Literature DB >> 29675680

A randomized, double-blind, phase 2 study of ruxolitinib or placebo in combination with capecitabine in patients with advanced HER2-negative breast cancer and elevated C-reactive protein, a marker of systemic inflammation.

Joyce O'Shaughnessy1, Angela DeMichele2, Cynthia X Ma3, Paul Richards4, Denise A Yardley5, Gail Shaw Wright6, Kevin Kalinsky7, Ronald Steis8, Sami Diab9, Gerard Kennealey10, Ryan Geschwindt10, Wei Jiang10, Hope S Rugo11.   

Abstract

PURPOSE: The Janus-associated kinase (JAK)/signal transducer and activator of transcription pathway is a key regulator of inflammatory signaling, associated with tumorigenesis, cell survival, and progression. This randomized phase 2 trial evaluated the efficacy and safety of the addition of ruxolitinib, a JAK1/JAK2 inhibitor, to capecitabine in patients with HER2-negative advanced breast cancer and high systemic inflammation (modified Glasgow Prognostic Score [mGPS] ≥ 1).
METHODS: Patients with ≤ 2 prior chemotherapy regimens for advanced or metastatic disease or hormone receptor-positive patients with disease progression on prior hormonal therapies were randomized 1:1 to 21-day cycles of ruxolitinib (n = 76) or placebo (n = 73) plus capecitabine. The primary endpoint was overall survival (OS).
RESULTS: Baseline characteristics were well balanced between groups. For ruxolitinib plus capecitabine versus placebo plus capecitabine, median OS was 11.2 months versus 10.9 months (log-rank test P = 0.762); median progression-free survival (PFS) was 4.5 months versus 2.5 months (log-rank test P = 0.151); and overall response rate (ORR) was 28.9% versus 13.7% (Cochran-Mantel-Haenszel test P = 0.024), respectively. A more favorable change in health-related quality of life (HRQoL) was observed with ruxolitinib plus capecitabine versus placebo plus capecitabine. Both regimens were generally tolerable. A higher incidence of grade 3/4 anemia (25.4% vs 5.6%) and a lower incidence of grade 3/4 palmar-plantar erythrodysesthesia (1.4% vs 12.7%) occurred with ruxolitinib plus capecitabine versus placebo plus capecitabine.
CONCLUSIONS: The addition of ruxolitinib to capecitabine for patients with advanced breast cancer and high systemic inflammation was generally tolerable; ORR was numerically greater, a more favorable change in HRQoL was observed, but neither OS nor PFS was improved compared with placebo plus capecitabine.

Entities:  

Keywords:  Advanced HER2-negative; Breast cancer; Capecitabine; Phase 2; Randomized study; Ruxolitinib

Mesh:

Substances:

Year:  2018        PMID: 29675680     DOI: 10.1007/s10549-018-4770-6

Source DB:  PubMed          Journal:  Breast Cancer Res Treat        ISSN: 0167-6806            Impact factor:   4.872


  15 in total

Review 1.  JAK-STAT signaling in human disease: From genetic syndromes to clinical inhibition.

Authors:  Yiming Luo; Madison Alexander; Massimo Gadina; John J O'Shea; Francoise Meylan; Daniella M Schwartz
Journal:  J Allergy Clin Immunol       Date:  2021-10       Impact factor: 14.290

Review 2.  Biomarkers in Triple-Negative Breast Cancer: State-of-the-Art and Future Perspectives.

Authors:  Stefania Cocco; Michela Piezzo; Alessandra Calabrese; Daniela Cianniello; Roberta Caputo; Vincenzo Di Lauro; Giuseppina Fusco; Germira di Gioia; Marina Licenziato; Michelino De Laurentiis
Journal:  Int J Mol Sci       Date:  2020-06-27       Impact factor: 5.923

3.  Effects of systemic inflammation on relapse in early breast cancer.

Authors:  Nicholas P McAndrew; Lisa Bottalico; Clementina Mesaros; Ian A Blair; Patricia Y Tsao; Jennifer M Rosado; Tapan Ganguly; Sarah J Song; Phyllis A Gimotty; Jun J Mao; Angela DeMichele
Journal:  NPJ Breast Cancer       Date:  2021-01-22

Review 4.  Recent Discoveries of Macromolecule- and Cell-Based Biomarkers and Therapeutic Implications in Breast Cancer.

Authors:  Hsing-Ju Wu; Pei-Yi Chu
Journal:  Int J Mol Sci       Date:  2021-01-10       Impact factor: 5.923

5.  Targeting the JAK/STAT pathway in solid tumors.

Authors:  Zoya Qureshy; Daniel E Johnson; Jennifer R Grandis
Journal:  J Cancer Metastasis Treat       Date:  2020-08-21

6.  C-reactive protein as an effector molecule in Covid-19 pathogenesis.

Authors:  Jesús A Mosquera-Sulbaran; Adriana Pedreañez; Yenddy Carrero; Diana Callejas
Journal:  Rev Med Virol       Date:  2021-02-17       Impact factor: 11.043

7.  Molecular Spectra and Frequency Patterns of Somatic Mutations in Arab Women with Breast Cancer.

Authors:  Humaid O Al-Shamsi; Ibrahim Abu-Gheida; Ahmed S Abdulsamad; Aydah AlAwadhi; Sadir Alrawi; Khaled M Musallam; Banu Arun; Nuhad K Ibrahim
Journal:  Oncologist       Date:  2021-08-14

8.  Genetically Predicted C-Reactive Protein Associated With Postmenopausal Breast Cancer Risk: Interrelation With Estrogen and Cancer Molecular Subtypes Using Mendelian Randomization.

Authors:  Su Yon Jung; Jeanette C Papp; Eric M Sobel; Matteo Pellegrini; Herbert Yu; Zuo-Feng Zhang
Journal:  Front Oncol       Date:  2021-02-03       Impact factor: 6.244

Review 9.  Proteomimetics of Natural Regulators of JAK-STAT Pathway: Novel Therapeutic Perspectives.

Authors:  Sara La Manna; Ilaria De Benedictis; Daniela Marasco
Journal:  Front Mol Biosci       Date:  2022-01-03

10.  The Relationship between Leptin, the Leptin Receptor and FGFR1 in Primary Human Breast Tumors.

Authors:  Wyatt Boothby-Shoemaker; Vanessa Benham; Shreya Paithankar; Rama Shankar; Bin Chen; Jamie J Bernard
Journal:  Cells       Date:  2020-10-01       Impact factor: 6.600

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