2988419 DOI： 10.1146/annurev.pa.25.040185.001205

Source DB: PubMed Journal: Annu Rev Pharmacol Toxicol ISSN： 0362-1642 Impact factor: 13.820

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16 in total

1. Dual labeled peptides as tools to study receptors: nanomolar affinity derivatives of TIPP (Tyr-Tic-Phe-Phe) containing an affinity label and biotin as probes of delta opioid receptors.

Authors: Jane V Aldrich; Vivek Kumar; Thomas F Murray; Wei Guang; Jia Bei Wang
Journal: Bioconjug Chem Date: 2009-02 Impact factor: 4.774

2. K303⁶·⁵⁸ in the μ opioid (MOP) receptor is important in conferring selectivity for covalent binding of β-funaltrexamine (β-FNA).

Authors: Kelly M DiMattio; Chongguang Chen; Lei Shi; Lee-Yuan Liu-Chen
Journal: Eur J Pharmacol Date: 2014-12-04 Impact factor: 4.432

3. Affinity labeling mu opioid receptors with novel radioligands.

Authors: Ke Yang; Amy Zuckerman; Gavril W Pasternak
Journal: Cell Mol Neurobiol Date: 2005-06 Impact factor: 5.046

4. Solid Phase Synthesis and Application of Labeled Peptide Derivatives: Probes of Receptor-Opioid Peptide Interactions.

Authors: Jane V Aldrich; Vivek Kumar; Bhaswati Dattachowdhury; Angela M Peck; Xin Wang; Thomas F Murray
Journal: Int J Pept Res Ther Date: 2008-12-01 Impact factor: 1.931

5. Discovery of dermorphin-based affinity labels with subnanomolar affinity for mu opioid receptors.

Authors: Bhaswati Sinha; Zhengyu Cao; Thomas F Murray; Jane V Aldrich
Journal: J Med Chem Date: 2009-12-10 Impact factor: 7.446

6. Synthesis and characterization of a dual kappa-delta opioid receptor agonist analgesic blocking cocaine reward behavior.

Authors: András Váradi; Gina F Marrone; Shainnel O Eans; Michelle L Ganno; Joan J Subrath; Valerie Le Rouzic; Amanda Hunkele; Gavril W Pasternak; Jay P McLaughlin; Susruta Majumdar
Journal: ACS Chem Neurosci Date: 2015-09-14 Impact factor: 4.418

Affinity labels for opioid receptors.

1. Dual labeled peptides as tools to study receptors: nanomolar affinity derivatives of TIPP (Tyr-Tic-Phe-Phe) containing an affinity label and biotin as probes of delta opioid receptors.

2. K303⁶·⁵⁸ in the μ opioid (MOP) receptor is important in conferring selectivity for covalent binding of β-funaltrexamine (β-FNA).

3. Affinity labeling mu opioid receptors with novel radioligands.

4. Solid Phase Synthesis and Application of Labeled Peptide Derivatives: Probes of Receptor-Opioid Peptide Interactions.

5. Discovery of dermorphin-based affinity labels with subnanomolar affinity for mu opioid receptors.

6. Synthesis and characterization of a dual kappa-delta opioid receptor agonist analgesic blocking cocaine reward behavior.

7. Optical Control of Dopamine Receptors Using a Photoswitchable Tethered Inverse Agonist.

8. Novel 6β-acylaminomorphinans with analgesic activity.

9. Discovery of lacosamide affinity bait agents that exhibit potent voltage-gated sodium channel blocking properties.

10. Lacosamide isothiocyanate-based agents: novel agents to target and identify lacosamide receptors.