Literature DB >> 29187493

BRAF, NRAS and C-KIT Advanced Melanoma: Clinico-pathological Features, Targeted-Therapy Strategies and Survival.

Giovanni Ponti1, Marco Manfredini2, Stefano Greco3, Giovanni Pellacani2, Roberta Depenni3, Aldo Tomasi4, Monia Maccaferri2, Stefano Cascinu3.   

Abstract

BACKGROUND/AIM: The mutational status of stage III and IV melanomas should be recognized in order to allow for targeted therapies. The aim of our study was the characterization of BRAF, NRAS and C-KIT melanoma patients, in order to define their optimal management. PATIENTS AND METHODS: Between 1991 and 2015, 63 mutated melanoma patients were treated and monitored during their diagnostic and therapeutic management at a single institution.
RESULTS: BRAF-mutated melanoma patients were the most common, representing 70% of the study population, while NRAS- and C-KIT-mutated melanoma represented 19% and 11% respectively. BRAF-mutated melanomas were mostly located at sites of intermittent sun exposure, and were associated with higher Breslow thickness and an increased number of mitosis. NRAS mutated melanoma were mainly observed in chronic sun-damaged areas and had a negative prognostic value, with shorter time to progression and a high incidence of central nervous system involvement. C-KIT mutated melanoma were located at acral and mucosal sites. Overall survival observed in the three groups of patients revealed wide differences.
CONCLUSION: BRAF, NRAS and C-KIT melanomas constitute distinct clinico-pathological entities. BRAF-mutated melanoma benefit from both anti-BRAF and anti-MEK targeted therapies while triple-negative melanomas could benefit from novel anti-CTLA-4 and anti-PD-L1 immunotherapeutic approaches. Copyright
© 2017, International Institute of Anticancer Research (Dr. George J. Delinasios), All rights reserved.

Entities:  

Keywords:  Advanced melanoma; BRAF, NRAS and C-KIT; survival; targeted therapies

Mesh:

Substances:

Year:  2017        PMID: 29187493     DOI: 10.21873/anticanres.12175

Source DB:  PubMed          Journal:  Anticancer Res        ISSN: 0250-7005            Impact factor:   2.480


  13 in total

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Authors:  Chi Yan; Chengzhi Zhao; Ke Yang; Hongyan Zhou; Limin Jing; Weixing Zhao; Wenguang Dou; Qingxin Xia; Jie Ma; Bing Wei; Yongjun Guo
Journal:  Front Mol Biosci       Date:  2022-06-02

2.  Synthesis, inverse docking-assisted identification and in vitro biological characterization of Flavonol-based analogs of fisetin as c-Kit, CDK2 and mTOR inhibitors against melanoma and non-melanoma skin cancers.

Authors:  Tithi Roy; Samuel T Boateng; Sergette Banang-Mbeumi; Pankaj K Singh; Pratik Basnet; Roxane-Cherille N Chamcheu; Federico Ladu; Isabel Chauvin; Vladimir S Spiegelman; Ronald A Hill; Konstantin G Kousoulas; Bolni Marius Nagalo; Anthony L Walker; Jean Fotie; Siva Murru; Mario Sechi; Jean Christopher Chamcheu
Journal:  Bioorg Chem       Date:  2020-12-30       Impact factor: 5.275

3.  KIT Mutation Incidence and Pattern of Melanoma in Central Europe.

Authors:  V Doma; T Barbai; M-A Beleaua; I Kovalszky; E Rásó; József Tímár
Journal:  Pathol Oncol Res       Date:  2019-12-17       Impact factor: 3.201

4.  Immunohistochemical mismatch repair proteins expression as a tool to predict the melanoma immunotherapy response.

Authors:  Giovanni Ponti; Giovanni Pellacani; Aldo Tomasi; Roberta Depenni; Monia Maccaferri; Antonio Maiorana; Giulia Orsi; Francesca Giusti; Stefano Cascinu; Marco Manfredini
Journal:  Mol Clin Oncol       Date:  2019-11-07

5.  PLA1A expression as a diagnostic marker of BRAF-mutant metastasis in melanoma cancer.

Authors:  Gang Yang; Shuya Liu; Mazaher Maghsoudloo; Marzieh Dehghan Shasaltaneh; Parham Jabbarzadeh Kaboli; Cuiwei Zhang; Youcai Deng; Hajar Heidari; Maliheh Entezari; ShaoZhi Fu; QingLian Wen; Saber Imani
Journal:  Sci Rep       Date:  2021-03-15       Impact factor: 4.379

6.  Difficulties in diagnosing anorectal melanoma: A case report and review of the literature.

Authors:  Raluca Cristina Apostu; Elena Stefanescu; Radu Razvan Scurtu; Gabriel Kacso; Radu Drasovean
Journal:  World J Clin Cases       Date:  2021-12-26       Impact factor: 1.337

7.  Comprehensive analysis identifies IFI16 as a novel signature associated with overall survival and immune infiltration of skin cutaneous melanoma.

Authors:  Hanwen Wang; Xiaoxia Xie; Junyou Zhu; Shaohai Qi; Julin Xie
Journal:  Cancer Cell Int       Date:  2021-12-20       Impact factor: 5.722

8.  BRAF, C-KIT, and NRAS mutations correlated with different clinicopathological features: an analysis of 691 melanoma patients from a single center.

Authors:  Min Ren; Jing Zhang; Yunyi Kong; Qianming Bai; Peng Qi; Ling Zhang; Qian Wang; Xiaoyan Zhou; Yong Chen; Xiaoli Zhu
Journal:  Ann Transl Med       Date:  2022-01

Review 9.  Revolutions in treatment options in gastrointestinal stromal tumours (GISTs): the latest updates

Authors:  Sheima Farag; Myles J Smith; Nicos Fotiadis; Anastasia Constantinidou; Robin L Jones
Journal:  Curr Treat Options Oncol       Date:  2020-05-27

10.  A Rare Case of Primary Anorectal Melanoma and a Review of the Current Landscape of Therapy.

Authors:  Ho-Man Yeung; Brinda Gupta; Bhishak Kamat
Journal:  J Community Hosp Intern Med Perspect       Date:  2020-08-02
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