Literature DB >> 29303047

Eltrombopag in the management of aplastic anaemia: real-world experience in a non-trial setting.

Yu-Yan Hwang1, Harinder Gill1, Thomas S Y Chan1, Garret M K Leung1, Carol Y M Cheung1, Yok-Lam Kwong1.   

Abstract

OBJECTIVE: The thrombopoietin mimetic eltrombopag has been used in clinical trials for the frontline and salvage treatment of aplastic anaemia (AA). Eltrombopag was investigated in AA patients on a non-trial all-comer basis.
METHODS: Consecutive newly diagnosed and relapsed/refractory AA patients were treated with eltrombopag.
RESULTS: In a 4.5-year period, 20 consecutive AA patients (newly diagnosed, N = 10; relapsed/refractory, N = 10) at a median age of 47 (22-84) years were treated with eltrombopag. For newly diagnosed patients, the frontline use of eltrombopag (concomitant medications: anti-thymocyte globulin, ATG, and ciclosporin, N = 4; ciclosporin, N = 5; nil, N = 1) at a median maximum dose of 150 (50-300) mg/day led to an overall response rate (ORR) of 90% (trilineage: 60%; neutrophil: 20%; platelet: 10%). After a median follow-up of 47 (14-179) weeks, responses were maintained in all cases. In relapsed/refractory patients, eltrombopag at a median maximum dose of 150 (50-300) mg/day led to an ORR of 50% (trilineage: 40%; neutrophil: 10%), with responses maintained after a median follow-up of 115 (53-253) weeks. Adverse effects included reversible skin pigmentation (observed in all patients taking eltrombopag at ≥150 mg/day), dyspepsia, and liver function derangement.
CONCLUSION: In a routine haematological practice, the use of eltrombopag in AA patients was feasible, safe, and associated with very favourable responses.

Entities:  

Keywords:  Aplastic anaemia; anti-thymocyte globulin; ciclosporin; eltrombopag; newly diagnosed; refractory; relapsed

Mesh:

Substances:

Year:  2018        PMID: 29303047     DOI: 10.1080/10245332.2017.1422306

Source DB:  PubMed          Journal:  Hematology        ISSN: 1024-5332            Impact factor:   2.269


  8 in total

Review 1.  Activity of eltrombopag in severe aplastic anemia.

Authors:  Phillip Scheinberg
Journal:  Hematology Am Soc Hematol Educ Program       Date:  2018-11-30

Review 2.  Activity of eltrombopag in severe aplastic anemia.

Authors:  Phillip Scheinberg
Journal:  Blood Adv       Date:  2018-11-13

3.  Relationship between CYP2C8, UGT1A1, and ABCG2 gene polymorphisms and the exposure, efficacy, and toxicity of eltrombopag in the treatment of refractory aplastic anemia.

Authors:  Wei Zuo; Bo Liu; Miao Chen; Bo Zhang; Bing Han
Journal:  Eur J Clin Pharmacol       Date:  2022-08-03       Impact factor: 3.064

4.  Eltrombopag in Combination with Rabbit Anti-thymocyte Globulin/Cyclosporine A in Immunosuppressive Therapy-naïve Patients with Aplastic Anemia in Japan.

Authors:  Kazunori Imada; Naoshi Obara; Hiroatsu Iida; Kenji Imajo; Tetsuo Maeda; Kensuke Usuki; Zhang Fanghong; Yosuke Hombo; Takeshi Tajima; Akiko Kumagai; Akira Matsuda; Shinji Nakao
Journal:  Intern Med       Date:  2020-11-23       Impact factor: 1.271

5.  Correlation of the Plasma Concentration of Eltrombopag With Efficacy in the Treatment of Refractory Aplastic Anemia: A Single-Centre Study in China.

Authors:  Wei Zuo; Bo Zhang; Jing Ruan; Miao Chen; Bing Han
Journal:  Front Pharmacol       Date:  2020-11-16       Impact factor: 5.810

6.  The Effectiveness of Rapamycin Combined with Eltrombopag in Murine Models of Immune-Mediated Bone Marrow Failure.

Authors:  Shaoxue Ding; Xiaowei Liang; Tian Zhang; Rong Fu
Journal:  J Immunol Res       Date:  2020-10-17       Impact factor: 4.818

Review 7.  Novel therapeutic choices in immune aplastic anemia.

Authors:  Phillip Scheinberg
Journal:  F1000Res       Date:  2020-09-10

8.  [How I treat refractory sever aplastic anemia].

Authors:  F K Zhang
Journal:  Zhonghua Xue Ye Xue Za Zhi       Date:  2020-09-14
  8 in total

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