Literature DB >> 29724385

Sildenafil added to pirfenidone in patients with advanced idiopathic pulmonary fibrosis and risk of pulmonary hypertension: A Phase IIb, randomised, double-blind, placebo-controlled study - Rationale and study design.

Jürgen Behr1, Steven D Nathan2, Sergio Harari3, Wim Wuyts4, Klaus-Uwe Kirchgaessler5, Monica Bengus5, Frank Gilberg5, Athol U Wells6.   

Abstract

BACKGROUND: Pulmonary hypertension (PH) is commonly observed in patients with advanced idiopathic pulmonary fibrosis (IPF). Despite the availability of therapies for both IPF and PH, none are approved for PH treatment in the context of significant pulmonary disease. This study will investigate the use of sildenafil added to pirfenidone in patients with advanced IPF and risk of PH, who represent a group with a high unmet medical need.
METHODS: This Phase IIb, randomised, double-blind, placebo-controlled trial is actively enrolling patients and will study the efficacy, safety and tolerability of sildenafil or placebo in patients with advanced IPF and intermediate or high probability of Group 3 PH who are receiving a stable dose of pirfenidone. Patients with advanced IPF (diffusing capacity for carbon monoxide ≤40% predicted) and risk of Group 3 PH (defined as mean pulmonary arterial pressure ≥20 mm Hg with pulmonary arterial wedge pressure ≤15 mm Hg on a previous right-heart catheterisation [RHC], or intermediate/high probability of Group 3 PH as defined by the 2015 European Society of Cardiology/European Respiratory Society guidelines) are eligible. In the absence of a previous RHC, patients with an echocardiogram showing a peak tricuspid valve regurgitation velocity ≥2.9 m/s can enrol if all other criteria are met. The primary efficacy endpoint is the proportion of patients with disease progression over a 52-week treatment period. Safety will be evaluated descriptively. DISCUSSION: Combination treatment with sildenafil and pirfenidone may warrant investigation of the treatment of patients with advanced IPF and pulmonary vascular involvement leading to PH.
Copyright © 2018 The Authors. Published by Elsevier Ltd.. All rights reserved.

Entities:  

Keywords:  6-Minute walk test; Clinical trial; Echocardiogram; Hypertension; Idiopathic pulmonary fibrosis; Phosphodiesterase-5 inhibitor; Pirfenidone; Sildenafil

Mesh:

Substances:

Year:  2018        PMID: 29724385     DOI: 10.1016/j.rmed.2018.03.019

Source DB:  PubMed          Journal:  Respir Med        ISSN: 0954-6111            Impact factor:   3.415


  10 in total

Review 1.  Idiopathic pulmonary fibrosis and pulmonary hypertension: Heracles meets the Hydra.

Authors:  Keshava Rajagopal; Andrew J Bryant; Sandeep Sahay; Nancy Wareing; Yang Zhou; Lavannya M Pandit; Harry Karmouty-Quintana
Journal:  Br J Pharmacol       Date:  2020-04-07       Impact factor: 8.739

Review 2.  Pharmacotherapy and adjunctive treatment for idiopathic pulmonary fibrosis (IPF).

Authors:  Shigeki Saito; Ala Alkhatib; Jay K Kolls; Yasuhiro Kondoh; Joseph A Lasky
Journal:  J Thorac Dis       Date:  2019-09       Impact factor: 2.895

3.  Survey on Sildenafil, Tadalafil, and Vardenafil Concentrations in Food Supplements for Erectile Dysfunction.

Authors:  Elina Petkova-Gueorguieva; Stanislav Gueorguiev; Hristina Lebanova; Vasil Madzharov; Anna Mihaylova
Journal:  Int J Anal Chem       Date:  2022-07-09       Impact factor: 1.698

4.  MiR-200a inversely correlates with Hedgehog and TGF-β canonical/non-canonical trajectories to orchestrate the anti-fibrotic effect of Tadalafil in a bleomycin-induced pulmonary fibrosis model.

Authors:  Suzan M Mansour; Hanan S El-Abhar; Ayman A Soubh
Journal:  Inflammopharmacology       Date:  2020-09-10       Impact factor: 4.473

Review 5.  Management of Idiopathic Pulmonary Fibrosis.

Authors:  Roy Pleasants; Robert M Tighe
Journal:  Ann Pharmacother       Date:  2019-07-07       Impact factor: 3.154

Review 6.  Idiopathic Pulmonary Fibrosis for Cardiologists: Differential Diagnosis, Cardiovascular Comorbidities, and Patient Management.

Authors:  Johan van Cleemput; Andrea Sonaglioni; Wim A Wuyts; Monica Bengus; John L Stauffer; Sergio Harari
Journal:  Adv Ther       Date:  2018-12-15       Impact factor: 3.845

7.  Curable Syncope in Primary Pulmonary Hypertension with Novel Atrial Flow Regulator.

Authors:  Babak Sharif-Kashani; Alireza Serati; Shadi Shafaghi; Neda Behzadnia; Farah Naghashzadeh; Mohammad Sadegh Keshmiri; Maedeh Moradi
Journal:  Tanaffos       Date:  2021-03

8.  Combined Pulmonary Fibrosis Emphysema: Role of Cigarette Smoking and Pulmonary Hypertension in a Rural Cohort.

Authors:  Rahul Sangani; Andrew Ghio; Stacey Culp; Zalak Patel; Sunil Sharma
Journal:  Int J Chron Obstruct Pulmon Dis       Date:  2021-06-21

9.  Phosphodiesterase 5 inhibitors for pulmonary hypertension.

Authors:  Hayley Barnes; Zoe Brown; Andrew Burns; Trevor Williams
Journal:  Cochrane Database Syst Rev       Date:  2019-01-31

10.  Targeting the NO-cGMP-PDE5 pathway in COVID-19 infection. The DEDALO project.

Authors:  Andrea M Isidori; Elisa Giannetta; Riccardo Pofi; Mary A Venneri; Daniele Gianfrilli; Federica Campolo; Claudio M Mastroianni; Andrea Lenzi; Gabriella d'Ettorre
Journal:  Andrology       Date:  2020-07-03       Impact factor: 4.456

  10 in total

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