Literature DB >> 28577687

True rate of mineralocorticoid receptor antagonists-related hyperkalemia in placebo-controlled trials: A meta-analysis.

Davor Vukadinović1, Daniel Lavall2, Aleksandra Nikolovska Vukadinović2, Bertram Pitt3, Stefan Wagenpfeil4, Michael Böhm2.   

Abstract

BACKGROUND: Mineralocorticoid receptor antagonists (MRA) improve survival in heart failure with reduced ejection fraction but are often underused, mostly due to concerns of hyperkalemia. Because hyperkalemia occurs also on placebo, we aimed to determine the truly MRA-related rate of hyperkalemia.
METHODS: We performed a meta-analysis including randomized, placebo-controlled trials reporting hyperkalemia on MRAs in patients after myocardial infarction or with chronic heart failure. We evaluated the truly MRA-related rate of hyperkalemia that represents hyperkalemia on MRA, corrected for hyperkalemia on placebo (Pla), according to the equation: True MRA (%)=(MRA (%) - Pla (%))/MRA (%).
RESULTS: A total number of 16,065 patients from 7 trials were analyzed. Hyperkalemia was more frequently observed on MRA (9.3%) vs placebo (4.3%) (risk ratio 2.17, 95% CI 1.92-2.45, P<.0001). Truly MRA-related hyperkalemia was 54%, whereas 46% were non-MRA related. In trials using eplerenone, hyperkalemia was documented in 5.0% on eplerenone and in 2.6% on placebo (P<.0001). In spironolactone trials, hyperkalemia was documented in 17.5% and in 7.5% of patients on placebo (P=.0001). Hypokalemia occurred less frequently in patients on MRA (9.3%) compared with placebo (14.8%) (risk ratio 0.58, CI 0.47-0.72, P<.0001).
CONCLUSION: This meta-analysis shows that in clinical trials, 54% of hyperkalemia cases were specifically related to the MRA treatment and 46% to other reasons. Therefore, non-MRA-related rises in potassium levels might be underestimated and should be rigorously explored before cessation of the evidence-based therapy with MRAs.
Copyright © 2017 Elsevier Inc. All rights reserved.

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Year:  2017        PMID: 28577687     DOI: 10.1016/j.ahj.2017.03.011

Source DB:  PubMed          Journal:  Am Heart J        ISSN: 0002-8703            Impact factor:   4.749


  15 in total

1.  Single- and multiple-dose escalation study to assess pharmacokinetics, pharmacodynamics and safety of oral esaxerenone in healthy Japanese subjects.

Authors:  Manabu Kato; Hidetoshi Furuie; Takako Shimizu; Atsuhiro Miyazaki; Fumiaki Kobayashi; Hitoshi Ishizuka
Journal:  Br J Clin Pharmacol       Date:  2018-06-07       Impact factor: 4.335

Review 2.  Hyperkalaemia in Heart Failure-Pathophysiology, Implications and Therapeutic Perspectives.

Authors:  Redi Llubani; Davor Vukadinović; Christian Werner; Nikolaus Marx; Stephen Zewinger; Michael Böhm
Journal:  Curr Heart Fail Rep       Date:  2018-12

3.  Efficacy and Safety of Esaxerenone (CS-3150) for the Treatment of Type 2 Diabetes with Microalbuminuria: A Randomized, Double-Blind, Placebo-Controlled, Phase II Trial.

Authors:  Sadayoshi Ito; Kenichi Shikata; Masaomi Nangaku; Yasuyuki Okuda; Tomoko Sawanobori
Journal:  Clin J Am Soc Nephrol       Date:  2019-06-27       Impact factor: 8.237

4.  Hyperkalemia Risk with Finerenone: Results from the FIDELIO-DKD Trial.

Authors:  Rajiv Agarwal; Amer Joseph; Stefan D Anker; Gerasimos Filippatos; Peter Rossing; Luis M Ruilope; Bertram Pitt; Peter Kolkhof; Charlie Scott; Robert Lawatscheck; Daniel J Wilson; George L Bakris
Journal:  J Am Soc Nephrol       Date:  2021-11-03       Impact factor: 10.121

Review 5.  [Update on heart failure].

Authors:  J Wintrich; I Kindermann; M Böhm
Journal:  Herz       Date:  2018-06-05       Impact factor: 1.443

6.  Mineralocorticoid receptor antagonist use after hospitalization of patients with heart failure and post-discharge outcomes: a single-center retrospective cohort study.

Authors:  Matthew S Durstenfeld; Stuart D Katz; Hannah Park; Saul Blecker
Journal:  BMC Cardiovasc Disord       Date:  2019-08-09       Impact factor: 2.298

Review 7.  Hyperkalemia: pathophysiology, risk factors and consequences.

Authors:  Robert W Hunter; Matthew A Bailey
Journal:  Nephrol Dial Transplant       Date:  2019-12-01       Impact factor: 7.186

Review 8.  Spotlight on Spironolactone Oral Suspension for the Treatment of Heart Failure: Focus on Patient Selection and Perspectives.

Authors:  Antonis A Manolis; Theodora A Manolis; Helen Melita; Antonis S Manolis
Journal:  Vasc Health Risk Manag       Date:  2019-12-30

9.  Synergistic reduction in albuminuria in type 2 diabetic mice by esaxerenone (CS-3150), a novel nonsteroidal selective mineralocorticoid receptor blocker, combined with an angiotensin II receptor blocker.

Authors:  Kiyoshi Arai; Yuka Morikawa; Naoko Ubukata; Kotaro Sugimoto
Journal:  Hypertens Res       Date:  2020-07-02       Impact factor: 3.872

10.  Perspective Review: Type 2 Diabetes and Readmission for Heart Failure.

Authors:  Merlin C Thomas
Journal:  Clin Med Insights Cardiol       Date:  2018-06-05
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