Literature DB >> 29630869

Can inhibition of retinoic acid biosynthesis function as a non-hormonal female contraceptive?

Jisun Paik1, Piper M Treuting2, Michael Haenisch2, John K Amory3.   

Abstract

OBJECTIVE: Vitamin A deficient females have reduced fertility due to decreased retinoic acid production. WIN 18,446 inhibits retinoic acid biosynthesis and functions as a contraceptive in males. We tested whether WIN 18,446 treatment would suppress fertility in female mice. STUDY
DESIGN: Female mice were treated with WIN 18,446 and mated. Pregnancy rates were compared using Fisher's exact test.
RESULTS: WIN 18,446 reduced pregnancy compared with control (p=.03). However, one animal became pregnant with malformed embryos.
CONCLUSIONS: WIN 18,446 treatment significantly reduces fecundity, but teratogenicity in the setting of contraceptive failure limits the appeal of this approach to female contraception.
Copyright © 2018 Elsevier Inc. All rights reserved.

Entities:  

Keywords:  aldehyde dehydrogenase 1A; enzyme inhibitor; pregnancy; retinoic acid

Year:  2018        PMID: 29630869      PMCID: PMC6174106          DOI: 10.1016/j.contraception.2018.03.035

Source DB:  PubMed          Journal:  Contraception        ISSN: 0010-7824            Impact factor:   3.375


  9 in total

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Authors:  P Taleporos; M P Salgo; G Oster
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2.  Meiosis initiation in the human ovary requires intrinsic retinoic acid synthesis.

Authors:  R Le Bouffant; M J Guerquin; C Duquenne; N Frydman; H Coffigny; V Rouiller-Fabre; R Frydman; R Habert; G Livera
Journal:  Hum Reprod       Date:  2010-07-29       Impact factor: 6.918

3.  Retinoic Acid Regulates Calcium Signaling to Promote Mouse Ovarian Granulosa Cell Proliferation.

Authors:  Michael Demczuk; Huiya Huang; Carl White; Jingjing L Kipp
Journal:  Biol Reprod       Date:  2016-08-03       Impact factor: 4.285

4.  Embryocidal action of a bis(dichloroacetyl)-diamine: an oral abortifacient for rats.

Authors:  G Oster; M P Salgo; P Taleporos
Journal:  Am J Obstet Gynecol       Date:  1974-07-01       Impact factor: 8.661

Review 5.  Nonsteroid nuclear receptors: what are genetic studies telling us about their role in real life?

Authors:  P Kastner; M Mark; P Chambon
Journal:  Cell       Date:  1995-12-15       Impact factor: 41.582

6.  Inhibition of retinoic acid biosynthesis by the bisdichloroacetyldiamine WIN 18,446 markedly suppresses spermatogenesis and alters retinoid metabolism in mice.

Authors:  Jisun Paik; Michael Haenisch; Charles H Muller; Alex S Goldstein; Samuel Arnold; Nina Isoherranen; Thea Brabb; Piper M Treuting; John K Amory
Journal:  J Biol Chem       Date:  2014-04-07       Impact factor: 5.157

7.  Suppression of spermatogenesis by bisdichloroacetyldiamines is mediated by inhibition of testicular retinoic acid biosynthesis.

Authors:  John K Amory; Charles H Muller; Jakob A Shimshoni; Nina Isoherranen; Jisun Paik; Jan S Moreb; David W Amory; Ryan Evanoff; Alex S Goldstein; Michael D Griswold
Journal:  J Androl       Date:  2010-08-12

Review 8.  The role of vitamin A in mammalian reproduction and embryonic development.

Authors:  Margaret Clagett-Dame; Hector F DeLuca
Journal:  Annu Rev Nutr       Date:  2002       Impact factor: 11.848

9.  De Novo-Synthesized Retinoic Acid in Ovarian Antral Follicles Enhances FSH-Mediated Ovarian Follicular Cell Differentiation and Female Fertility.

Authors:  Tomoko Kawai; Noriyuki Yanaka; JoAnne S Richards; Masayuki Shimada
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  9 in total

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