Literature DB >> 29482352

Dolutegravir Plus Rilpivirine as a Switch Option in cART-Experienced Patients: 96-Week Data.

Amedeo Ferdinando Capetti1, Maria Vittoria Cossu1, Gaetana Sterrantino2, Giorgio Barbarini3, Simona Di Giambenedetto4, Giuseppe Vittorio De Socio5, GianCarlo Orofino6, Antonio Di Biagio7, Benedetto M Celesia8, Stefano Rusconi1, Barbara Argenteri1, Giuliano Rizzardini1,9.   

Abstract

BACKGROUND: Data from clinical studies confirm the efficacy of switching to dolutegravir (DTG) plus rilpivirine (RPV) in selected patients.
OBJECTIVE: The primary objective is to report the 96-week virological suppression in our cohort, assessing the durability of this strategy in complicated situations. The secondary objective is to describe the safety and metabolic profile.
METHODS: All patients who had switched to DTG plus RPV between October 1, 2014, and September 30, 2015, were analyzed using a retrospective-prospective design, approved by ethics committees. Routine metabolic, immunological, and virological data were regularly sent to the coordinating center. Viral control was classified as HIV-1 RNA ≥50 copies/mL, 1 to 49 copies/mL, or undetectable (no virus detected [NVD]).
RESULTS: We followed 145 patients for a median of 101 weeks. The median age was 52 years; 31.7% were women, and 9.6% non-Caucasian; 50.3% had failed at least 1 antiretroviral regimen; and 15% had ≥50 copies/mL at baseline. The reasons for switching were as follows: simplification (51.7%), toxicity (36.5%), drug-drug interactions (6.9%), persistent low-level viremia (3.0%), nonadherence (2.1%), and viral failure (1.4%). By week 96, seven patients dropped out. At week 96, none had ≥50 HIV-1 RNA copies/mL, 138 (95.2%) had <50 copies/mL, and 123 (84.8%) had NVD. The low- to high-density lipoprotein cholesterol (LDL-C/HDL-C) ratio decreased significantly ( P = 0.04). Of the 287 baseline altered laboratory parameters, 32.7% normalized by week 96. Serum glucose and total- and LDL-cholesterol normalization were statistically significant.
CONCLUSIONS: Switching to DTG plus RPV improved viral suppression and LDL-C/HDL-C ratio.

Entities:  

Keywords:  HIV/AIDS; adverse drug reactions; antiretrovirals; drug utilization; metabolism; pharmacoeconomics

Mesh:

Substances:

Year:  2018        PMID: 29482352     DOI: 10.1177/1060028018761600

Source DB:  PubMed          Journal:  Ann Pharmacother        ISSN: 1060-0280            Impact factor:   3.154


  9 in total

Review 1.  Simplifying ARV Therapy in the Setting of Resistance.

Authors:  Neha Sheth Pandit; Daniel B Chastain; Andrea M Pallotta; Melissa E Badowski; Emily C Huesgen; Sarah M Michienzi
Journal:  Curr Infect Dis Rep       Date:  2019-09-07       Impact factor: 3.725

Review 2.  Dolutegravir/Rilpivirine: A Review in HIV-1 Infection.

Authors:  Hannah A Blair
Journal:  Drugs       Date:  2018-11       Impact factor: 11.431

Review 3.  Two-drug regimens for treatment of naïve HIV-1 infection and as maintenance therapy.

Authors:  Katya C Corado; Margaret R Caplan; Eric S Daar
Journal:  Drug Des Devel Ther       Date:  2018-11-01       Impact factor: 4.162

4.  Comparative efficacy and safety and dolutegravir and lamivudine in treatment naive HIV patients.

Authors:  Matthew Radford; Daniel C Parks; Shannon Ferrante; Yogesh Punekar
Journal:  AIDS       Date:  2019-09-01       Impact factor: 4.177

5.  Forgiveness of INSTI-Containing Regimens at Drug Concentrations Simulating Variable Adherence In Vitro.

Authors:  Rima K Acosta; Michelle L D'Antoni; Andrew Mulato; Stephen R Yant; Tomas Cihlar; Kirsten L White
Journal:  Antimicrob Agents Chemother       Date:  2022-04-07       Impact factor: 5.938

6.  Dolutegravir plus rilpivirine: benefits beyond viral suppression: DORIPEX retrospective study.

Authors:  Jesús Troya; Carlos Dueñas; Idoia Irazola; Ignacio de Los Santos; Sara de la Fuente; Desiré Gil; Cristina Hernández; María José Galindo; Julia Gómez; Elisabeth Delgado; Estela Moreno-García; Guillermo Posada; Teresa Aldámiz; Jose Antonio Iribarren; José Manuel Guerra; Miguel Ángel Morán; Carlos Galera; Javier Fuente; Ana Peláez; Miguel Cervero; María Garcinuño; Marta Montero; Francisco Ceballos; Luis Buzón
Journal:  Medicine (Baltimore)       Date:  2022-06-17       Impact factor: 1.817

Review 7.  Two's a Company, Three's a Crowd: A Review of Initiating or Switching to a Two-Drug Antiretroviral Regimen in Treatment-Naïve and Treatment-Experienced Patients Living with HIV-1.

Authors:  Melissa Badowski; Sarah E Pérez; David Silva; Andrea Lee
Journal:  Infect Dis Ther       Date:  2020-03-19

Review 8.  Non-Nucleoside Reverse Transcriptase Inhibitors Join Forces with Integrase Inhibitors to Combat HIV.

Authors:  Daniel M Himmel; Eddy Arnold
Journal:  Pharmaceuticals (Basel)       Date:  2020-06-11

9.  Cohort profile: The Observational cohort for the study of DOlutegravir in Antiretroviral Combination REgimens (ODOACRE).

Authors:  Arturo Ciccullo; Gianmaria Baldin; Amedeo Capetti; Vanni Borghi; Gaetana Sterrantino; Alessandra Latini; Giordano Madeddu; Luigi Celani; Francesca Vignale; Barbara Rossetti; Alex Dusina; Maria Vittoria Cossu; Sibilla Restelli; William Gennari; Filippo Lagi; Andrea Giacomelli; Manuela Colafigli; Lucia Brescini; Alberto Borghetti; Cristina Mussini; Stefano Rusconi; Simona Di Giambenedetto
Journal:  BMJ Open       Date:  2019-12-02       Impact factor: 2.692

  9 in total

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