Literature DB >> 29722661

Phase 2 Study of Bortezomib Combined With Temozolomide and Regional Radiation Therapy for Upfront Treatment of Patients With Newly Diagnosed Glioblastoma Multiforme: Safety and Efficacy Assessment.

Xiao-Tang Kong1, Nhung T Nguyen2, Yoon J Choi2, Guicheng Zhang3, HuyTram N Nguyen2, Emese Filka2, Stacey Green2, William H Yong4, Linda M Liau5, Richard M Green6, Tania Kaprealian7, Whitney B Pope8, P Leia Nghiemphu2, Timothy Cloughesy2, Andrew Lassman9, Albert Lai10.   

Abstract

PURPOSE: To assess the safety and efficacy of upfront treatment using bortezomib combined with standard radiation therapy (RT) and temozolomide (TMZ), followed by adjuvant bortezomib and TMZ for ≤24 cycles, in patients with newly diagnosed glioblastoma multiforme (GBM). METHODS AND MATERIALS: Twenty-four patients with newly diagnosed GBM were enrolled. The patients received standard external beam regional RT with concurrent TMZ beginning 3 to 6 weeks after surgery, followed by adjuvant TMZ and bortezomib for ≤24 cycles or until tumor progression. During RT, bortezomib was given at 1.3 mg/m2 on days 1, 4, 8, 11, 29, 32, 36, and 39. After RT, bortezomib was given at 1.3 mg/m2 on days 1, 4, 8, and 11 every 4 weeks.
RESULTS: No unexpected adverse events occurred from the addition of bortezomib. The efficacy analysis showed a median progression-free survival (PFS) of 6.2 months (95% confidence interval [CI] 3.7-8.8), with promising PFS rates at ≥18 months compared with historical norms (25.0% at 18 and 24 months; 16.7% at 30 months). In terms of overall survival (OS), the median OS was 19.1 months (95% CI 6.7-31.4), with improved OS rates at ≥12 months (87.5% at 12, 50.0% at 24, 34.1% at 36-60 months) compared with the historical norms. The median PFS was 24.7 months (95% CI 8.5-41.0) in 10 MGMT methylated and 5.1 months (95% CI 3.9-6.2) in 13 unmethylated patients. The estimated median OS was 61 months (95% CI upper bound not reached) in the methylated and 16.4 months (95% CI 11.8-21.0) in the unmethylated patients.
CONCLUSIONS: The addition of bortezomib to current standard radiochemotherapy in newly diagnosed GBM patients was tolerable. The PFS and OS rates appeared promising, with more benefit to MGMT methylated patients. Further clinical investigation is warranted in a larger cohort of patients.
Copyright © 2018 Elsevier Inc. All rights reserved.

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Year:  2018        PMID: 29722661      PMCID: PMC6277207          DOI: 10.1016/j.ijrobp.2018.01.001

Source DB:  PubMed          Journal:  Int J Radiat Oncol Biol Phys        ISSN: 0360-3016            Impact factor:   7.038


  20 in total

1.  Updated response assessment criteria for high-grade gliomas: response assessment in neuro-oncology working group.

Authors:  Patrick Y Wen; David R Macdonald; David A Reardon; Timothy F Cloughesy; A Gregory Sorensen; Evanthia Galanis; John Degroot; Wolfgang Wick; Mark R Gilbert; Andrew B Lassman; Christina Tsien; Tom Mikkelsen; Eric T Wong; Marc C Chamberlain; Roger Stupp; Kathleen R Lamborn; Michael A Vogelbaum; Martin J van den Bent; Susan M Chang
Journal:  J Clin Oncol       Date:  2010-03-15       Impact factor: 44.544

2.  NFKBIA deletion in glioblastomas.

Authors:  Markus Bredel; Denise M Scholtens; Ajay K Yadav; Angel A Alvarez; Jaclyn J Renfrow; James P Chandler; Irene L Y Yu; Maria S Carro; Fangping Dai; Michael J Tagge; Roberto Ferrarese; Claudia Bredel; Heidi S Phillips; Paul J Lukac; Pierre A Robe; Astrid Weyerbrock; Hannes Vogel; Steven Dubner; Bret Mobley; Xiaolin He; Adrienne C Scheck; Branimir I Sikic; Kenneth D Aldape; Arnab Chakravarti; Griffith R Harsh
Journal:  N Engl J Med       Date:  2010-12-22       Impact factor: 91.245

