Literature DB >> 28368443

Continuous Kisspeptin Administration in Postmenopausal Women: Impact of Estradiol on Luteinizing Hormone Secretion.

Margaret F Lippincott1, Yee-Ming Chan1,2, Dianali Rivera Morales1, Stephanie B Seminara1.   

Abstract

Context: Kisspeptin stimulates the reproductive endocrine cascade in both men and women. Circulating sex steroids are thought to modulate the ability of kisspeptin to stimulate gonadotropin-releasing hormone (GnRH)-induced luteinizing hormone (LH) release. Objective: To probe the effects of sex steroids on kisspeptin-stimulated GnRH-induced LH pulses. Participants: Eight healthy postmenopausal women. Intervention: Subjects underwent every-10-minute blood sampling to measure GnRH-induced LH secretion at baseline and in response to a continuous kisspeptin infusion (12.5 µg/kg/h) over 24 hours. A subset of the participants also received kisspeptin (0.313 µg/kg) and GnRH (75 ng/kg) intravenous boluses.
Results: Postmenopausal women are resistant to the stimulatory effect of continuous kisspeptin on LH secretion. Postmenopausal women receiving estradiol replacement therapy are also resistant to kisspeptin initially, but they demonstrate a significant increase in LH pulse amplitude in direct proportion to the circulating estradiol concentration and duration of kisspeptin administration. Conclusions: Kisspeptin administration has complex effects on GnRH, and by extension, on LH secretion. The ability of kisspeptin to affect LH secretion can be modulated by the ambient sex-steroid milieu in a time- and dose-dependent manner.
Copyright © 2017 Endocrine Society

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Year:  2017        PMID: 28368443      PMCID: PMC5470760          DOI: 10.1210/jc.2016-3952

Source DB:  PubMed          Journal:  J Clin Endocrinol Metab        ISSN: 0021-972X            Impact factor:   5.958


  47 in total

1.  Peripheral administration of kisspeptin-10 increases plasma concentrations of GH as well as LH in prepubertal Holstein heifers.

Authors:  H Kadokawa; M Matsui; K Hayashi; N Matsunaga; C Kawashima; T Shimizu; K Kida; A Miyamoto
Journal:  J Endocrinol       Date:  2008-02       Impact factor: 4.286

2.  Ontogeny and mechanisms of action for the stimulatory effect of kisspeptin on gonadotropin-releasing hormone system of the rat.

Authors:  J M Castellano; V M Navarro; R Fernández-Fernández; J P Castaño; M M Malagón; E Aguilar; C Dieguez; P Magni; L Pinilla; M Tena-Sempere
Journal:  Mol Cell Endocrinol       Date:  2006-08-22       Impact factor: 4.102

3.  Evidence that GnRH decreases with gonadal steroid feedback but increases with age in postmenopausal women.

Authors:  Sabrina Gill; Julie L Sharpless; Kimberly Rado; Janet E Hall
Journal:  J Clin Endocrinol Metab       Date:  2002-05       Impact factor: 5.958

4.  Kisspeptin Induces Dynamic Chromatin Modifications to Control GnRH Gene Expression.

Authors:  H J Novaira; M L Sonko; S Radovick
Journal:  Mol Neurobiol       Date:  2015-06-17       Impact factor: 5.590

5.  Advanced vaginal opening and precocious activation of the reproductive axis by KiSS-1 peptide, the endogenous ligand of GPR54.

Authors:  V M Navarro; R Fernández-Fernández; J M Castellano; J Roa; A Mayen; M L Barreiro; F Gaytan; E Aguilar; L Pinilla; C Dieguez; M Tena-Sempere
Journal:  J Physiol       Date:  2004-10-14       Impact factor: 5.182

6.  Kisspeptin increases GnRH mRNA expression and secretion in GnRH secreting neuronal cell lines.

Authors:  Horacio J Novaira; Yewade Ng; Andrew Wolfe; Sally Radovick
Journal:  Mol Cell Endocrinol       Date:  2009-07-01       Impact factor: 4.102

7.  The GPR54 gene as a regulator of puberty.

Authors:  Stephanie B Seminara; Sophie Messager; Emmanouella E Chatzidaki; Rosemary R Thresher; James S Acierno; Jenna K Shagoury; Yousef Bo-Abbas; Wendy Kuohung; Kristine M Schwinof; Alan G Hendrick; Dirk Zahn; John Dixon; Ursula B Kaiser; Susan A Slaugenhaupt; James F Gusella; Stephen O'Rahilly; Mark B L Carlton; William F Crowley; Samuel A J R Aparicio; William H Colledge
Journal:  N Engl J Med       Date:  2003-10-23       Impact factor: 91.245

8.  Hypogonadotropic hypogonadism due to loss of function of the KiSS1-derived peptide receptor GPR54.

Authors:  Nicolas de Roux; Emmanuelle Genin; Jean-Claude Carel; Fumihiko Matsuda; Jean-Louis Chaussain; Edwin Milgrom
Journal:  Proc Natl Acad Sci U S A       Date:  2003-08-27       Impact factor: 11.205

9.  Regulation of GPR54 signaling by GRK2 and {beta}-arrestin.

Authors:  Macarena Pampillo; Natasha Camuso; Jay E Taylor; Jacob M Szereszewski; Maryse R Ahow; Mateusz Zajac; Robert P Millar; Moshmi Bhattacharya; Andy V Babwah
Journal:  Mol Endocrinol       Date:  2009-10-21

10.  The effects of kisspeptin-10 on reproductive hormone release show sexual dimorphism in humans.

Authors:  Channa N Jayasena; Gurjinder M K Nijher; Alexander N Comninos; Ali Abbara; Adam Januszewki; Meriel L Vaal; Labosshy Sriskandarajah; Kevin G Murphy; Zohreh Farzad; Mohammad A Ghatei; Stephen R Bloom; Waljit S Dhillo
Journal:  J Clin Endocrinol Metab       Date:  2011-10-05       Impact factor: 5.958

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  2 in total

Review 1.  Does the KNDy Model for the Control of Gonadotropin-Releasing Hormone Pulses Apply to Monkeys and Humans?

Authors:  Michael N Lehman; Wen He; Lique M Coolen; Jon E Levine; Robert L Goodman
Journal:  Semin Reprod Med       Date:  2019-12-17       Impact factor: 1.912

2.  Assessing Sex Steroid Influence on Kisspeptin Responsiveness in Idiopathic Hypogonadotropic Hypogonadism.

Authors:  Margaret F Lippincott; Kiana Nguyen; Angela Delaney; Yee-Ming Chan; Stephanie Beth Seminara
Journal:  J Endocr Soc       Date:  2018-09-20
  2 in total

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