Literature DB >> 29182361

Ado-trastuzumab emtansine (T-DM1) in HER2+ advanced breast cancer patients: does pretreatment with pertuzumab matter?

Alessandra Fabi1, Diana Giannarelli2, Luca Moscetti3, Daniele Santini4, Alberto Zambelli5, Michelino De Laurentiis6, Michele Caruso7, Daniele Generali8, Enrichetta Valle9, Vita Leonardi10, Katia Cannita11, Grazia Arpino12, Gianfranco Filippelli13, Gianluigi Ferretti1, Marianna Giampaglia14, Filippo Montemurro15, Cecilia Nisticò1, Simona Gasparro1, Francesco Cognetti1.   

Abstract

AIM: We evaluated the outcomes of patients treated with ado-trastuzumab emantasine (T-DM1) after first-line pertuzumab/trastuzumab, compared with those receiving a trastuzumab-only-based regimen. PATIENTS &
METHODS: Patients who received second-line T-DM1 after pertuzumab/trastuzumab (n = 34) were compared with those who received only trastuzumab (n = 73).
RESULTS: Overall response rate was 33.3% in patients with prior pertuzumab and 57.1% in the remaining subjects. Disease control rate was 47 and 43%, respectively, and the clinical benefit rate was 43.3 and 71.1%, respectively. Median progression-free survival was 5.0 and 11.0 months, respectively (hazard ratio: 2.02; 95% CI: 1.14-3.58; p = 0.01).
CONCLUSION: Patients treated with T-DM1 who previously received pertuzumab present poorer clinical outcomes compared with those receiving a trastuzumab-only-based regimen in the first-line setting.

Entities:  

Keywords:  HER2 second-line; HER2-positive tumors; T-DM1; metastatic breast cancer; pertuzumab

Mesh:

Substances:

Year:  2017        PMID: 29182361     DOI: 10.2217/fon-2017-0336

Source DB:  PubMed          Journal:  Future Oncol        ISSN: 1479-6694            Impact factor:   3.404


  9 in total

Review 1.  Antibody-Drug Conjugates in Breast Cancer: a Comprehensive Review.

Authors:  Noam Pondé; Philippe Aftimos; Martine Piccart
Journal:  Curr Treat Options Oncol       Date:  2019-04-01

2.  Tucatinib Combined With Ado-Trastuzumab Emtansine in Advanced ERBB2/HER2-Positive Metastatic Breast Cancer: A Phase 1b Clinical Trial.

Authors:  Virginia F Borges; Cristiano Ferrario; Nathalie Aucoin; Carla Falkson; Qamar Khan; Ian Krop; Stephen Welch; Alison Conlin; Jorge Chaves; Philippe L Bedard; Marc Chamberlain; Todd Gray; Alex Vo; Erika Hamilton
Journal:  JAMA Oncol       Date:  2018-09-01       Impact factor: 31.777

Review 3.  The trastuzumab era: current and upcoming targeted HER2+ breast cancer therapies.

Authors:  Jordyn Kreutzfeldt; Brett Rozeboom; Nandini Dey; Pradip De
Journal:  Am J Cancer Res       Date:  2020-04-01       Impact factor: 6.166

4.  T-DM1 after Pertuzumab plus Trastuzumab: Treatment Sequence-Induced Selection Bias in HER2-Positive Metastatic Breast Cancer.

Authors:  Thibaut Sanglier; Alessandra Fabi; Carlos Flores; Evelyn M Flahavan; Claudia Pena-Murillo; Anne-Marie Meyer; Filippo Montemurro
Journal:  Cancers (Basel)       Date:  2022-05-17       Impact factor: 6.575

5.  T-DM1 efficacy in trastuzumab-pertuzumab pre-treated HER2 positive metastatic breast cancer patients: a meta-analysis.

Authors:  Claudia Omarini; Federico Piacentini; Isabella Sperduti; Krisida Cerma; Monica Barbolini; Fabio Canino; Cecilia Nasso; Christel Isca; Federica Caggia; Massimo Dominici; Luca Moscetti
Journal:  BMC Cancer       Date:  2022-06-07       Impact factor: 4.638

6.  A tipping-point for apoptosis following dual inhibition of HER2 signaling network by T-DM1 plus GDC-0980 maximizes anti-tumor efficacy.

Authors:  Nandini Dey; Jennifer Aske; Xiaoqian Lin; Yuliang Sun; Brian Leyland-Jones; Lori Friedman; Pradip De
Journal:  Am J Cancer Res       Date:  2021-06-15       Impact factor: 6.166

7.  Pertuzumab and Trastuzumab Emtansine for Human Epidermal Growth Factor Receptor-2-Positive Metastatic Breast Cancer: Contemporary Population-Based Outcomes.

Authors:  Sasha Lupichuk; Winson Y Cheung; Douglas Stewart
Journal:  Breast Cancer (Auckl)       Date:  2019-10-09

8.  Liquid biopsy identifies actionable dynamic predictors of resistance to Trastuzumab Emtansine (T-DM1) in advanced HER2-positive breast cancer.

Authors:  Matteo Allegretti; Alessandra Fabi; Elena Giordani; Cristiana Ercolani; Paolo Romania; Cecilia Nisticò; Simona Gasparro; Vittoria Barberi; Maria Ciolina; Edoardo Pescarmona; Diana Giannarelli; Gennaro Ciliberto; Francesco Cognetti; Patrizio Giacomini
Journal:  Mol Cancer       Date:  2021-11-29       Impact factor: 27.401

9.  Second line trastuzumab emtansine following horizontal dual blockade in a real-life setting.

Authors:  Salvatore Del Prete; Liliana Montella; Grazia Arpino; Giuseppe Buono; Carlo Buonerba; Pasquale Dolce; Olga Fiorentino; Maria Aliberti; Antonio Febbraro; Clementina Savastano; Giuseppe Colantuoni; Ferdinando Riccardi; Angela Ruggiero; Sabino De Placido; Michele Orditura
Journal:  Oncotarget       Date:  2020-06-02
  9 in total

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