Literature DB >> 29653820

Afatinib as First-line Treatment of Older Patients With EGFR Mutation-Positive Non-Small-Cell Lung Cancer: Subgroup Analyses of the LUX-Lung 3, LUX-Lung 6, and LUX-Lung 7 Trials.

Yi-Long Wu1, Lecia V Sequist2, Eng-Huat Tan3, Sarayut L Geater4, Sergey Orlov5, Li Zhang6, Ki Hyeong Lee7, Chun-Ming Tsai8, Terufumi Kato9, Carlos H Barrios10, Martin Schuler11, Vera Hirsh12, Nobuyuki Yamamoto13, Kenneth O'Byrne14, Michael Boyer15, Tony Mok16, Barbara Peil17, Angela Märten17, James Chih-Hsin Yang18, Luis Paz-Ares19, Keunchil Park20.   

Abstract

BACKGROUND: Afatinib is approved in the US, Europe, and several other regions for first-line treatment for epidermal growth factor receptor mutation-positive (EGFRm+) non-small-cell lung cancer (NSCLC). PATIENTS AND METHODS: Treatment-naive patients with advanced EGFRm+ NSCLC were randomized to afatinib (40 mg/d) versus cisplatin/pemetrexed (LUX-Lung 3 [LL3]) or cisplatin/gemcitabine (LUX-Lung 6 [LL6]), or versus gefitinib (250 mg/d; LUX-Lung 7 [LL7]). We report subgroup analyses according to age, including 65 years or older versus younger than 65 years (preplanned; LL3/LL6) and additional cutoffs up to 75 years and older (exploratory; LL7). Progression-free survival (PFS), overall survival (OS), and adverse events (AEs) were evaluated.
RESULTS: Among the 134 of 345 (39%) and 86 of 364 (24%) patients aged 65 years and older in LL3 and LL6, median PFS was improved with afatinib versus chemotherapy (LL3: hazard ratio [HR], 0.64 [95% confidence interval (CI), 0.39-1.03]; LL6: HR, 0.16 [95% CI, 0.07-0.39]). Afatinib significantly improved OS versus chemotherapy in elderly patients with Del19+ NSCLC in LL3 (HR, 0.39 [95% CI, 0.19-0.80]). Among the 40 of 319 patients (13%) aged 75 years or older in LL7, median PFS (HR, 0.69 [95% CI, 0.33-1.44]) favored afatinib, consistent with the overall population. Afatinib-associated AEs in older patients were consistent with the overall populations.
CONCLUSIONS: Subgroup analyses of the LL3, LL6, and LL7 trials show that afatinib is an effective and tolerable treatment for patients with EGFRm+ NSCLC, independent of age.
Copyright © 2018 The Authors. Published by Elsevier Inc. All rights reserved.

Entities:  

Keywords:  EGFR blocker; Elderly; Gefitinib; NSCLC; Tyrosine kinase inhibitor

Mesh:

Substances:

Year:  2018        PMID: 29653820     DOI: 10.1016/j.cllc.2018.03.009

Source DB:  PubMed          Journal:  Clin Lung Cancer        ISSN: 1525-7304            Impact factor:   4.785


  21 in total

Review 1.  Afatinib as First-Line Treatment in Asian Patients with EGFR Mutation-Positive NSCLC: A Narrative Review of Real-World Evidence.

Authors:  Shun Lu; Jin-Yuan Shih; Tae-Won Jang; Chong-Kin Liam; Yongfeng Yu
Journal:  Adv Ther       Date:  2021-03-17       Impact factor: 3.845

2.  Risk Factors for Severe Diarrhea with an Afatinib Treatment of Non-Small Cell Lung Cancer: A Pooled Analysis of Clinical Trials.

Authors:  Ashley M Hopkins; Anh-Minh Nguyen; Christos S Karapetis; Andrew Rowland; Michael J Sorich
Journal:  Cancers (Basel)       Date:  2018-10-15       Impact factor: 6.639

Review 3.  A Review of Recent Advances in the Treatment of Elderly and Poor Performance NSCLC.

Authors:  Juliet A Carmichael; Daisy Wing-San Mak; Mary O'Brien
Journal:  Cancers (Basel)       Date:  2018-07-18       Impact factor: 6.639

4.  Immunogenicity of Del19 EGFR mutations in Chinese patients affected by lung adenocarcinoma.

Authors:  Deng Pan; Dapeng Zhou; Weijing Cai; Weibo Wu; Wen Ling Tan; Caicun Zhou; Yanyan Lou
Journal:  BMC Immunol       Date:  2019-11-13       Impact factor: 3.615

Review 5.  MicroRNAs in non-small cell lung cancer: Gene regulation, impact on cancer cellular processes, and therapeutic potential.

Authors:  Hannah Petrek; Ai-Ming Yu
Journal:  Pharmacol Res Perspect       Date:  2019-12

Review 6.  First-Line Treatment of Metastatic Non-Small Cell Lung Cancer in the Elderly.

Authors:  Tania Losanno; Cesare Gridelli
Journal:  Curr Oncol Rep       Date:  2021-08-03       Impact factor: 5.075

7.  Afatinib in EGFR TKI-Naïve Patients with Locally Advanced or Metastatic EGFR Mutation-Positive Non-Small Cell Lung Cancer: A Pooled Analysis of Three Phase IIIb Studies.

Authors:  Antonio Passaro; Filippo de Marinis; Hai-Yan Tu; Konstantin K Laktionov; Jifeng Feng; Artem Poltoratskiy; Jun Zhao; Eng Huat Tan; Maya Gottfried; Victor Lee; Dariusz Kowalski; Cheng Ta Yang; B J Srinivasa; Laura Clementi; Tejaswini Jalikop; Dennis Chin Lun Huang; Agnieszka Cseh; Keunchil Park; Yi-Long Wu
Journal:  Front Oncol       Date:  2021-07-09       Impact factor: 6.244

8.  Microwave hyperthermia promotes caspase‑3-dependent apoptosis and induces G2/M checkpoint arrest via the ATM pathway in non‑small cell lung cancer cells.

Authors:  Yan-Yan Zhao; Qiong Wu; Zhi-Bing Wu; Jing-Jing Zhang; Lu-Cheng Zhu; Yang Yang; Sheng-Lin Ma; Shi-Rong Zhang
Journal:  Int J Oncol       Date:  2018-06-13       Impact factor: 5.650

Review 9.  Second-generation EGFR and ErbB tyrosine kinase inhibitors as first-line treatments for non-small cell lung cancer.

Authors:  Shouzheng Wang; Junling Li
Journal:  Onco Targets Ther       Date:  2019-08-15       Impact factor: 4.147

10.  Adverse event profiles of epidermal growth factor receptor-tyrosine kinase inhibitors in cancer patients: A systematic review and meta-analysis.

Authors:  Xiaonan Yin; Zhou Zhao; Yuan Yin; Chaoyong Shen; Xin Chen; Zhaolun Cai; Jian Wang; Zhixin Chen; Yiqiong Yin; Bo Zhang
Journal:  Clin Transl Sci       Date:  2021-01-25       Impact factor: 4.689

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