3.  Activity of bortezomib in glioblastoma.

Authors:  Jan Styczynski; Dorota Olszewska-Slonina; Beata Kolodziej; Malgorzata Napieraj; Mariusz Wysocki
Journal:  Anticancer Res       Date:  2006 Nov-Dec       Impact factor: 2.480

4.  Subcutaneous versus intravenous administration of bortezomib in patients with relapsed multiple myeloma: a randomised, phase 3, non-inferiority study.

Authors:  Philippe Moreau; Halyna Pylypenko; Sebastian Grosicki; Ievgenii Karamanesht; Xavier Leleu; Maria Grishunina; Grigoriy Rekhtman; Zvenyslava Masliak; Tadeusz Robak; Anna Shubina; Bertrand Arnulf; Martin Kropff; James Cavet; Dixie-Lee Esseltine; Huaibao Feng; Suzette Girgis; Helgi van de Velde; William Deraedt; Jean-Luc Harousseau
Journal:  Lancet Oncol       Date:  2011-04-18       Impact factor: 41.316

Review 5.  Bortezomib as the first proteasome inhibitor anticancer drug: current status and future perspectives.

Authors:  D Chen; M Frezza; S Schmitt; J Kanwar; Q P Dou
Journal:  Curr Cancer Drug Targets       Date:  2011-03       Impact factor: 3.428

6.  Bortezomib primes glioblastoma, including glioblastoma stem cells, for TRAIL by increasing tBid stability and mitochondrial apoptosis.

Authors:  Thomas Unterkircher; Silvia Cristofanon; Sri Hari Krishna Vellanki; Lisa Nonnenmacher; Georg Karpel-Massler; Christian Rainer Wirtz; Klaus-Michael Debatin; Simone Fulda
Journal:  Clin Cancer Res       Date:  2011-04-27       Impact factor: 12.531

7.  Bevacizumab plus radiotherapy-temozolomide for newly diagnosed glioblastoma.

Authors:  Olivier L Chinot; Wolfgang Wick; Warren Mason; Roger Henriksson; Frank Saran; Ryo Nishikawa; Antoine F Carpentier; Khe Hoang-Xuan; Petr Kavan; Dana Cernea; Alba A Brandes; Magalie Hilton; Lauren Abrey; Timothy Cloughesy
Journal:  N Engl J Med       Date:  2014-02-20       Impact factor: 91.245

8.  A randomized trial of bevacizumab for newly diagnosed glioblastoma.

Authors:  Mark R Gilbert; James J Dignam; Terri S Armstrong; Jeffrey S Wefel; Deborah T Blumenthal; Michael A Vogelbaum; Howard Colman; Arnab Chakravarti; Stephanie Pugh; Minhee Won; Robert Jeraj; Paul D Brown; Kurt A Jaeckle; David Schiff; Volker W Stieber; David G Brachman; Maria Werner-Wasik; Ivo W Tremont-Lukats; Erik P Sulman; Kenneth D Aldape; Walter J Curran; Minesh P Mehta
Journal:  N Engl J Med       Date:  2014-02-20       Impact factor: 91.245

9.  Proteasome inhibition with bortezomib induces cell death in GBM stem-like cells and temozolomide-resistant glioma cell lines, but stimulates GBM stem-like cells' VEGF production and angiogenesis.

Authors:  Daniela A Bota; Daniela Alexandru; Stephen T Keir; Darell Bigner; James Vredenburgh; Henry S Friedman
Journal:  J Neurosurg       Date:  2013-10-04       Impact factor: 5.115

10.  Bortezomib overcomes MGMT-related resistance of glioblastoma cell lines to temozolomide in a schedule-dependent manner.

