Literature DB >> 28811242

Natural NS5A inhibitor resistance associated substitutions in hepatitis C virus genotype 1 infected patients from Italy.

C Caudai1, A Materazzi2, F Saladini2, S Di Giambenedetto3, C Torti4, B Ricciardi5, B Rossetti6, P Almi7, A De Luca8, M Zazzi2.   

Abstract

OBJECTIVES: Genetic variability in NS5A is associated with different levels of resistance to the currently licensed NS5A inhibitors. The aim of this study was to detect NS5A inhibitor resistance associated substitutions (RASs) in hepatitis C virus (HCV) genotype 1 (GT1) patients who are naive to direct-acting HCV antivirals.
METHODS: Amplification, Sanger sequencing and phylogenetic analysis of the HCV NS5A region were performed on plasma obtained from 122 consecutive patients with HCV chronic infection attending four different clinics in Italy.
RESULTS: NS5A inhibitor RASs were detected in 14/61 (23.0%) HCV GT1b and 3/61 (4.9%) HCV GT1a infected patients (p 0.007). The pan-genotypic RAS Y93H was detected in 1 (1.6%) GT1a and 4 (6.6%) GT1b patients. GT1a sequences clustered into two different clades with RASs detected in 1/34 (2.9%) clade I and 2/27 (7.4%) clade II sequences.
CONCLUSIONS: Although the impact of naturally occurring NS5A RASs might be limited with upcoming pan-genotypic treatment regimens, this information is still useful to map naturally occurring HCV variants in different geographic areas in the context of current HCV therapy.
Copyright © 2017 European Society of Clinical Microbiology and Infectious Diseases. Published by Elsevier Ltd. All rights reserved.

Entities:  

Keywords:  Direct-acting antivirals; Drug resistance; Hepatitis C virus; NS5A; Pegylated interferon-α and ribavirin

Mesh:

Substances:

Year:  2017        PMID: 28811242     DOI: 10.1016/j.cmi.2017.08.003

Source DB:  PubMed          Journal:  Clin Microbiol Infect        ISSN: 1198-743X            Impact factor:   8.067


  5 in total

Review 1.  Resistance detection and re-treatment options in hepatitis C virus-related chronic liver diseases after DAA-treatment failure.

Authors:  Evangelista Sagnelli; Mario Starace; Carmine Minichini; Mariantonietta Pisaturo; Margherita Macera; Caterina Sagnelli; Nicola Coppola
Journal:  Infection       Date:  2018-08-06       Impact factor: 3.553

2.  Molecular Epidemiology and Baseline Resistance of Hepatitis C Virus to Direct Acting Antivirals in Croatia.

Authors:  Petra Simicic; Anamarija Slovic; Leona Radmanic; Adriana Vince; Snjezana Zidovec Lepej
Journal:  Pathogens       Date:  2022-07-19

3.  Prevalence of Single and Multiple Natural NS3, NS5A and NS5B Resistance-Associated Substitutions in Hepatitis C Virus Genotypes 1-4 in Italy.

Authors:  Ada Bertoli; Maria Chiara Sorbo; Marianna Aragri; Ilaria Lenci; Elisabetta Teti; Ennio Polilli; Velia Chiara Di Maio; Laura Gianserra; Elisa Biliotti; Chiara Masetti; Carlo F Magni; Sergio Babudieri; Laura A Nicolini; Martina Milana; Pierluigi Cacciatore; Loredana Sarmati; Adriano Pellicelli; Stefania Paolucci; Antonio Craxì; Filomena Morisco; Valeria Pace Palitti; Massimo Siciliano; Nicola Coppola; Nerio Iapadre; Massimo Puoti; Giuliano Rizzardini; Gloria Taliani; Caterina Pasquazzi; Massimo Andreoni; Giustino Parruti; Mario Angelico; Carlo Federico Perno; Valeria Cento; Francesca Ceccherini-Silberstein
Journal:  Sci Rep       Date:  2018-06-12       Impact factor: 4.379

Review 4.  Hepatitis C Viral Replication Complex.

Authors:  Hui-Chun Li; Chee-Hing Yang; Shih-Yen Lo
Journal:  Viruses       Date:  2021-03-22       Impact factor: 5.048

5.  Effectiveness of direct-acting antivirals for hepatitis C virus infection in hepatitis C/HIV coinfected individuals: A multicenter study.

Authors:  Soraia M Machado; Aline G Vigani; Andrea G Leite; Ana Claudia M Diaz; Paulo Roberto A Ferreira; Dimas Carnaúba-Júnior; Simone B Tenore; Carlos Eduardo Brandão-Mello; Mario P Gonzalez; Fabiana Siroma; Kleber D Prado; Delzi V Nunes; Gaspar Lisboa-Neto; João Renato R Pinho; Fernanda M Malta; Raymundo S Azevedo; Steven S Witkin; Maria Cássia Mendes-Correa
Journal:  Medicine (Baltimore)       Date:  2020-07-24       Impact factor: 1.817

  5 in total

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