Literature DB >> 28405826

Everolimus as first line therapy for pancreatic neuroendocrine tumours: current knowledge and future perspectives.

Marco Gallo1, Pasqualino Malandrino2, Giuseppe Fanciulli3, Francesca Rota4, Antongiulio Faggiano5, Annamaria Colao6.   

Abstract

PURPOSE: Everolimus has been shown to be effective for advanced pancreatic neuroendocrine tumours (pNETs), but its positioning in the therapeutic algorithm for pNETs is matter of debate.
METHODS: With the aim to shed light on this point, we performed an up-to-date critical review taking into account the results of both retrospective and prospective published studies, and the recommendations of international guidelines. In addition, we performed an extensive search on the Clinical Trial Registries databases worldwide, to gather information on the ongoing clinical trials related to this specific topic.
RESULTS: We identified eight retrospective published studies, two prospective published studies, and five registered clinical trials. Moreover, we analyzed the content of four widespread international guidelines.
CONCLUSIONS: Our critical review confirms the lack of high-quality data to recommend everolimus as the first line therapy for pNETs. The ongoing clinical trials reported in this review will hopefully help clinicians, in the near future, to better evaluate the role of everolimus as the first line therapy for pNETs. However, at the moment, there is already enough evidence to recommend everolimus as the first line therapy for patients with symptomatic malignant unresectable insulin-secreting pNETs, to control the endocrine syndrome regardless of tumour growth.

Entities:  

Keywords:  Everolimus; Neuroendocrine tumours; Therapy; mTOR inhibitors

Mesh:

Substances:

Year:  2017        PMID: 28405826     DOI: 10.1007/s00432-017-2407-5

Source DB:  PubMed          Journal:  J Cancer Res Clin Oncol        ISSN: 0171-5216            Impact factor:   4.553


  72 in total

1.  ENETS Consensus Guidelines for the management of patients with liver and other distant metastases from neuroendocrine neoplasms of foregut, midgut, hindgut, and unknown primary.

Authors:  Marianne Pavel; Eric Baudin; Anne Couvelard; Eric Krenning; Kjell Öberg; Thomas Steinmüller; Martin Anlauf; Bertram Wiedenmann; Ramon Salazar
Journal:  Neuroendocrinology       Date:  2012-02-15       Impact factor: 4.914

2.  Everolimus in combination with octreotide long-acting repeatable in a first-line setting for patients with neuroendocrine tumors: an ITMO group study.

Authors:  Emilio Bajetta; Laura Catena; Nicola Fazio; Sara Pusceddu; Pamela Biondani; Giusi Blanco; Sergio Ricci; Michele Aieta; Francesca Pucci; Monica Valente; Nadia Bianco; Chiara Maria Mauri; Francesca Spada
Journal:  Cancer       Date:  2014-04-18       Impact factor: 6.860

3.  A cytosolic binding protein for the immunosuppressant FK506 has peptidyl-prolyl isomerase activity but is distinct from cyclophilin.

Authors:  J J Siekierka; S H Hung; M Poe; C S Lin; N H Sigal
Journal:  Nature       Date:  1989-10-26       Impact factor: 49.962

4.  Targets for cell cycle arrest by the immunosuppressant rapamycin in yeast.

Authors:  J Heitman; N R Movva; M N Hall
Journal:  Science       Date:  1991-08-23       Impact factor: 47.728

5.  mTOR activation in well differentiated pancreatic neuroendocrine tumors: a retrospective study on 34 cases.