Authors:  Panagiotis J Vlachostergios; Eleana Hatzidaki; Christina D Befani; Panagiotis Liakos; Christos N Papandreou
Journal:  Invest New Drugs       Date:  2013-05-05       Impact factor: 3.850

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  13 in total

1.  G3BP1 knockdown sensitizes U87 glioblastoma cell line to Bortezomib by inhibiting stress granules assembly and potentializing apoptosis.

Authors:  L F F Bittencourt; G L Negreiros-Lima; L P Sousa; A G Silva; I B S Souza; R I M A Ribeiro; M F Dutra; R F Silva; A C F Dias; F M Soriani; W K Martins; L S Barcelos
Journal:  J Neurooncol       Date:  2019-08-07       Impact factor: 4.130

Review 2.  Radiosensitizers in the temozolomide era for newly diagnosed glioblastoma.

Authors:  Peter Mathen; Lindsay Rowe; Megan Mackey; DeeDee Smart; Philip Tofilon; Kevin Camphausen
Journal:  Neurooncol Pract       Date:  2019-11-30

3.  Corilagin induces human glioblastoma U251 cell apoptosis by impeding activity of (immuno)proteasome.

Authors:  Xianyun Qin; Jilan Liu; Dongfeng Pan; Wenyuan Ma; Panpan Cheng; Feng Jin
Journal:  Oncol Rep       Date:  2021-03-02       Impact factor: 3.906

Review 4.  Potential roads for reaching the summit: an overview on target therapies for high-grade gliomas.

Authors:  Alice Giotta Lucifero; Sabino Luzzi; Ilaria Brambilla; Lucia Schena; Mario Mosconi; Thomas Foiadelli; Salvatore Savasta
Journal:  Acta Biomed       Date:  2020-06-30

5.  Revealing Temozolomide Resistance Mechanisms via Genome-Wide CRISPR Libraries.

Authors:  Clarissa Ribeiro Reily Rocha; Alexandre Reily Rocha; Matheus Molina Silva; Luciana Rodrigues Gomes; Marcela Teatin Latancia; Marina Andrade Tomaz; Izadora de Souza; Linda Karolynne Seregni Monteiro; Carlos Frederico Martins Menck
Journal:  Cells       Date:  2020-12-01       Impact factor: 6.600

6.  Comprehensive Molecular Analyses of a Novel Mutational Signature Classification System with Regard to Prognosis, Genomic Alterations, and Immune Landscape in Glioma.

Authors:  Zaoqu Liu; Taoyuan Lu; Libo Wang; Long Liu; Lifeng Li; Xinwei Han
Journal:  Front Mol Biosci       Date:  2021-07-07

Review 7.  Glioblastoma: Pathogenesis and Current Status of Chemotherapy and Other Novel Treatments.

Authors:  Vilashini Rajaratnam; Mohammad Mohiminul Islam; Maixee Yang; Rachel Slaby; Hilda Martinez Ramirez; Shama Parveen Mirza
Journal:  Cancers (Basel)       Date:  2020-04-10       Impact factor: 6.639

8.  Bortezomib inhibits growth and sensitizes glioma to temozolomide (TMZ) via down-regulating the FOXM1-Survivin axis.

Authors:  Jun-Hai Tang; Lin Yang; Ju-Xiang Chen; Qing-Rui Li; Li-Rong Zhu; Qing-Fu Xu; Guo-Hao Huang; Zuo-Xin Zhang; Yan Xiang; Lei Du; Zheng Zhou; Sheng-Qing Lv
Journal:  Cancer Commun (Lond)       Date:  2019-12-03

Review 9.  Radioresistance in Glioblastoma and the Development of Radiosensitizers.

Authors:  Md Yousuf Ali; Claudia R Oliva; Abu Shadat M Noman; Bryan G Allen; Prabhat C Goswami; Yousef Zakharia; Varun Monga; Douglas R Spitz; John M Buatti; Corinne E Griguer
Journal:  Cancers (Basel)       Date:  2020-09-03       Impact factor: 6.639

Review 10.  Small-molecule drug repurposing to target DNA damage repair and response pathways.

Authors:  Jacqueline A Brinkman; Yue Liu; Stephen J Kron
Journal:  Semin Cancer Biol       Date:  2020-02-27       Impact factor: 15.707

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