Literature DB >> 28643356

Bimagrumab improves body composition and insulin sensitivity in insulin-resistant individuals.

Tania Garito1,2, Ronenn Roubenoff2, Marcus Hompesch3, Linda Morrow3, Katherine Gomez3, Daniel Rooks4, Charles Meyers4, Monte S Buchsbaum5, Srikanth Neelakantham6, Therese Swan4, Lee Anne Filosa4, Didier Laurent2, Olivier Petricoul2, Marjorie Zakaria4.   

Abstract

AIM: To test the hypothesis that an improving body composition in insulin-resistant individuals could enhance insulin sensitivity.
METHODS: A total of 16 people with a mean body mass index of 29.3 kg/m2 and insulin resistance, received a single dose of bimagrumab or placebo and were assessed at week 10 for insulin sensitivity, using a hyperinsulinaemic-euglycaemic clamp and an intravenous glucose tolerance test (IVGTT), and for body composition using dual energy X-ray absorptiometry and positron-emission tomography.
RESULTS: Bimagrumab increased lean mass by 2.7% (P < .05) and reduced fat mass by 7.9% (P = .011) at week 10 compared with placebo, and had a neutral effect on body weight. Bimagrumab reduced glycated haemoglobin by 0.21% at week 18 (P < .001) and improved insulin sensitivity by ~20% (according to the clamp) to ~40% (according to the IVGTT).
CONCLUSION: Taking the observed changes together, and given that these occurred without accompanying dietary intervention and without any prescribed regular physical exercise, bimagrumab may offer a novel approach for the treatment of the metabolic complications of obesity.
© 2017 John Wiley & Sons Ltd.

Entities:  

Keywords:  HbA1c; activin receptor II; bimagrumab; body composition; insulin resistance; obesity

Mesh:

Substances:

Year:  2017        PMID: 28643356     DOI: 10.1111/dom.13042

Source DB:  PubMed          Journal:  Diabetes Obes Metab        ISSN: 1462-8902            Impact factor:   6.577


  14 in total

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Journal:  Proc Natl Acad Sci U S A       Date:  2017-11-06       Impact factor: 11.205

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5.  Mechanisms involved in follistatin-induced hypertrophy and increased insulin action in skeletal muscle.

Authors:  Xiuqing Han; Lisbeth Liliendal Valbjørn Møller; Estelle De Groote; Kirstine Nyvold Bojsen-Møller; Jonathan Davey; Carlos Henríquez-Olguin; Zhencheng Li; Jonas Roland Knudsen; Thomas Elbenhardt Jensen; Sten Madsbad; Paul Gregorevic; Erik Arne Richter; Lykke Sylow
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7.  Commentary: Blockade of activin type II receptors with a dual anti-ActRIIA/IIB antibody is critical to promote maximal skeletal muscle hypertrophy.

Authors:  Javier Durán; Manuel Estrada
Journal:  Front Pharmacol       Date:  2018-04-19       Impact factor: 5.810

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Authors:  Mohamed A Alfaleh; Hashem O Alsaab; Ahmad Bakur Mahmoud; Almohanad A Alkayyal; Martina L Jones; Stephen M Mahler; Anwar M Hashem
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Review 9.  Multifaceted Interweaving Between Extracellular Matrix, Insulin Resistance, and Skeletal Muscle.

Authors:  Khurshid Ahmad; Eun Ju Lee; Jun Sung Moon; So-Young Park; Inho Choi
Journal:  Cells       Date:  2018-09-22       Impact factor: 6.600

10.  Effects of Roux-en-Y gastric bypass on circulating follistatin, activin A, and peripheral ActRIIB signaling in humans with obesity and type 2 diabetes.

Authors:  Tang Cam Phung Pham; Kirstine Nyvold Bojsen-Møller; Sten Madsbad; Jørgen Frank Pind Wojtaszewski; Erik Arne Richter; Lykke Sylow
Journal:  Int J Obes (Lond)       Date:  2020-09-01       Impact factor: 5.095

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