Literature DB >> 29655834

Metformin Use Is Associated With Longer Progression-Free Survival of Patients With Diabetes and Pancreatic Neuroendocrine Tumors Receiving Everolimus and/or Somatostatin Analogues.

Sara Pusceddu1, Claudio Vernieri2, Massimo Di Maio3, Riccardo Marconcini4, Francesca Spada5, Sara Massironi6, Toni Ibrahim7, Maria Pia Brizzi8, Davide Campana9, Antongiulio Faggiano10, Dario Giuffrida11, Maria Rinzivillo12, Sara Cingarlini13, Francesca Aroldi14, Lorenzo Antonuzzo15, Rossana Berardi16, Laura Catena17, Chiara De Divitiis18, Paola Ermacora19, Vittorio Perfetti20, Annalisa Fontana21, Paola Razzore22, Carlo Carnaghi23, Maria Vittoria Davì24, Carolina Cauchi25, Marilina Duro26, Sergio Ricci4, Nicola Fazio5, Federica Cavalcoli6, Alberto Bongiovanni7, Anna La Salvia8, Nicole Brighi9, Annamaria Colao27, Ivana Puliafito11, Francesco Panzuto12, Silvia Ortolani13, Alberto Zaniboni14, Francesco Di Costanzo15, Mariangela Torniai16, Emilio Bajetta17, Salvatore Tafuto18, Silvio Ken Garattini19, Daniela Femia28, Natalie Prinzi28, Laura Concas28, Giuseppe Lo Russo29, Massimo Milione28, Luca Giacomelli30, Roberto Buzzoni28, Gianfranco Delle Fave12, Vincenzo Mazzaferro31, Filippo de Braud31.   

Abstract

BACKGROUND & AIMS: Metformin seems to have anticancer effects. However, it is not clear whether use of glycemia and metformin affect outcomes of patients with advanced pancreatic neuroendocrine tumors (pNETs). We investigated the association between glycemia and progression-free survival (PFS) of patients with pNETs treated with everolimus and/or somatostatin analogues, as well as the association between metformin use and PFS time.
METHODS: We performed a retrospective analysis of 445 patients with advanced pNET treated at 24 medical centers in Italy from 1999 through 2015. Data on levels of glycemia were collected at time of diagnosis of pNET, before treatment initiation, and during treatment with everolimus (with or without somatostatin analogues), octreotide, or lanreotide. Diabetes was defined as prior or current use of glycemia control medication and/or fasting plasma glucose level ≥ 126 mg/dL, hemoglobin A1c ≥ 6.5% (48 mmol/L), or a random sample of plasma glucose ≥ 200 mg/dL (11.1 mmol/L), with reported classic symptoms of hyperglycemia or hyperglycemic crisis. Patients were assigned to groups based on diagnosis of diabetes before or during antitumor therapy. PFS was compared between patients with vs without diabetes. Among patients with diabetes, the association between metformin use and PFS was assessed. We performed sensitivity and landmark analyses to exclude patients who developed diabetes while receiving cancer treatment and to exclude a potential immortal time bias related to metformin intake.
RESULTS: PFS was significantly longer in patients with diabetes (median, 32.0 months) than without diabetes (median, 15.1 months) (hazard ratio for patients with vs without diabetes, 0.63; 95% confidence interval, 0.50-0.80; P = .0002). PFS of patients treated with metformin was significantly longer (median PFS, 44.2 months) than for patients without diabetes (hazard ratio for survival of patients with diabetes receiving metformin vs without diabetes, 0.45; 95% confidence interval, 0.32-0.62; P < .00001) and longer than for patients with diabetes receiving other treatments (median PFS, 20.8 months; hazard ratio, 0.49; 95% confidence interval, 0.34-0.69; P < .0001). In multivariable analysis, adjusted for other factors associated with outcomes, metformin was associated with longer PFS but level of glycemia was not. Metformin was associated with increased PFS of patients receiving somatostatin analogues and in those receiving everolimus, with or without somatostatin analogues. Sensitivity and landmark analyses produced similar results.
CONCLUSIONS: In a retrospective study of patients with pNETs, we found a significant association between metformin use and longer PFS.
Copyright © 2018 AGA Institute. Published by Elsevier Inc. All rights reserved.

Entities:  

Keywords:  Chemoprevention; Drug; Insulin Resistance; Pancreas

Mesh:

Substances:

Year:  2018        PMID: 29655834     DOI: 10.1053/j.gastro.2018.04.010

Source DB:  PubMed          Journal:  Gastroenterology        ISSN: 0016-5085            Impact factor:   22.682


  20 in total

Review 1.  The role of an anti-diabetic drug metformin in the treatment of endocrine tumors.