Authors:  Chen-Fei Zhou; Jun Ji; Fei Yuan; Min Shi; Jun Zhang; Bing-Ya Liu; Zheng-Gang Zhu
Journal:  Hepatogastroenterology       Date:  2011 Nov-Dec

6.  Sunitinib malate for the treatment of pancreatic neuroendocrine tumors.

Authors:  Eric Raymond; Laetitia Dahan; Jean-Luc Raoul; Yung-Jue Bang; Ivan Borbath; Catherine Lombard-Bohas; Juan Valle; Peter Metrakos; Denis Smith; Aaron Vinik; Jen-Shi Chen; Dieter Hörsch; Pascal Hammel; Bertram Wiedenmann; Eric Van Cutsem; Shem Patyna; Dongrui Ray Lu; Carolyn Blanckmeister; Richard Chao; Philippe Ruszniewski
Journal:  N Engl J Med       Date:  2011-02-10       Impact factor: 91.245

7.  mTOR inhibitors response and mTOR pathway in pancreatic neuroendocrine tumors.

Authors:  Simona Falletta; Stefano Partelli; Corrado Rubini; Dominik Nann; Andrea Doria; Ilaria Marinoni; Vanessa Polenta; Carmelina Di Pasquale; Ettore Degli Uberti; Aurel Perren; Massimo Falconi; Maria Chiara Zatelli
Journal:  Endocr Relat Cancer       Date:  2016-10-03       Impact factor: 5.678

8.  Octreotide and the mTOR inhibitor RAD001 (everolimus) block proliferation and interact with the Akt-mTOR-p70S6K pathway in a neuro-endocrine tumour cell Line.

Authors:  Simona Grozinsky-Glasberg; Giulia Franchi; Mabel Teng; Chrysanthia A Leontiou; Antônio Ribeiro de Oliveira; Paolo Dalino; Nabila Salahuddin; Márta Korbonits; Ashley B Grossman
Journal:  Neuroendocrinology       Date:  2007-11-16       Impact factor: 4.914

9.  Target of rapamycin in yeast, TOR2, is an essential phosphatidylinositol kinase homolog required for G1 progression.

Authors:  J Kunz; R Henriquez; U Schneider; M Deuter-Reinhard; N R Movva; M N Hall
Journal:  Cell       Date:  1993-05-07       Impact factor: 41.582

10.  Efficacy of RAD001 (everolimus) and octreotide LAR in advanced low- to intermediate-grade neuroendocrine tumors: results of a phase II study.

Authors:  James C Yao; Alexandria T Phan; David Z Chang; Robert A Wolff; Kenneth Hess; Sanjay Gupta; Carmen Jacobs; Jeannette E Mares; Andrea N Landgraf; Asif Rashid; Funda Meric-Bernstam
Journal:  J Clin Oncol       Date:  2008-09-10       Impact factor: 44.544

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  3 in total

Review 1.  Pancreatic Neuroendocrine Tumors: Molecular Mechanisms and Therapeutic Targets.

Authors:  Chandra K Maharjan; Po Hien Ear; Catherine G Tran; James R Howe; Chandrikha Chandrasekharan; Dawn E Quelle
Journal:  Cancers (Basel)       Date:  2021-10-12       Impact factor: 6.639

2.  Expression of γ-globin genes in β-thalassemia patients treated with sirolimus: results from a pilot clinical trial (Sirthalaclin).

Authors:  Cristina Zuccato; Lucia Carmela Cosenza; Matteo Zurlo; Jessica Gasparello; Chiara Papi; Elisabetta D'Aversa; Giulia Breveglieri; Ilaria Lampronti; Alessia Finotti; Monica Borgatti; Chiara Scapoli; Alice Stievano; Monica Fortini; Eric Ramazzotti; Nicola Marchetti; Marco Prosdocimi; Maria Rita Gamberini; Roberto Gambari
Journal:  Ther Adv Hematol       Date:  2022-06-21

3.  Treatment of Erythroid Precursor Cells from β-Thalassemia Patients with Cinchona Alkaloids: Induction of Fetal Hemoglobin Production.

Authors:  Cristina Zuccato; Lucia Carmela Cosenza; Matteo Zurlo; Ilaria Lampronti; Monica Borgatti; Chiara Scapoli; Roberto Gambari; Alessia Finotti
Journal:  Int J Mol Sci       Date:  2021-12-14       Impact factor: 5.923

  3 in total

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