Literature DB >> 28684048

Dihydrocapsaicin (DHC) enhances the hypothermia-induced neuroprotection following ischemic stroke via PI3K/Akt regulation in rat.

Di Wu1, Jingfei Shi2, Omar Elmadhoun3, Yunxia Duan4, Hong An4, Jun Zhang4, Xiaoduo He4, Ran Meng4, Xiangrong Liu4, Xunming Ji5, Yuchuan Ding6.   

Abstract

OBJECTIVE: Hypothermia has demonstrated neuroprotection following ischemia in preclinical studies while its clinical application is still very limited. The aim of this study was to explore whether combining local hypothermia in ischemic territory achieved by intra-arterial cold infusions (IACIs) with pharmacologically induced hypothermia enhances therapeutic outcomes, as well as the underlying mechanism.
METHODS: Sprague-Dawley rats were subjected to right middle cerebral artery occlusion (MCAO) for 2h using intraluminal hollow filament. The ischemic rats were randomized to receive: 1) pharmacological hypothermia by intraperitoneal (i.p.) injection of dihydrocapsaicin (DHC); 2) physical hypothermia by IACIs for 10min; or 3) the combined treatments. Extent of brain injury was determined by neurological deficit, infarct volume, and apoptotic cell death at 24h and/or 7d following reperfusion. ATP and ROS levels were measured. Expression of p-Akt, cleaved Caspase-3, pro-apoptotic (AIF, Bax) and anti-apoptotic proteins (Bcl-2, Bcl-xL) was evaluated at 24h. Finally, PI3K inhibitor was used to determine the effect of p-Akt.
RESULTS: DHC or IACIs each exhibited hypothermic effect and neuroprotection in rat MCAO models. The combination of pharmacological and physical approaches led to a faster and sustained reduction in brain temperatures and improved ischemia-induced injury than either alone (P<0.01). Furthermore, the combination treatment favorably increased the expression of anti-apoptotic proteins and decreased pro-apoptotic protein levels (P<0.01 or 0.05). This neuroprotective effect was largely blocked by p-Akt inhibition, indicating a potential role of Akt pathway in this mechanism (P<0.01 or 0.05).
CONCLUSIONS: The combination approach is able to enhance the efficiency of hypothermia and efficacy of hypothermia-induced neuroprotection following ischemic stroke. The findings here move us a step closer towards translating this long recognized TH from bench to bedside.
Copyright © 2017 Elsevier B.V. All rights reserved.

Entities:  

Keywords:  Apoptotic cell death; Intra-arterial cold infusions (IACIs); Ischemia/reperfusion injury; Middle cerebral artery; Pharmacological hypothermia

Mesh:

Substances:

Year:  2017        PMID: 28684048     DOI: 10.1016/j.brainres.2017.06.029

Source DB:  PubMed          Journal:  Brain Res        ISSN: 0006-8993            Impact factor:   3.252


  12 in total

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2.  A Direct Comparison of Physical Versus Dihydrocapsaicin-Induced Hypothermia in a Rat Model of Traumatic Spinal Cord Injury.

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4.  MiR-199a-5p inhibition protects cognitive function of ischemic stroke rats by AKT signaling pathway.

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Review 5.  Neuroprotective Phytochemicals in Experimental Ischemic Stroke: Mechanisms and Potential Clinical Applications.

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6.  Less hippocampal neuronal death in young gerbils following transient global cerebral ischemia is associated with long‑term maintenance of insulin‑like growth factor 1 and its receptors in the hippocampal CA1 region.

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Journal:  Mol Med Rep       Date:  2017-12-11       Impact factor: 2.952

7.  Cardioprotective effect of IGF-1 against myocardial ischemia/reperfusion injury through activation of PI3K/Akt pathway in rats in vivo.

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Review 8.  Intra-arterial Cold Saline Infusion in Stroke: Historical Evolution and Future Prospects.

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Review 9.  Therapeutic hypothermia and targeted temperature management for traumatic brain injury: Experimental and clinical experience.

Authors:  W Dalton Dietrich; Helen M Bramlett
Journal:  Brain Circ       Date:  2017-12-29

Review 10.  Nutraceuticals in the Prevention of Neonatal Hypoxia-Ischemia: A Comprehensive Review of their Neuroprotective Properties, Mechanisms of Action and Future Directions.

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