Literature DB >> 28593453

Targeting Small Bowel Receptors to Treat Constipation and Diarrhea.

Elizabeth S John1, Sita Chokhavatia2.   

Abstract

BACKGROUND: The options for the treatment of diarrhea and constipation are evolving as emerging therapies target small bowel receptors. The goal of this review is to discuss small bowel receptors involved in intestinal absorption, secretion, and motility. The review highlights therapies already approved or currently being studied for the modulation of these receptors.
METHODS: The articles cited in this review focus on the molecular level of pathways involved in diarrhea and constipation, and highlight the respective pharmacotherapies.
RESULTS: The majority of the studies in the current literature investigate the effects of both the small and large intestine receptors on diarrhea and constipation. There are fewer studies that isolate the effects of these receptors solely on the small bowel, and focusing more on the receptors found distinctly in the small intestine may be an area of interest for future studies as this can inspire more targeted therapies.

Entities:  

Keywords:  Constipation; Diarrhea; Gastroenterology; Small bowel receptors; Small intestine

Mesh:

Substances:

Year:  2017        PMID: 28593453     DOI: 10.1007/s11894-017-0573-x

Source DB:  PubMed          Journal:  Curr Gastroenterol Rep        ISSN: 1522-8037


  51 in total

Review 1.  Muscarinic receptor subtypes of the bladder and gastrointestinal tract.

Authors:  Toshimitsu Uchiyama; Russell Chess-Williams
Journal:  J Smooth Muscle Res       Date:  2004-12

2.  A randomized trial of 5-hydroxytryptamine4-receptor agonist, YKP10811, on colonic transit and bowel function in functional constipation.

Authors:  Andrea Shin; Andres Acosta; Michael Camilleri; Amy Boldingh; Duane Burton; Michael Ryks; Deborah Rhoten; Alan R Zinsmeister
Journal:  Clin Gastroenterol Hepatol       Date:  2014-08-19       Impact factor: 11.382

Review 3.  Postoperative ileus: Recent developments in pathophysiology and management.

Authors:  Damian Bragg; Ahmed M El-Sharkawy; Emmanouil Psaltis; Charles A Maxwell-Armstrong; Dileep N Lobo
Journal:  Clin Nutr       Date:  2015-01-31       Impact factor: 7.324

4.  Sensitization of enteric neurons to morphine by HIV-1 Tat protein.

Authors:  S Fitting; J Ngwainmbi; M Kang; F A Khan; D L Stevens; W L Dewey; P E Knapp; K F Hauser; H I Akbarali
Journal:  Neurogastroenterol Motil       Date:  2015-02-19       Impact factor: 3.598

Review 5.  Chronic Diarrhea: Diagnosis and Management.

Authors:  Lawrence R Schiller; Darrell S Pardi; Joseph H Sellin
Journal:  Clin Gastroenterol Hepatol       Date:  2016-08-02       Impact factor: 11.382

6.  What about clonidine for diarrhoea? A systematic review and meta-analysis of its effect in humans.

Authors:  Konstantinos C Fragkos; Natalia Zárate-Lopez; Christos C Frangos
Journal:  Therap Adv Gastroenterol       Date:  2016-01-25       Impact factor: 4.409

7.  Effect of a chloride channel activator, lubiprostone, on colonic sensory and motor functions in healthy subjects.

Authors:  Seth Sweetser; Irene A Busciglio; Michael Camilleri; Adil E Bharucha; Lawrence A Szarka; Athanasios Papathanasopoulos; Duane D Burton; Deborah J Eckert; Alan R Zinsmeister
Journal:  Am J Physiol Gastrointest Liver Physiol       Date:  2008-11-25       Impact factor: 4.052

8.  The expanding role of somatostatin analogs in the management of neuroendocrine tumors.

Authors:  Edward M Wolin
Journal:  Gastrointest Cancer Res       Date:  2012-09

Review 9.  Lubiprostone Is Effective in the Treatment of Chronic Idiopathic Constipation and Irritable Bowel Syndrome: A Systematic Review and Meta-Analysis of Randomized Controlled Trials.

Authors:  Fan Li; Tao Fu; Wei-Dong Tong; Bao-Hua Liu; Chun-Xue Li; Yu Gao; Jin-Song Wu; Xiang-Feng Wang; An-Ping Zhang
Journal:  Mayo Clin Proc       Date:  2016-04       Impact factor: 7.616

Review 10.  Optimizing the Use of Linaclotide in Patients with Constipation-Predominant Irritable Bowel Syndrome: An Expert Consensus Report.

Authors:  Enrique Rey; Fermín Mearin; Javier Alcedo; Constanza Ciriza; Silvia Delgado-Aros; Teresa Freitas; Miguel Mascarenhas; Miguel Mínguez; Javier Santos; Jordi Serra
Journal:  Adv Ther       Date:  2017-01-12       Impact factor: 3.845

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  1 in total

1.  Paracellular Filtration Secretion Driven by Mechanical Force Contributes to Small Intestinal Fluid Dynamics.

Authors:  Randal K Buddington; Thomas Wong; Scott C Howard
Journal:  Med Sci (Basel)       Date:  2021-02-09
  1 in total

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