Literature DB >> 29397527

Effect of roflumilast on chronic obstructive pulmonary disease: a systematic review and meta-analysis.

Lu-Fei Shen1, Xiao-Dong Lv1, Wen-Yu Chen2, Qi Yang3, Zhi-Xian Fang1, Wei-Fen Lu1.   

Abstract

BACKGROUND: Randomized controlled trials (RCTs) of roflumilast effect on chronic obstructive pulmonary disease (COPD) have been reported in the last decade. The current meta-analysis was designed to systematically review and perform meta-analysis of the RCTs of roflumilast treatment in COPD.
METHODS: Electronic databases including PubMed, EMBASE, Web of Science, and Cochrane clinical trials database were searched to identify RCTs of roflumilast treatment on COPD. The primary outcomes were effect of roflumilast on pre-bronchodilator FEV1, post-bronchodilator FEV1, and exacerbation rate. Secondary outcomes were effect of roflumilast on airway inflammation and adverse effect.
RESULTS: A total of 11 RCTs were enrolled into the current analysis. Roflumilast significantly improved both pre-bronchodilator FEV1 (standardized difference in mean ± SD was 0.621 ± 0.161; 95% CI 0.306~0.936, p < 0.001) and post-bronchodilator FEV1 (standardized difference in mean ± SD was 0.563 ± 0.149, 95% CI 0.270~0.855, p < 0.001) compared with placebo. Roflumilast also significantly reduced exacerbation of COPD (standardized difference in mean ± SD 0.099 ± 0.020, 95% CI 0.061~0.138; p < 0.001) and suppressed airway inflammation (standardized difference in mean ± SD 1.354 ± 0.260, 95% CI 0.845~1.862, p < 0.001) compared with placebo. However, roflumilast significantly increased adverse effect such as diarrhea (rate ratio 2.945, 95% CI 2.453~3.536, p < 0.001) and weight loss (rate ratio 3.814, 95% CI 3.091~4.707, p < 0.001) compared with placebo.
CONCLUSION: These findings indicated that roflumilast treatment could improve COPD patients' lung function and reduce exacerbation, and that inhibition of airway inflammation by roflumilast might contribute to the beneficial effect of PDE-4 inhibitors on COPD.

Entities:  

Keywords:  COPD; Meta-analysis; Roflumilast

Mesh:

Substances:

Year:  2018        PMID: 29397527     DOI: 10.1007/s11845-018-1738-9

Source DB:  PubMed          Journal:  Ir J Med Sci        ISSN: 0021-1265            Impact factor:   1.568


  28 in total

1.  Physiological effects of roflumilast at rest and during exercise in COPD.

Authors:  Denis E O'Donnell; Dirk Bredenbröker; Manja Brose; Katherine A Webb
Journal:  Eur Respir J       Date:  2011-09-29       Impact factor: 16.671

2.  Roflumilast with long-acting β2-agonists for COPD: influence of exacerbation history.

Authors:  E D Bateman; K F Rabe; P M A Calverley; U M Goehring; M Brose; D Bredenbröker; L M Fabbri
Journal:  Eur Respir J       Date:  2011-07-07       Impact factor: 16.671

Review 3.  Pathogenesis of COPD.

Authors:  John R Spurzem; Stephen I Rennard
Journal:  Semin Respir Crit Care Med       Date:  2005-04       Impact factor: 3.119

4.  Effect of Roflumilast and Inhaled Corticosteroid/Long-Acting β2-Agonist on Chronic Obstructive Pulmonary Disease Exacerbations (RE(2)SPOND). A Randomized Clinical Trial.

Authors:  Fernando J Martinez; Klaus F Rabe; Sanjay Sethi; Emilio Pizzichini; Andrew McIvor; Antonio Anzueto; Vijay K T Alagappan; Shahid Siddiqui; Ludmyla Rekeda; Christopher J Miller; Sofia Zetterstrand; Colin Reisner; Stephen I Rennard
Journal:  Am J Respir Crit Care Med       Date:  2016-09-01       Impact factor: 21.405

Review 5.  PDE4: a novel target in the treatment of chronic obstructive pulmonary disease.

