Literature DB >> 28646

Structural requirements of imidazole compounds to be inhibitors or activators of histamine methyltransferase: investigation of histamine analogues and H2-receptor antagonists.

H Barth, W Lorenz.   

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Year:  1978        PMID： 28646     DOI： 10.1007/BF01968615

Source DB:  PubMed          Journal:  Agents Actions        ISSN： 0065-4299


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  15 in total

1.  Cyanoguanidine-thiourea equivalence in the development of the histamine H2-receptor antagonist, cimetidine.

Authors:  G J Durant; J C Emmett; C R Ganellin; P D Miles; M E Parsons; H D Prain; G R White
Journal:  J Med Chem       Date:  1977-07       Impact factor: 7.446

2.  Definition and antagonism of histamine H 2 -receptors.

Authors:  J W Black; W A Duncan; C J Durant; C R Ganellin; E M Parsons
Journal:  Nature       Date:  1972-04-21       Impact factor: 49.962

3.  Speculations about the binding sites of S-adenosyl-L-homocysteine and some of its synthetic analogues to histamine methyltransferase.

Authors:  H Barth; I Niemeyer; W Lorenz
Journal:  Agents Actions       Date:  1974-08

4.  Evidence for a less high acceptor substrate specificity of gastric histamine methyltransferase: methylation of imidazole compounds.

Authors:  H Barth; M Crombach; W Schunack; W Lorenz
Journal:  Biochem Pharmacol       Date:  1980-05-15       Impact factor: 5.858

5.  Sulphur-methylene isosterism in the development of metiamide, a new histamine H2-receptor antagonist.

Authors:  J W Black; G J Durant; J C Emmett; C R Ganellin
Journal:  Nature       Date:  1974-03-01       Impact factor: 49.962

6.  Studies on the mode of action of histamine H1- and H2-receptor antagonists on gastric histamine methyltransferase.

Authors:  H Barth; I Niemeyer; W Lorenz
Journal:  Agents Actions       Date:  1973-10

7.  Similar actions of methylated histamines and histamine receptor antagonists on gastric histamine methyltransferase.

Authors:  H Barth; I Niemeyer; W Lorenz
Journal:  Agents Actions       Date:  1973-10

8.  A sensitive and specific method for the determination of histomine in human whole blood and plasma.

Authors:  W Lorenz; H J Reimann; H Barth; J Kusche; R Meyer; A Doenicke; M Hutzel
Journal:  Hoppe Seylers Z Physiol Chem       Date:  1972-06

9.  Dimaprit, (S-[3-(N,N-dimethylamino)propyl]isothiourea). A highly specific histamine H2-receptor agonist. Part 2. Structure-activity considerations.

Authors:  G J Durant; C R Ganellin; M E Parsons
Journal:  Agents Actions       Date:  1977-03

10.  Sex differences and hormonal control of histamine methyltransferase activity.

Authors:  S H Snyder; J Axelrod
Journal:  Biochim Biophys Acta       Date:  1965-12-16
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  9 in total

1.  Inhibition of histamine methylation in vivo by the dimaprit analog, SKF Compound 91488.

Authors:  M A Beaven; R E Shaff
Journal:  Agents Actions       Date:  1979-12

2.  Histamine uptake and metabolism in intact isolated parietal cells.

Authors:  M Albinus; K F Sewing
Journal:  Agents Actions       Date:  1981-05

3.  Inhibition of histamine-N-methyltransferase activity by neuromuscular blocking drugs.

Authors:  D G Harle; B A Baldo; M M Fisher
Journal:  Agents Actions       Date:  1985-10

4.  Histamine N-methyltransferase: inhibition by monoamine oxidase inhibitors.

Authors:  B Boudíková-Girard; M C Scott; R Weinshilboum
Journal:  Agents Actions       Date:  1993-09

5.  Gastric histamine methyltransferase: different methylation rates for enantiomers of side-chain methylated histamine analogues using a highly purified enzyme preparation.

Authors:  H Barth; W Schunack; M Crombach; W Lorenz
Journal:  Agents Actions       Date:  1984-04

6.  Histamine N-methyl transferase: inhibition by drugs.

Authors:  G M Pacifici; P Donatelli; L Giuliani
Journal:  Br J Clin Pharmacol       Date:  1992-10       Impact factor: 4.335

7.  H1 + H2-receptor antagonists for premedication in anaesthesia and surgery: a critical view based on randomized clinical trials with Haemaccel and various antiallergic drugs.

Authors:  W Lorenz; A Doenicke; B Schöning; J Mamorski; D Weber; E Hinterlang; B Schwarz; E Neugebauer
Journal:  Agents Actions       Date:  1980-04

8.  Inhibition of plant and mammalian diamine oxidase by substrate analogues.

Authors:  T Biegański; Z Osińska; C Masliński
Journal:  Agents Actions       Date:  1982-04

9.  Dual role of imidazole as activator/inhibitor of sweet almond (Prunus dulcis) β-glucosidase.

Authors:  Sara Caramia; Angela Gala Morena Gatius; Fabrizio Dal Piaz; Denis Gaja; Alejandro Hochkoeppler
Journal:  Biochem Biophys Rep       Date:  2017-03-24
  9 in total

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