Literature DB >> 28782191

Tadalafil, a phosphodiesterase type 5 inhibitor, improves bladder blood supply and restores the initial phase of lower urinary tract dysfunction in diabetic rats.

Daisuke Gotoh1, Kazumasa Torimoto1, Yoshihiro Tatsumi1, Shunta Hori1, Atsushi Yamada1, Makito Miyake1, Yosuke Morizawa1, Katsuya Aoki1, Nobumichi Tanaka1, Akihide Hirayama2, Kiyohide Fujimoto1.   

Abstract

AIMS: To investigate the effect of tadalafil on bladder blood flow and lower urinary tract function in a rat model of diabetes.
MATERIALS AND METHODS: We studied female Sprague-Dawley rats and induced diabetes in some using a single intraperitoneal injection of streptozotocin. We divided the rats into nondiabetes (ND), diabetes (D), and diabetes with tadalafil (DT) groups. The rats were raised for an additional 7 weeks after diabetes induction. The DT group received oral tadalafil (2 mg/kg/day) for 7 days before the experiments. At 7 weeks after diabetes induction, we performed cystometry, resected the bladders for immunohistochemistry (hypoxia-inducible factor-1α [HIF-1α] and 8-oxo-2'-deoxyguanosine [8-OHdG] staining), and measured bladder blood supply using a laser blood flow meter.
RESULTS: The opening pressure, when the urethra opens and urine flow starts, was significantly lower in the DT group than in the D group (24.9 ± 5.9 vs 43.6 ± 12.3 cmH2 O). The inter-contraction interval was significantly longer in the D group than in the ND and DT groups (1566.2 ± 168.7 vs 702.9 ± 165.2 and 787.4 ± 148.8 s). Immunohistochemistry showed positive staining of the urothelial layer for both HIF-1α and 8-OHdG in the D group, but not in the ND or DT groups. Bladder blood flow was significantly lower in the D group than in the ND or DT groups.
CONCLUSIONS: Tadalafil improves bladder blood supply and lower urinary tract function in diabetic rats. Tadalafil may be a promising drug that restores lower urinary tract dysfunction in the early phase of diabetes.
© 2017 Wiley Periodicals, Inc.

Entities:  

Keywords:  ischemia; bladder; phosphodiesterase 5; rat

Mesh:

Substances:

Year:  2017        PMID: 28782191     DOI: 10.1002/nau.23372

Source DB:  PubMed          Journal:  Neurourol Urodyn        ISSN: 0733-2467            Impact factor:   2.696


  8 in total

1.  NLRP3 Promotes Diabetic Bladder Dysfunction and Changes in Symptom-Specific Bladder Innervation.

Authors:  Francis M Hughes; Nathan A Hirshman; Brian M Inouye; Huixia Jin; Eloise W Stanton; Chloe E Yun; Leah G Davis; Jonathan C Routh; J Todd Purves
Journal:  Diabetes       Date:  2018-11-13       Impact factor: 9.461

2.  Oxidative stress marker 8-hydroxyguanosine is more highly expressed in prostate cancer than in benign prostatic hyperplasia.

Authors:  Shinji Ohtake; Takashi Kawahara; Yukari Ishiguro; Teppei Takeshima; Shinnosuke Kuroda; Koji Izumi; Hiroshi Miyamoto; Hiroji Uemura
Journal:  Mol Clin Oncol       Date:  2018-07-03

3.  Therapeutic effects of a soluble guanylate cyclase activator, BAY 60-2770, on lower urinary tract dysfunction in mice with spinal cord injury.

Authors:  Daisuke Gotoh; Tetsuichi Saito; Sergei Karnup; Yosuke Morizawa; Shunta Hori; Yasushi Nakai; Makito Miyake; Kazumasa Torimoto; Kiyohide Fujimoto; Naoki Yoshimura
Journal:  Am J Physiol Renal Physiol       Date:  2022-08-11

Review 4.  Established and emerging treatments for diabetes-associated lower urinary tract dysfunction.

Authors:  Betül R Erdogan; Guiming Liu; Ebru Arioglu-Inan; Martin C Michel
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  2022-05-12       Impact factor: 3.195

5.  Efficacy of Tadalafil Therapy and Changes in Oxidative Stress Levels in Male Patients with Lower Urinary Tract Symptoms and Overactive Bladder.

Authors:  Tomohiro Matsuo; Yasuyoshi Miyata; Kyohei Araki; Yuta Mukae; Asato Otsubo; Kojiro Ohba; Hideki Sakai
Journal:  Low Urin Tract Symptoms       Date:  2019-08-13       Impact factor: 1.592

6.  Metformin and Sildenafil Attenuate Inflammation and Suppress Apoptosis After Ischemia/Reperfusion Injuries in Rat Urinary Bladder.

Authors:  Jong Mok Park; Ju Hyun Shin; Seung Woo Yang; Ji Yong Lee; Chung Lyul Lee; Jae Sung Lim; Ki Hak Song; Gun Hwa Kim; Yong Gil Na
Journal:  Int Neurourol J       Date:  2021-09-03       Impact factor: 2.835

7.  The preventive effect of a free radical scavenger on oxidative stress after the relief of partial bladder outlet obstruction in a rat model.

Authors:  Min Soo Choo; SongZhe Piao; Seung-June Oh
Journal:  PLoS One       Date:  2018-10-22       Impact factor: 3.240

8.  Pathophysiological changes of the lower urinary tract behind voiding dysfunction in streptozotocin-induced long-term diabetic rats.

Authors:  Kazuki Masuda; Naoki Aizawa; Daiji Watanabe; Takatsugu Okegawa; Haruki Kume; Yasuhiko Igawa; Hiroshi Fukuhara
Journal:  Sci Rep       Date:  2020-03-06       Impact factor: 4.379

  8 in total

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