Literature DB >> 29790904

Exploring drug space with ChemMaps.com.

Alexandre Borrel1,2, Nicole C Kleinstreuer2,3, Denis Fourches1.   

Abstract

Motivation: Easily navigating chemical space has become more important due to the increasing size and diversity of publicly-accessible databases such as DrugBank, ChEMBL or Tox21. To do so, modelers typically rely on complex projection techniques using molecular descriptors computed for all the chemicals to be visualized. However, the multiple cheminformatics steps required to prepare, characterize, compute and explore those molecules, are technical, typically necessitate scripting skills, and thus represent a real obstacle for non-specialists.
Results: We developed the ChemMaps.com webserver to easily browse, navigate and mine chemical space. The first version of ChemMaps.com features more than 8000 approved, in development, and rejected drugs, as well as over 47 000 environmental chemicals. Availability and implementation: The webserver is freely available at http://www.chemmaps.com.

Mesh:

Year:  2018        PMID: 29790904      PMCID: PMC6454477          DOI: 10.1093/bioinformatics/bty412

Source DB:  PubMed          Journal:  Bioinformatics        ISSN: 1367-4803            Impact factor:   6.937


  8 in total

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Authors:  T I Oprea; J Gottfries
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2.  ChemGPS-NP(Web): chemical space navigation online.

Authors:  Josefin Rosén; Anders Lövgren; Thierry Kogej; Sorel Muresan; Johan Gottfries; Anders Backlund
Journal:  J Comput Aided Mol Des       Date:  2008-12-10       Impact factor: 3.686

3.  PyDPI: freely available python package for chemoinformatics, bioinformatics, and chemogenomics studies.

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Journal:  J Chem Inf Model       Date:  2013-10-24       Impact factor: 4.956

4.  Generative Topographic Mapping (GTM): Universal Tool for Data Visualization, Structure-Activity Modeling and Dataset Comparison.

Authors:  N Kireeva; I I Baskin; H A Gaspar; D Horvath; G Marcou; A Varnek
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5.  Using Graph Indices for the Analysis and Comparison of Chemical Datasets.

Authors:  Denis Fourches; Alexander Tropsha
Journal:  Mol Inform       Date:  2013-09-09       Impact factor: 3.353

Review 6.  Trust, but Verify II: A Practical Guide to Chemogenomics Data Curation.

Authors:  Denis Fourches; Eugene Muratov; Alexander Tropsha
Journal:  J Chem Inf Model       Date:  2016-06-22       Impact factor: 4.956

7.  DrugBank 4.0: shedding new light on drug metabolism.

Authors:  Vivian Law; Craig Knox; Yannick Djoumbou; Tim Jewison; An Chi Guo; Yifeng Liu; Adam Maciejewski; David Arndt; Michael Wilson; Vanessa Neveu; Alexandra Tang; Geraldine Gabriel; Carol Ly; Sakina Adamjee; Zerihun T Dame; Beomsoo Han; You Zhou; David S Wishart
Journal:  Nucleic Acids Res       Date:  2013-11-06       Impact factor: 16.971

8.  Web-based 3D-visualization of the DrugBank chemical space.

Authors:  Mahendra Awale; Jean-Louis Reymond
Journal:  J Cheminform       Date:  2016-05-04       Impact factor: 5.514

  8 in total
  3 in total

1.  Progress on open chemoinformatic tools for expanding and exploring the chemical space.

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Journal:  J Comput Aided Mol Des       Date:  2021-06-18       Impact factor: 4.179

2.  Finding Constellations in Chemical Space Through Core Analysis.

Authors:  J Jesús Naveja; José L Medina-Franco
Journal:  Front Chem       Date:  2019-07-16       Impact factor: 5.221

3.  DrugSpaceX: a large screenable and synthetically tractable database extending drug space.

Authors:  Tianbiao Yang; Zhaojun Li; Yingjia Chen; Dan Feng; Guangchao Wang; Zunyun Fu; Xiaoyu Ding; Xiaoqin Tan; Jihui Zhao; Xiaomin Luo; Kaixian Chen; Hualiang Jiang; Mingyue Zheng
Journal:  Nucleic Acids Res       Date:  2021-01-08       Impact factor: 16.971

  3 in total

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