Literature DB >> 29363025

CNS-Targeted Antiretroviral Strategies: When Are They Needed and What to Choose.

Andrea Calcagno1, Ambra Barco2, Mattia Trunfio2, Stefano Bonora2.   

Abstract

PURPOSE OF REVIEW: Neurocognitive disorders are not uncommon in HIV-positive patients but their pathogenesis is multifactorial and incompletely understood. After excluding contributing comorbidities, several factors may impair neurocognition including severe immune suppression, incomplete antiviral efficacy, drugs' persistent immune activation, vascular abnormalities, and drugs' neurotoxicity. The effectiveness of targeted antiretroviral strategies on these risk factors is unknown. RECENT
FINDINGS: Recent studies support the idea that residual cerebrospinal fluid HIV RNA in the setting of plasma viral suppression is associated with compartmental immune activation but the link to neuronal damage is debated. Some authors have reported an incomplete antiviral efficacy in macrophage-derived cells but targeted antiretroviral regimen switches have not been performed. Additionally, improvements in neurocognition using drugs with better central nervous system penetration or maraviroc (associated with favorable immunological properties) have been observed in pilot studies. Trials evaluating specific interventions for cardiovascular health (including brain white matter abnormalities) and neurotoxicity of antiretrovirals are warranted. Central nervous system-targeted antiretroviral strategies are needed in patients with uncontrolled cerebrospinal HIV replication, and they may be suggested in subjects with low CD4 nadir, individuals carrying drug-resistant viruses, and those with compartmental immune activation.

Entities:  

Keywords:  Antiretrovirals; Cerebrospinal fluid; Compartmentalization; HIV-associated neurocognitive disorders; Pharmacodynamics; Pharmacokinetics

Mesh:

Substances:

Year:  2018        PMID: 29363025     DOI: 10.1007/s11904-018-0375-2

Source DB:  PubMed          Journal:  Curr HIV/AIDS Rep        ISSN: 1548-3568            Impact factor:   5.071


  46 in total

1.  HIV-1 CNS in vitro infectivity models based on clinical CSF samples.

Authors:  Borja Mora-Peris; Alan Winston; Lucy Garvey; Laura J Else; Robin J Shattock; Carolina Herrera
Journal:  J Antimicrob Chemother       Date:  2015-10-15       Impact factor: 5.790

Review 2.  Antiretroviral therapy in macrophages: implication for HIV eradication.

Authors:  Christina Gavegnano; Raymond F Schinazi
Journal:  Antivir Chem Chemother       Date:  2009-10-19

3.  Antiretroviral neurotoxicity.

Authors:  Kevin Robertson; Jeff Liner; Rick B Meeker
Journal:  J Neurovirol       Date:  2012-07-19       Impact factor: 2.643

Review 4.  Mechanisms underlying activity of antiretroviral drugs in HIV-1-infected macrophages: new therapeutic strategies.

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Journal:  J Leukoc Biol       Date:  2006-08-24       Impact factor: 4.962

5.  Randomized trial of central nervous system-targeted antiretrovirals for HIV-associated neurocognitive disorder.

Authors:  Ronald J Ellis; Scott Letendre; Florin Vaida; Richard Haubrich; Robert K Heaton; Ned Sacktor; David B Clifford; Brookie M Best; Susanne May; Anya Umlauf; Mariana Cherner; Chelsea Sanders; Craig Ballard; David M Simpson; Cheryl Jay; J Allen McCutchan
Journal:  Clin Infect Dis       Date:  2013-12-18       Impact factor: 9.079

Review 6.  CCR5 blockade for neuroinflammatory diseases--beyond control of HIV.

Authors:  Guillaume Martin-Blondel; David Brassat; Jan Bauer; Hans Lassmann; Roland S Liblau
Journal:  Nat Rev Neurol       Date:  2016-01-18       Impact factor: 42.937

7.  Maraviroc-intensified combined antiretroviral therapy improves cognition in virally suppressed HIV-associated neurocognitive disorder.

Authors:  Thomas M Gates; Lucette A Cysique; Krista J Siefried; Joga Chaganti; Kirsten J Moffat; Bruce J Brew
Journal:  AIDS       Date:  2016-02-20       Impact factor: 4.177

8.  Discordance between cerebral spinal fluid and plasma HIV replication in patients with neurological symptoms who are receiving suppressive antiretroviral therapy.

Authors:  Ana Canestri; François-Xavier Lescure; Stephane Jaureguiberry; Antoine Moulignier; Corinne Amiel; Anne Geneviève Marcelin; Gilles Peytavin; Roland Tubiana; Gilles Pialoux; Christine Katlama
Journal:  Clin Infect Dis       Date:  2010-03-01       Impact factor: 9.079

9.  Health-adjusted life expectancy in HIV-positive and HIV-negative men and women in British Columbia, Canada: a population-based observational cohort study.

