Literature DB >> 27977318

Nebulized Recombinant Human Tissue Factor Pathway Inhibitor Attenuates Coagulation and Exerts Modest Anti-inflammatory Effects in Rat Models of Lung Injury.

Florry E van den Boogaard1,2,3, Jorrit J Hofstra1,4, Xanthe Brands1,2, Marcel M Levi5, Joris J T H Roelofs6, Sebastiaan A J Zaat3,4, Cornelis Van't Veer2,3, Tom van der Poll2,3,7, Marcus J Schultz1,8.   

Abstract

BACKGROUND: Critically ill patients are at a constant risk of direct (e.g., by pneumonia) or indirect lung injury (e.g., by sepsis). Excessive alveolar fibrin deposition is a prominent feature of lung injury, undermining pulmonary integrity and function.
METHODS: We examined the effect of local administration of recombinant human tissue factor pathway inhibitor (rh-TFPI), a natural anticoagulant, in two well-established models of lung injury in rats. Rats received intratracheal instillation of Pseudomonas aeruginosa, causing direct lung injury, or they received an intravenous injection of Escherichia coli lipopolysaccharide (LPS), causing indirect lung injury. Rats were randomized to local treatment with rh-TFPI or placebo through repeated nebulization.
RESULTS: Challenge with P. aeruginosa or LPS was associated with increased coagulation and decreased fibrinolysis in bronchoalveolar lavage fluid (BALF) and plasma. Rh-TFPI levels in BALF increased after nebulization, whereas plasma rh-TFPI levels remained low and systemic TFPI activity was not affected. Nebulization of rh-TFPI attenuated pulmonary and systemic coagulation in both models, without affecting fibrinolysis. Nebulization of rh-TFPI modestly reduced the inflammatory response and bacterial growth of P. aeruginosa in the alveolar compartment.
CONCLUSIONS: Local treatment with rh-TFPI does not alter systemic TFPI activity; however, it attenuates both pulmonary and systemic coagulopathy. Furthermore, nebulized rh-TFPI modestly reduces the pulmonary inflammatory response and allows increased bacterial clearance in rats with direct lung injury caused by P. aeruginosa.

Entities:  

Keywords:  Pseudomonas aeruginosa; coagulation; endotoxemia; lung; pneumonia; tissue factor pathway inhibitor

Mesh:

Substances:

Year:  2016        PMID: 27977318     DOI: 10.1089/jamp.2016.1317

Source DB:  PubMed          Journal:  J Aerosol Med Pulm Drug Deliv        ISSN: 1941-2711            Impact factor:   2.849


  7 in total

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Journal:  Ann Transl Med       Date:  2018-01

Review 2.  Nebulized anticoagulants in lung injury in critically ill patients-an updated systematic review of preclinical and clinical studies.

Authors:  Jenny Juschten; Pieter R Tuinman; Nicole P Juffermans; Barry Dixon; Marcel Levi; Marcus J Schultz
Journal:  Ann Transl Med       Date:  2017-11

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Journal:  Crit Care       Date:  2020-06-19       Impact factor: 9.097

4.  ZNF354C Mediated by DNMT1 Ameliorates Lung Ischemia-Reperfusion Oxidative Stress Injury by Reducing TFPI Promoter Methylation to Upregulate TFPI.

Authors:  Qi Shi; Nana Feng; Qingyun Ma; Shaohua Wang; Huijun Zhang; Dayu Huang; Jiayuan Sun; Meng Shi
Journal:  Oxid Med Cell Longev       Date:  2022-07-19       Impact factor: 7.310

Review 5.  Targeting coagulation activation in severe COVID-19 pneumonia: lessons from bacterial pneumonia and sepsis.

Authors:  Ricardo J José; Andrew Williams; Ari Manuel; Jeremy S Brown; Rachel C Chambers
Journal:  Eur Respir Rev       Date:  2020-10-01

6.  Unfractionated heparin improves the clinical efficacy in adult sepsis patients: a systematic review and meta-analysis.

Authors:  Sifeng Fu; Sihan Yu; Liang Wang; Xiaochun Ma; Xu Li
Journal:  BMC Anesthesiol       Date:  2022-01-21       Impact factor: 2.217

7.  Different Profiles of Cytokines, Chemokines and Coagulation Mediators Associated with Severity in Brazilian Patients Infected with Dengue Virus.

Authors:  Victor Edgar Fiestas Solórzano; Nieli Rodrigues da Costa Faria; Caroline Fernandes Dos Santos; Gladys Corrêa; Márcio da Costa Cipitelli; Marcos Dornelas Ribeiro; Luiz José de Souza; Paulo Vieira Damasco; Rivaldo Venâncio da Cunha; Flavia Barreto Dos Santos; Luzia Maria de Oliveira Pinto; Elzinandes Leal de Azeredo
Journal:  Viruses       Date:  2021-09-08       Impact factor: 5.048

  7 in total

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