Literature DB >> 29605835

Microwave-assisted green synthesis of 4,5-dihydro-1H-pyrazole-1-carbothioamides in water.

Hamid Reza Farmani1, Mohammad Hossein Mosslemin2, Bahareh Sadeghi2.   

Abstract

Rapid, efficient, simple and green procedure for the synthesis of 4,5-dihydro-1H-pyrazole-1-carbothioamides via the multicomponent reaction of aryl aldehydes, acetophenones and thiosemicarbazide in water in the presence of tetrabutylammonium hydroxide under microwave irradiation is reported.

Entities:  

Keywords:  4,5-Dihydro-1H-pyrazole-1-carbothioamides; Green chemistry; MCRs; Microwave irradiation; Multicomponent reaction; TBAOH; Water

Mesh：

Substances：

Year:  2018        PMID： 29605835     DOI： 10.1007/s11030-018-9814-7

Source DB:  PubMed          Journal:  Mol Divers        ISSN： 1381-1991            Impact factor:   2.943


  28 in total

Review 1.  Microwave-assisted synthesis in water as solvent.

Authors:  Doris Dallinger; C Oliver Kappe
Journal:  Chem Rev       Date:  2007-04-24       Impact factor: 60.622

2.  Organic chemistry in water.

Authors:  Chao-Jun Li; Liang Chen
Journal:  Chem Soc Rev       Date:  2005-11-21       Impact factor: 54.564

3.  Synthesis and studies on antidepressant and anticonvulsant activities of some 3-(2-furyl)-pyrazoline derivatives.

Authors:  Zuhal Ozdemir; H Burak Kandilci; Bülent Gümüşel; Unsal Caliş; A Altan Bilgin
Journal:  Eur J Med Chem       Date:  2006-10-25       Impact factor: 6.514

4.  Microwave assisted synthesis of some novel 2-pyrazoline derivatives as possible antimicrobial agents.

Authors:  Rakesh Chawla; Ujjwal Sahoo; Anshu Arora; Prabodh Chander Sharma; Vijayaraj Radhakrishnan
Journal:  Acta Pol Pharm       Date:  2010 Jan-Feb       Impact factor: 0.330

5.  Synthesis, molecular modeling studies, and selective inhibitory activity against monoamine oxidase of 1-thiocarbamoyl-3,5-diaryl-4,5-dihydro-(1H)- pyrazole derivatives.

Authors:  Franco Chimenti; Elias Maccioni; Daniela Secci; Adriana Bolasco; Paola Chimenti; Arianna Granese; Olivia Befani; Paola Turini; Stefano Alcaro; Francesco Ortuso; Roberto Cirilli; Francesco La Torre; Maria C Cardia; Simona Distinto
Journal:  J Med Chem       Date:  2005-11-17       Impact factor: 7.446

Review 6.  Recent advances in bioactive pyrazoles.

Authors:  Ş Güniz Küçükgüzel; Sevil Şenkardeş
Journal:  Eur J Med Chem       Date:  2014-12-05       Impact factor: 6.514

7.  Synthesis, biological evaluation and 3D-QSAR study of novel 4,5-dihydro-1H-pyrazole thiazole derivatives as BRAF(V⁶⁰⁰E) inhibitors.

Authors:  Meng-Yue Zhao; Yong Yin; Xiao-Wei Yu; Chetan B Sangani; Shu-Fu Wang; Ai-Min Lu; Li-Fang Yang; Peng-Cheng Lv; Ming-Guo Jiang; Hai-Liang Zhu
Journal:  Bioorg Med Chem       Date:  2014-11-26       Impact factor: 3.641

Review 8.  Organic synthesis "on water".

Authors:  Arani Chanda; Valery V Fokin
Journal:  Chem Rev       Date:  2009-02       Impact factor: 60.622

9.  Synthesis and antiviral activity of new pyrazole and thiazole derivatives.

Authors:  Osama I el-Sabbagh; Mohamed M Baraka; Samy M Ibrahim; Christophe Pannecouque; Graciela Andrei; Robert Snoeck; Jan Balzarini; Adel A Rashad
Journal:  Eur J Med Chem       Date:  2009-04-05       Impact factor: 6.514

10.  Synthesis of New 3-Heteroarylindoles as Potential Anticancer Agents.

Authors:  Abdou O Abdelhamid; Sobhi M Gomha; Nadia A Abdelriheem; Saher M Kandeel
Journal:  Molecules       Date:  2016-07-16       Impact factor: 4.411
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