Literature DB >> 28244745

The Ecstasy and Agony of Assay Interference Compounds.

Courtney Aldrich1, Carolyn Bertozzi2, Gunda I Georg3, Laura Kiessling4, Craig Lindsley5, Dennis Liotta6, Kenneth M Merz7, Alanna Schepartz8, Shaomeng Wang3.   

Abstract

Mesh：

Substances：

Year:  2017        PMID： 28244745     DOI： 10.1021/acs.jmedchem.7b00229

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


× No keyword cloud information.
  30 in total

1.  Customizable de novo design strategies for DOCK: Application to HIVgp41 and other therapeutic targets.

Authors:  William J Allen; Brian C Fochtman; Trent E Balius; Robert C Rizzo
Journal:  J Comput Chem       Date:  2017-09-22       Impact factor: 3.376

2.  Colloidal Drug Aggregate Stability in High Serum Conditions and Pharmacokinetic Consequence.

Authors:  Ahil N Ganesh; Ahmed Aman; Jennifer Logie; Ben L Barthel; Peter Cogan; Rima Al-Awar; Tad H Koch; Brian K Shoichet; Molly S Shoichet
Journal:  ACS Chem Biol       Date:  2019-03-12       Impact factor: 5.100

3.  Small-Molecule Inhibitors of Haemophilus influenzae IgA1 Protease.

Authors:  Livia Shehaj; Santosh K Choudary; Kamlesh M Makwana; Mary C Gallo; Timothy F Murphy; Joshua A Kritzer
Journal:  ACS Infect Dis       Date:  2019-05-03       Impact factor: 5.084

4.  Argininamide-type neuropeptide Y Y1 receptor antagonists: the nature of N ω-carbamoyl substituents determines Y1R binding mode and affinity.

Authors:  Jonas Buschmann; Theresa Seiler; Günther Bernhardt; Max Keller; David Wifling
Journal:  RSC Med Chem       Date:  2020-01-20

5.  Discovery of the First Vitamin K Analogue as a Potential Treatment of Pharmacoresistant Seizures.

Authors:  Xiaoyang Li; Richard A Himes; Lyndsey C Prosser; Charleston F Christie; Emma Watt; Sharon F Edwards; Cameron S Metcalf; Peter J West; Karen S Wilcox; Sherine S L Chan; C James Chou
Journal:  J Med Chem       Date:  2020-05-22       Impact factor: 7.446

6.  Colloidal aggregation: from screening nuisance to formulation nuance.

Authors:  Ahil N Ganesh; Eric N Donders; Brian K Shoichet; Molly S Shoichet
Journal:  Nano Today       Date:  2018-03-10       Impact factor: 20.722

7.  Protein Stability Effects in Aggregate-Based Enzyme Inhibition.

Authors:  Hayarpi Torosyan; Brian K Shoichet
Journal:  J Med Chem       Date:  2019-10-17       Impact factor: 7.446

8.  Reevaluating the Substrate Specificity of the L-Type Amino Acid Transporter (LAT1).

Authors:  Huan-Chieh Chien; Claire Colas; Karissa Finke; Seth Springer; Laura Stoner; Arik A Zur; Brooklynn Venteicher; Jerome Campbell; Colton Hall; Andrew Flint; Evan Augustyn; Christopher Hernandez; Nathan Heeren; Logan Hansen; Abby Anthony; Justine Bauer; Dimitrios Fotiadis; Avner Schlessinger; Kathleen M Giacomini; Allen A Thomas
Journal:  J Med Chem       Date:  2018-08-10       Impact factor: 7.446

9.  Small-Molecule Inhibitors of the CD40-CD40L Costimulatory Protein-Protein Interaction.

Authors:  Jinshui Chen; Yun Song; Damir Bojadzic; Alejandro Tamayo-Garcia; Ana Marie Landin; Bonnie B Blomberg; Peter Buchwald
Journal:  J Med Chem       Date:  2017-10-25       Impact factor: 7.446

10.  PAIN-less identification and evaluation of small molecule inhibitors against protein tyrosine phosphatase 1B.

Authors:  Hamid R Nasiri; Philipp Mracek; Steffen K Grimm; Janine Gastaldello; Adrian Kolodzik; Dirk Ullmann
Journal:  Medchemcomm       Date:  2017-04-07       Impact factor: 3.597
View more

北京卡尤迪生物科技股份有限公司 © 2022-2023.