Literature DB >> 29272700

Multi-targeting Drug Community Challenge.

Avner Schlessinger1, Ruben Abagyan2, Heather A Carlson3, Kristen K Dang4, Justin Guinney4, Ross L Cagan5.   

Abstract

Mesh:

Year:  2017        PMID: 29272700     DOI: 10.1016/j.chembiol.2017.12.006

Source DB:  PubMed          Journal:  Cell Chem Biol        ISSN: 2451-9448            Impact factor:   8.116


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  6 in total

1.  Extended Multitarget Pharmacology of Anticancer Drugs.

Authors:  Da Shi; Feroz Khan; Ruben Abagyan
Journal:  J Chem Inf Model       Date:  2019-05-03       Impact factor: 4.956

2.  Key Parameters of Tumor Epitope Immunogenicity Revealed Through a Consortium Approach Improve Neoantigen Prediction.

Authors:  Daniel K Wells; Marit M van Buuren; Kristen K Dang; Vanessa M Hubbard-Lucey; Kathleen C F Sheehan; Katie M Campbell; Andrew Lamb; Jeffrey P Ward; John Sidney; Ana B Blazquez; Andrew J Rech; Jesse M Zaretsky; Begonya Comin-Anduix; Alphonsus H C Ng; William Chour; Thomas V Yu; Hira Rizvi; Jia M Chen; Patrice Manning; Gabriela M Steiner; Xengie C Doan; Taha Merghoub; Justin Guinney; Adam Kolom; Cheryl Selinsky; Antoni Ribas; Matthew D Hellmann; Nir Hacohen; Alessandro Sette; James R Heath; Nina Bhardwaj; Fred Ramsdell; Robert D Schreiber; Ton N Schumacher; Pia Kvistborg; Nadine A Defranoux
Journal:  Cell       Date:  2020-10-09       Impact factor: 41.582

3.  Crowdsourced mapping of unexplored target space of kinase inhibitors.

Authors:  Anna Cichońska; Balaguru Ravikumar; Robert J Allaway; Fangping Wan; Sungjoon Park; Olexandr Isayev; Shuya Li; Michael Mason; Andrew Lamb; Ziaurrehman Tanoli; Minji Jeon; Sunkyu Kim; Mariya Popova; Stephen Capuzzi; Jianyang Zeng; Kristen Dang; Gregory Koytiger; Jaewoo Kang; Carrow I Wells; Timothy M Willson; Tudor I Oprea; Avner Schlessinger; David H Drewry; Gustavo Stolovitzky; Krister Wennerberg; Justin Guinney; Tero Aittokallio
Journal:  Nat Commun       Date:  2021-06-03       Impact factor: 14.919

4.  Integrated computational and Drosophila cancer model platform captures previously unappreciated chemicals perturbing a kinase network.

Authors:  Peter M U Ung; Masahiro Sonoshita; Alex P Scopton; Arvin C Dar; Ross L Cagan; Avner Schlessinger
Journal:  PLoS Comput Biol       Date:  2019-04-26       Impact factor: 4.475

5.  Successive Statistical and Structure-Based Modeling to Identify Chemically Novel Kinase Inhibitors.

Authors:  Lindsey Burggraaff; Eelke B Lenselink; Willem Jespers; Jesper van Engelen; Brandon J Bongers; Marina Gorostiola González; Rongfang Liu; Holger H Hoos; Herman W T van Vlijmen; Adriaan P IJzerman; Gerard J P van Westen
Journal:  J Chem Inf Model       Date:  2020-05-12       Impact factor: 4.956

6.  Crowdsourced identification of multi-target kinase inhibitors for RET- and TAU- based disease: The Multi-Targeting Drug DREAM Challenge.

Authors:  Zhaoping Xiong; Minji Jeon; Robert J Allaway; Jaewoo Kang; Donghyeon Park; Jinhyuk Lee; Hwisang Jeon; Miyoung Ko; Hualiang Jiang; Mingyue Zheng; Aik Choon Tan; Xindi Guo; Kristen K Dang; Alex Tropsha; Chana Hecht; Tirtha K Das; Heather A Carlson; Ruben Abagyan; Justin Guinney; Avner Schlessinger; Ross Cagan
Journal:  PLoS Comput Biol       Date:  2021-09-14       Impact factor: 4.779

  6 in total

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