Authors:  Shilpa Thakur; Brianna Daley; Joanna Klubo-Gwiezdzinska
Journal:  J Mol Endocrinol       Date:  2019-08       Impact factor: 5.098

2.  Hyperglycemia is associated with adverse prognosis in patients with pancreatic neuroendocrine neoplasms.

Authors:  Pin Zhang; Zhiwen Xiao; Huaxiang Xu; Xinzhe Zhu; Lei Wang; Dan Huang; Yun Liang; Quanxing Ni; Jie Chen; Xianjun Yu; Guopei Luo
Journal:  Endocrine       Date:  2022-07-05       Impact factor: 3.925

3.  METNET: a phase II trial of metformin in patients with well-differentiated neuroendocrine tumours.

Authors:  João Glasberg; Aley Talans; Thomás Rivelli Giollo; Débora Zachello Recchimuzzi; João Evangelista Bezerra Neto; Rossana Veronica Mendonza Lopez; Paulo Marcelo Gehm Hoff; Rachel P Riechelmann
Journal:  Ecancermedicalscience       Date:  2022-03-31

4.  Survival of Patients With Gastroenteropancreatic Neuroendocrine Tumors and Diabetes Mellitus.

Authors:  Sahityasri Thapi; Kiwoon Baeg; Michelle K Kim; Emily J Gallagher
Journal:  Pancreas       Date:  2021-10-01       Impact factor: 3.243

5.  Impact of Metformin Use and Diabetic Status During Adjuvant Fluoropyrimidine-Oxaliplatin Chemotherapy on the Outcome of Patients with Resected Colon Cancer: A TOSCA Study Subanalysis.

Authors:  Claudio Vernieri; Fabio Galli; Laura Ferrari; Paolo Marchetti; Sara Lonardi; Evaristo Maiello; Rosario V Iaffaioli; Maria G Zampino; Alberto Zaniboni; Sabino De Placido; Maria Banzi; Azzurra Damiani; Daris Ferrari; Gerardo Rosati; Roberto F Labianca; Paolo Bidoli; Giovanni L Frassineti; Mario Nicolini; Lorenzo Pavesi; Maria C Tronconi; Angela Buonadonna; Sabrina Ferrario; Giovanni Lo Re; Vincenzo Adamo; Emiliano Tamburini; Mario Clerico; Paolo Giordani; Francesco Leonardi; Sandro Barni; Andrea Ciarlo; Luigi Cavanna; Stefania Gori; Saverio Cinieri; Marina Faedi; Massimo Aglietta; Maria Antista; Katia F Dotti; Francesca Galli; Maria Di Bartolomeo
Journal:  Oncologist       Date:  2019-01-03

6.  Octreotide long-acting release (LAR) in combination with other therapies for treatment of neuroendocrine neoplasia: a systematic review.

Authors:  Maria Rinzivillo; Ilaria De Felice; Ludovica Magi; Bruno Annibale; Francesco Panzuto
Journal:  J Gastrointest Oncol       Date:  2021-04

Review 7.  Repurposing metformin for the treatment of gastrointestinal cancer.

Authors:  Ademar Dantas Cunha Júnior; Arinilda Campos Bragagnoli; Felipe Osório Costa; José Barreto Campello Carvalheira
Journal:  World J Gastroenterol       Date:  2021-05-07       Impact factor: 5.742

Review 8.  Pleiotropic Effects of Metformin on Cancer.

Authors:  Hans-Juergen Schulten
Journal:  Int J Mol Sci       Date:  2018-09-20       Impact factor: 5.923

Review 9.  Novel application of metformin combined with targeted drugs on anticancer treatment.

Authors:  Jun Deng; Mei Peng; Zhiren Wang; Sichun Zhou; Di Xiao; Jiating Deng; Xue Yang; Jingyuan Peng; Xiaoping Yang
Journal:  Cancer Sci       Date:  2018-11-28       Impact factor: 6.716

10.  Implications of neuroendocrine tumor and diabetes mellitus on patient outcomes and care: a matched case-control study.

Authors:  Yael N Kusne; Heidi E Kosiorek; Matthew R Buras; Patricia M Verona; Kyle E Coppola; Kelley A Rone; Curtiss B Cook; Nina J Karlin
Journal:  Future Sci OA       Date:  2021-02-15
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