Literature DB >> 27942928

Efficacy and safety of everolimus and sunitinib in patients with gastroenteropancreatic neuroendocrine tumor.

Changhoon Yoo1, Hyungwoo Cho1, Min Jeong Song2, Seung-Mo Hong2, Kyu-Pyo Kim1, Heung-Moon Chang1, Heejung Chae1, Tae Won Kim1, Yong Sang Hong1, Min-Hee Ryu1, Yoon-Koo Kang1, Song Cheol Kim3, Baek-Yeol Ryoo4.   

Abstract

PURPOSE: Efficacy of targeted agents, such as everolimus and sunitinib, has been demonstrated in prospective trials on patients with gastroenteropancreatic neuroendocrine tumors (GEP-NETs). Considering the heterogeneous clinicopathological characteristics of neuroendocrine tumors (NETs), evaluation of treatment outcomes in a real-world setting is necessary.
METHODS: Clinical records of 44 patients with GEP-NET who were treated with everolimus or sunitinib between March 2007 and October 2014 were retrospectively reviewed. Considering the distinct characteristics of pancreatic NETs (pNETs) and non-pancreatic gastrointestinal NETs (GI-NETs), efficacy analysis was performed separately.
RESULTS: Pancreas was the most common primary site (n = 28, 64%), followed by rectum (n = 10, 23%) and stomach (n = 3, 7%). Sunitinib and everolimus were administered in 27 (61%) and 17 (39%) patients, respectively. In patients with pNET, median progression-free survival (PFS) with everolimus and sunitinib was 16.6 months (95% CI 8.0-25.1) and 8.0 months (95% CI 0.0-17.4), respectively (p = 0.51). Among non-pancreatic GI-NET patients, median PFS with everolimus and sunitinib was 14.7 months (95% CI 2.4-27.0) and 1.7 months (95% CI 0.5-3.0), respectively (p = 0.001). Compared to patients treated with everolimus, tumor grade 3 (30 vs. 0%) and history of prior cytotoxic chemotherapy (70 vs. 50%) were more common in patients treated with sunitinib.
CONCLUSIONS: Both everolimus and sunitinib were effective in GEP-NET patients. Outcomes of everolimus therapy in GEP-NETs were consistent with those reported elsewhere. Poor efficacy of sunitinib in non-pancreatic GI-NETs may be attributable to the baseline characteristics associated with poor clinical outcomes.

Entities:  

Keywords:  Everolimus; Gastroenteropancreatic; Neuroendocrine tumor; Sunitinib

Mesh:

Substances:

Year:  2016        PMID: 27942928     DOI: 10.1007/s00280-016-3215-3

Source DB:  PubMed          Journal:  Cancer Chemother Pharmacol        ISSN: 0344-5704            Impact factor:   3.333


  10 in total

1.  Efficacy and safety of lanreotide in Korean patients with metastatic, well-differentiated gastroenteropancreatic-neuroendocrine tumors: a retrospective analysis.

Authors:  Junho Kang; Changhoon Yoo; Hee-Sang Hwang; Seung-Mo Hong; Kyu-Pyo Kim; Sun Young Kim; Yong-Sang Hong; Tae Won Kim; Baek-Yeol Ryoo
Journal:  Invest New Drugs       Date:  2018-12-10       Impact factor: 3.850

2.  EPB41L5 is Associated With the Metastatic Potential of Low-grade Pancreatic Neuroendocrine Tumors.

Authors:  James Saller; Shabnam Seydafkan; Mohammad Shahid; Manoj Gadara; Mauro Cives; Steven A Eschrich; David Boulware; Jonathan R Strosberg; Nasir Aejaz; Domenico Coppola
Journal:  Cancer Genomics Proteomics       Date:  2019 Sep-Oct       Impact factor: 4.069

3.  Extended cycle streptozotocin/5-FU chemotherapy for maintenance therapy in pancreatic neuroendocrine tumors.

Authors:  Joerg Schrader; Frank O Henes; Michael Blaeker; Katharina Zimmermann-Fraedrich; Andrea Pace; Daniel Perez; Jakob R Izbicki; Ansgar W Lohse; Daniel Benten
Journal:  Endocrine       Date:  2019-04-29       Impact factor: 3.633

4.  Everolimus in the treatment of neuroendocrine tumors: efficacy, side-effects, resistance, and factors affecting its place in the treatment sequence.

Authors:  Lingaku Lee; Tetsuhide Ito; Robert T Jensen
Journal:  Expert Opin Pharmacother       Date:  2018-05-24       Impact factor: 3.889

5.  Downgrading of a G3 Neuroendocrine Tumor to a G2 Tumor: Can First-Line Cytotoxic Chemotherapy Change the Tumor Biology?

Authors:  Andreas Blesl; Elisabeth Krones; Marion J Pollheimer; Johannes Haybaeck; Ulrike Wiesspeiner; Rainer W Lipp; Patrizia Kump
Journal:  Case Rep Oncol       Date:  2017-12-20

Review 6.  Emerging use of everolimus in the treatment of neuroendocrine tumors.

Authors:  Pablo Gajate; Olga Martínez-Sáez; Teresa Alonso-Gordoa; Enrique Grande
Journal:  Cancer Manag Res       Date:  2017-06-20       Impact factor: 3.989

7.  Oncolytic vaccinia virus GLV-1h68 exhibits profound antitumoral activities in cell lines originating from neuroendocrine neoplasms.

Authors:  Linus D Kloker; Susanne Berchtold; Irina Smirnow; Julia Beil; Andreas Krieg; Bence Sipos; Ulrich M Lauer
Journal:  BMC Cancer       Date:  2020-07-06       Impact factor: 4.430

8.  Anti-tumour activity of everolimus and sunitinib in neuroendocrine neoplasms.

Authors:  Kosmas Daskalakis; Marina Tsoli; Anna Angelousi; Evanthia Kassi; Krystallenia I Alexandraki; Denise Kolomodi; Gregory Kaltsas; Anna Koumarianou
Journal:  Endocr Connect       Date:  2019-06       Impact factor: 3.335

Review 9.  Management of Gastrointestinal Neuroendocrine Tumors.

Authors:  Rongzhi Wang; Rui Zheng-Pywell; H Alexander Chen; James A Bibb; Herbert Chen; J Bart Rose
Journal:  Clin Med Insights Endocrinol Diabetes       Date:  2019-10-24

10.  Therapeutic strategies for gastroenteropancreatic neuroendocrine neoplasms: State-of-the-art and future perspectives.

Authors:  Elettra Merola; Andrea Michielan; Umberto Rozzanigo; Marco Erini; Sandro Sferrazza; Stefano Marcucci; Chiara Sartori; Chiara Trentin; Giovanni de Pretis; Franca Chierichetti
Journal:  World J Gastrointest Surg       Date:  2022-02-27
  10 in total

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