Authors:  J M Michalski; G Golden; J Ikari; S I Rennard
Journal:  Clin Pharmacol Ther       Date:  2011-11-30       Impact factor: 6.875

6.  Reduction in sputum neutrophil and eosinophil numbers by the PDE4 inhibitor roflumilast in patients with COPD.

Authors:  Diana C Grootendorst; Stefanie A Gauw; Renate M Verhoosel; Peter J Sterk; Jeannette J Hospers; Dirk Bredenbröker; Thomas D Bethke; Pieter S Hiemstra; Klaus F Rabe
Journal:  Thorax       Date:  2007-06-15       Impact factor: 9.139

7.  Roflumilast in symptomatic chronic obstructive pulmonary disease: two randomised clinical trials.

Authors:  Peter M A Calverley; Klaus F Rabe; Udo-Michael Goehring; Søren Kristiansen; Leonardo M Fabbri; Fernando J Martinez
Journal:  Lancet       Date:  2009-08-29       Impact factor: 79.321

Review 8.  Phosphodiesterase 4 inhibitors for chronic obstructive pulmonary disease.

Authors:  Jimmy Chong; Bonnie Leung; Phillippa Poole
Journal:  Cochrane Database Syst Rev       Date:  2013-11-04

9.  Pooled subpopulation analyses of the effects of roflumilast on exacerbations and lung function in COPD.

Authors:  Nicola A Hanania; Peter M A Calverley; Mark T Dransfield; Jill P Karpel; Manja Brose; Haiyuan Zhu; Udo-Michael Goehring; Paul Rowe
Journal:  Respir Med       Date:  2013-09-30       Impact factor: 3.415

10.  No relevant cardiac, pharmacokinetic or safety interactions between roflumilast and inhaled formoterol in healthy subjects: an open-label, randomised, actively controlled study.

Authors:  Christian de Mey; Nassr Nassr; Gezim Lahu
Journal:  BMC Clin Pharmacol       Date:  2011-06-01
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  6 in total

1.  Efficacy and safety profile of roflumilast in a real-world experience.

Authors:  Aykut Cilli; Halid Bal; Hakan Gunen
Journal:  J Thorac Dis       Date:  2019-04       Impact factor: 2.895

2.  Inhibition of Recruitment and Activation of Neutrophils by Pyridazinone-Scaffold-Based Compounds.

Authors:  Aurélie Moniot; Julien Braux; Renaud Siboni; Christine Guillaume; Sandra Audonnet; Ingrid Allart-Simon; Janos Sapi; Rabindra Tirouvanziam; Stéphane Gérard; Sophie C Gangloff; Frédéric Velard
Journal:  Int J Mol Sci       Date:  2022-06-29       Impact factor: 6.208

3.  Phosphodiesterase-4 inhibitors for chronic obstructive pulmonary disease.

Authors:  Sadia Janjua; Rebecca Fortescue; Phillippa Poole
Journal:  Cochrane Database Syst Rev       Date:  2020-05-01

Review 4.  Phosphodiesterase-4 Inhibitors for the Treatment of Inflammatory Diseases.

Authors:  Heng Li; Jianping Zuo; Wei Tang
Journal:  Front Pharmacol       Date:  2018-10-17       Impact factor: 5.810

Review 5.  New putative insights into neprilysin (NEP)-dependent pharmacotherapeutic role of roflumilast in treating COVID-19.

Authors:  Manar Mohammed El Tabaa; Maram Mohammed El Tabaa
Journal:  Eur J Pharmacol       Date:  2020-10-01       Impact factor: 4.432

Review 6.  The Role of the Pharmacist in Optimizing Outcomes With Roflumilast, a PDE4 Inhibitor for the Treatment of COPD.

Authors:  Dennis Williams
Journal:  J Pharm Pract       Date:  2020-12-03
  6 in total

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