Literature DB >> 28858337

Prostate cancer: Place your BETs.

Louise Stone.   

Abstract

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Year:  2017        PMID: 28858337     DOI: 10.1038/nrurol.2017.147

Source DB:  PubMed          Journal:  Nat Rev Urol        ISSN: 1759-4812            Impact factor:   14.432


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  3 in total

1.  Opposing effects of cancer-type-specific SPOP mutants on BET protein degradation and sensitivity to BET inhibitors.

Authors:  Hana Janouskova; Geniver El Tekle; Elisa Bellini; Namrata D Udeshi; Anna Rinaldi; Anna Ulbricht; Tiziano Bernasocchi; Gianluca Civenni; Marco Losa; Tanya Svinkina; Craig M Bielski; Gregory V Kryukov; Luciano Cascione; Sara Napoli; Radoslav I Enchev; David G Mutch; Michael E Carney; Andrew Berchuck; Boris J N Winterhoff; Russell R Broaddus; Peter Schraml; Holger Moch; Francesco Bertoni; Carlo V Catapano; Matthias Peter; Steven A Carr; Levi A Garraway; Peter J Wild; Jean-Philippe P Theurillat
Journal:  Nat Med       Date:  2017-08-14       Impact factor: 53.440

2.  Intrinsic BET inhibitor resistance in SPOP-mutated prostate cancer is mediated by BET protein stabilization and AKT-mTORC1 activation.

Authors:  Pingzhao Zhang; Dejie Wang; Yu Zhao; Shancheng Ren; Kun Gao; Zhenqing Ye; Shangqian Wang; Chun-Wu Pan; Yasheng Zhu; Yuqian Yan; Yinhui Yang; Di Wu; Yundong He; Jun Zhang; Daru Lu; Xiuping Liu; Long Yu; Shimin Zhao; Yao Li; Dong Lin; Yuzhuo Wang; Liguo Wang; Yu Chen; Yinghao Sun; Chenji Wang; Haojie Huang
Journal:  Nat Med       Date:  2017-08-14       Impact factor: 53.440

3.  Prostate cancer-associated SPOP mutations confer resistance to BET inhibitors through stabilization of BRD4.

Authors:  Xiangpeng Dai; Wenjian Gan; Xiaoning Li; Shangqian Wang; Wei Zhang; Ling Huang; Shengwu Liu; Qing Zhong; Jianping Guo; Jinfang Zhang; Ting Chen; Kouhei Shimizu; Francisco Beca; Mirjam Blattner; Divya Vasudevan; Dennis L Buckley; Jun Qi; Lorenz Buser; Pengda Liu; Hiroyuki Inuzuka; Andrew H Beck; Liewei Wang; Peter J Wild; Levi A Garraway; Mark A Rubin; Christopher E Barbieri; Kwok-Kin Wong; Senthil K Muthuswamy; Jiaoti Huang; Yu Chen; James E Bradner; Wenyi Wei
Journal:  Nat Med       Date:  2017-08-14       Impact factor: 53.440

  3 in total

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