Authors:  Robert S Hogg; Oghenowede Eyawo; Alexandra B Collins; Wendy Zhang; Shahab Jabbari; Mark W Hull; Viviane Dias Lima; Tareq Ahmed; Claire E Kendall; Keri N Althoff; Amy C Justice; Rolando Barrios; Jeannie Shoveller; Julio S G Montaner
Journal:  Lancet HIV       Date:  2017-03-03       Impact factor: 12.767

10.  Multicenter European Prevalence Study of Neurocognitive Impairment and Associated Factors in HIV Positive Patients.

Authors:  Lewis J Haddow; Rosanna Laverick; Marina Daskalopoulou; Jeffrey McDonnell; Fiona C Lampe; Richard Gilson; Andrew Speakman; Andrea Antinori; Pietro Balestra; Tina Bruun; Jan Gerstoft; Lars Nielsen; Anna Vassilenko; Simon Collins; Alison J Rodger
Journal:  AIDS Behav       Date:  2018-05
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  8 in total

Review 1.  Current and Future Therapeutic Strategies for Lentiviral Eradication from Macrophage Reservoirs.

Authors:  Tiffany A Peterson; Andrew G MacLean
Journal:  J Neuroimmune Pharmacol       Date:  2018-10-13       Impact factor: 4.147

Review 2.  Pharmacologic approaches to HIV-associated neurocognitive disorders.

Authors:  Sean N Avedissian; Shetty Ravi Dyavar; Howard S Fox; Courtney V Fletcher
Journal:  Curr Opin Pharmacol       Date:  2020-10-10       Impact factor: 5.547

3.  Screening Accuracy of Mini Addenbrooke's Cognitive Examination Test for HIV-Associated Neurocognitive Disorders in People Ageing with HIV.

Authors:  Mattia Trunfio; Davide De Francesco; Daniela Vai; Caterina Medina; Maurizio Milesi; Simone Domini; Chiara Alcantarini; Daniele Imperiale; Stefano Bonora; Giovanni Di Perri; Andrea Calcagno
Journal:  AIDS Behav       Date:  2022-01-04

Review 4.  Clinical Treatment Options and Randomized Clinical Trials for Neurocognitive Complications of HIV Infection: Combination Antiretroviral Therapy, Central Nervous System Penetration Effectiveness, and Adjuvants.

Authors:  Shih-Ping Lin; Andrea Calcagno; Scott L Letendre; Qing Ma
Journal:  Curr Top Behav Neurosci       Date:  2021

5.  Correlations between cerebrospinal fluid biomarkers, neurocognitive tests, and resting-state electroencephalography (rsEEG) in patients with HIV-associated neurocognitive disorders.

Authors:  A Barco; S Orlando; G Stroffolini; V Pirriatore; A Lazzaro; D Vai; G Guastamacchia; G Noce; C Atzori; M Trunfio; S Bonora; G Di Perri; A Calcagno
Journal:  J Neurovirol       Date:  2022-01-19       Impact factor: 2.643

Review 6.  Co-receptor signaling in the pathogenesis of neuroHIV.

Authors:  E A Nickoloff-Bybel; L Festa; O Meucci; P J Gaskill
Journal:  Retrovirology       Date:  2021-08-24       Impact factor: 4.602

7.  Legacy effect on neuropsychological function in HIV-infected men on combination antiretroviral therapy.

Authors:  Yang Qu; Andrea Weinstein; Zheng Wang; Yu Cheng; Lawrence Kingsley; Andrew Levine; Eileen Martin; Cynthia Munro; Ann B Ragin; Leah H Rubin; Ned W Sacktor; Eric C Seaberg; James T Becker
Journal:  AIDS       Date:  2022-01-01       Impact factor: 4.177

8.  HIV-1-Associated Neurocognitive Disorders: Is HLA-C Binding Stability to β2-Microglobulin a Missing Piece of the Pathogenetic Puzzle?

Authors:  Donato Zipeto; Michela Serena; Simona Mutascio; Francesca Parolini; Erica Diani; Elisabetta Guizzardi; Valentina Muraro; Emanuela Lattuada; Sebastiano Rizzardo; Marina Malena; Massimiliano Lanzafame; Giovanni Malerba; Maria Grazia Romanelli; Stefano Tamburin; Davide Gibellini
Journal:  Front Neurol       Date:  2018-09-21       Impact factor: 4.003

  8 in total

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