Literature DB >> 28710329

Open-label trial of ranolazine for the treatment of myotonia congenita.

W David Arnold1, David Kline2, Alan Sanderson2, Ahmed A Hawash2, Amy Bartlett2, Kevin R Novak2, Mark M Rich2, John T Kissel2.   

Abstract

OBJECTIVE: To determine open-label, pilot study whether ranolazine could improve signs and symptoms of myotonia and muscle stiffness in patients with myotonia congenita (MC).
METHODS: Thirteen participants were assessed at baseline and 2, 4, and 5 weeks. Ranolazine was started after baseline assessment (500 mg twice daily), increased as tolerated after week 2 (1,000 mg twice daily), and maintained until week 4. Outcomes included change from baseline to week 4 in self-reported severity of symptoms (stiffness, weakness, and pain), Timed Up and Go (TUG), hand grip and eyelid myotonia, and myotonia on EMG.
RESULTS: Self-reported severity of stiffness (p < 0.0001) and weakness (p < 0.01) was significantly improved compared with baseline. TUG and grip myotonia times were reduced (p = 0.03, p = 0.01). EMG of the abductor digiti minimi and tibialis anterior showed significantly reduced myotonia duration (p < 0.001, p < 0.01) at week 4. No participant discontinued ranolazine because of side effects.
CONCLUSIONS: Ranolazine appeared to be well tolerated over a period of 4 weeks in individuals with MC, and ranolazine resulted in improvement of signs and symptoms of muscle stiffness. The findings of this study suggest that ranolazine should be investigated in a larger controlled study. CLASSIFICATION OF EVIDENCE: This study provides Class IV evidence that ranolazine improves myotonia in myotonia congenita.
© 2017 American Academy of Neurology.

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Year:  2017        PMID: 28710329      PMCID: PMC5562961          DOI: 10.1212/WNL.0000000000004229

Source DB:  PubMed          Journal:  Neurology        ISSN: 0028-3878            Impact factor:   9.910


  10 in total

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2.  Ranolazine block of human Na v 1.4 sodium channels and paramyotonia congenita mutants.

Authors:  Nesrine El-Bizri; Kristopher M Kahlig; John C Shyrock; Alfred L George; Luiz Belardinelli; Sridharan Rajamani
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3.  Sodium channel slow inactivation as a therapeutic target for myotonia congenita.

Authors:  Kevin R Novak; Jennifer Norman; Jacob R Mitchell; Martin J Pinter; Mark M Rich
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4.  Nondystrophic myotonia: challenges and future directions.

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5.  Treatment of myotonia with antiarrhythmic drugs.

Authors:  H Kwieciński; B Ryniewicz; A Ostrzycki
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6.  Comparative actions of mexiletine on sodium channels in nerve, skeletal and cardiac muscle.

Authors:  K R Courtney
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7.  The timed "Up & Go": a test of basic functional mobility for frail elderly persons.

Authors:  D Podsiadlo; S Richardson
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8.  Preclinical evaluation of marketed sodium channel blockers in a rat model of myotonia discloses promising antimyotonic drugs.

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9.  Mexiletine for symptoms and signs of myotonia in nondystrophic myotonia: a randomized controlled trial.

Authors:  Jeffrey M Statland; Brian N Bundy; Yunxia Wang; Dipa Raja Rayan; Jaya R Trivedi; Valeria A Sansone; Mohammad K Salajegheh; Shannon L Venance; Emma Ciafaloni; Emma Matthews; Giovanni Meola; Laura Herbelin; Robert C Griggs; Richard J Barohn; Michael G Hanna
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  10 in total
  9 in total

1.  Open-label trial of ranolazine for the treatment of paramyotonia congenita.

Authors:  Samantha Lorusso; David Kline; Amy Bartlett; Miriam Freimer; Julie Agriesti; Ahmed A Hawash; Mark M Rich; John T Kissel; W David Arnold
Journal:  Muscle Nerve       Date:  2018-12-21       Impact factor: 3.217

Review 2.  Genetic neuromuscular disorders: living the era of a therapeutic revolution. Part 2: diseases of motor neuron and skeletal muscle.

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Journal:  Muscle Nerve       Date:  2020-05-27       Impact factor: 3.217

Review 4.  Treatment Updates for Neuromuscular Channelopathies.

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Review 5.  Skeletal Muscle Channelopathies.

Authors:  Lauren Phillips; Jaya R Trivedi
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Review 6.  Myotonic Dystrophies: Targeting Therapies for Multisystem Disease.

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7.  Targeted Therapies for Skeletal Muscle Ion Channelopathies: Systematic Review and Steps Towards Precision Medicine.

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8.  Chaperone activity of niflumic acid on ClC-1 chloride channel mutants causing myotonia congenita.

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Review 9.  Ranolazine: An Old Drug with Emerging Potential; Lessons from Pre-Clinical and Clinical Investigations for Possible Repositioning.

Authors:  Sarah Rouhana; Anne Virsolvy; Nassim Fares; Sylvain Richard; Jérôme Thireau
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  9 in total

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