Literature DB >> 27913920

NS5A resistance-associated variants undermine the effectiveness of ledipasvir and sofosbuvir for cirrhotic patients infected with HCV genotype 1b.

Eiichi Ogawa1, Norihiro Furusyo1, Hideyuki Nomura2, Kazufumi Dohmen3, Nobuhiko Higashi4, Kazuhiro Takahashi5, Akira Kawano6, Koichi Azuma7, Takeaki Satoh8, Makoto Nakamuta9, Toshimasa Koyanagi10, Masaki Kato11, Shinji Shimoda12, Eiji Kajiwara13, Jun Hayashi14.   

Abstract

BACKGROUND: Little real-world cohort data has been reported for Asians who have received interferon-free regimens with sofosbuvir (SOF) for chronic hepatitis C virus (HCV) infection. We evaluated the effectiveness and safety in clinical practice of ledipasvir (LDV) plus SOF for Japanese patients infected with HCV genotype 1.
METHODS: This large, multicenter, real-world cohort study consisted of 772 patients treatment-naive or -experienced, with or without compensated cirrhosis, who were treated with LDV (90 mg)/SOF (400 mg) for a fixed 12-week duration. Direct sequence analysis of the NS5A genes (L31 and Y93) was performed at baseline.
RESULTS: Almost all (99.6%) were infected with HCV genotype 1b. The overall sustained virological response 12 weeks after the end of treatment (SVR12) rate was 98.8% (763/772). Multivariable logistic regression analysis extracted male (odds ratio [OR] 6.62, p = 0.024), cirrhosis (OR 20.1, p = 0.0054), and baseline NS5A resistance-associated variants (RAVs) (OR 29.3, p = 0.0018) as independently associated with treatment failure. Notably, the SVR12 rate for cirrhosis patients with baseline NS5A RAVs (87.5%, 49/56) was statistically lower than for the other groups. This tendency was found except for patients with prior daclatasvir/asunaprevir failure. All patients with treatment failure had NS5A Y93H at relapse, whether or not they had NS5A RAVs at baseline. Serious adverse effects were very rare, and discontinuation was required for only five (0.6%) patients.
CONCLUSIONS: LDV/SOF for HCV genotype 1b was exceptionally effective, however, NS5A RAVs undermined the virological effect for cirrhosis patients. Moreover, LDV/SOF was shown to be safe, irrespective of age or fibrosis status.

Entities:  

Keywords:  Cirrhosis; DAA; Hepatitis C virus; Ledipasvir; Sofosbuvir

Mesh:

Substances:

Year:  2016        PMID: 27913920     DOI: 10.1007/s00535-016-1290-1

Source DB:  PubMed          Journal:  J Gastroenterol        ISSN: 0944-1174            Impact factor:   7.527


  19 in total

1.  Development of a simple noninvasive index to predict significant fibrosis in patients with HIV/HCV coinfection.

Authors:  Richard K Sterling; Eduardo Lissen; Nathan Clumeck; Ricard Sola; Mendes Cassia Correa; Julio Montaner; Mark S Sulkowski; Francesca J Torriani; Doug T Dieterich; David L Thomas; Diethelm Messinger; Mark Nelson
Journal:  Hepatology       Date:  2006-06       Impact factor: 17.425

2.  Evaluation of proton pump inhibitor use on treatment outcomes with ledipasvir and sofosbuvir in a real-world cohort study.

Authors:  Elliot B Tapper; Bruce R Bacon; Michael P Curry; Douglas T Dieterich; Steven L Flamm; Lauren E Guest; Kris V Kowdley; Yoori Lee; Naoky C Tsai; Zobair M Younossi; Nezam H Afdhal
Journal:  Hepatology       Date:  2016-10-05       Impact factor: 17.425

3.  Ledipasvir and sofosbuvir fixed-dose combination with and without ribavirin for 12 weeks in treatment-naive and previously treated Japanese patients with genotype 1 hepatitis C: an open-label, randomised, phase 3 trial.

Authors:  Masashi Mizokami; Osamu Yokosuka; Tetsuo Takehara; Naoya Sakamoto; Masaaki Korenaga; Hitoshi Mochizuki; Kunio Nakane; Hirayuki Enomoto; Fusao Ikeda; Mikio Yanase; Hidenori Toyoda; Takuya Genda; Takeji Umemura; Hiroshi Yatsuhashi; Tatsuya Ide; Nobuo Toda; Kazushige Nirei; Yoshiyuki Ueno; Yoichi Nishigaki; Juan Betular; Bing Gao; Akinobu Ishizaki; Masa Omote; Hongmei Mo; Kim Garrison; Phillip S Pang; Steven J Knox; William T Symonds; John G McHutchison; Namiki Izumi; Masao Omata
Journal:  Lancet Infect Dis       Date:  2015-04-08       Impact factor: 25.071

4.  Comparative effectiveness and safety study of triple therapy with simeprevir or telaprevir for non-cirrhotic patients with chronic hepatitis C virus genotype 1b infection.

Authors:  Eiichi Ogawa; Norihiro Furusyo; Eiji Kajiwara; Hideyuki Nomura; Akira Kawano; Kazuhiro Takahashi; Kazufumi Dohmen; Takeaki Satoh; Koichi Azuma; Makoto Nakamuta; Toshimasa Koyanagi; Kazuhiro Kotoh; Shinji Shimoda; Jun Hayashi
Journal:  J Gastroenterol Hepatol       Date:  2015-12       Impact factor: 4.029

5.  Evaluation of the adverse effect of premature discontinuation of pegylated interferon α-2b and ribavirin treatment for chronic hepatitis C virus infection: results from Kyushu University Liver Disease Study.

Authors:  Eiichi Ogawa; Norihiro Furusyo; Eiji Kajiwara; Kazuhiro Takahashi; Hideyuki Nomura; Yuichi Tanabe; Takeaki Satoh; Toshihiro Maruyama; Makoto Nakamuta; Kazuhiro Kotoh; Koichi Azuma; Kazufumi Dohmen; Shinji Shimoda; Jun Hayashi
Journal:  J Gastroenterol Hepatol       Date:  2012-07       Impact factor: 4.029

6.  The longitudinal quantitative assessment by transient elastography of chronic hepatitis C patients treated with pegylated interferon alpha-2b and ribavirin.

Authors:  Eiichi Ogawa; Norihiro Furusyo; Kazuhiro Toyoda; Hiroaki Takeoka; Shinji Maeda; Jun Hayashi
Journal:  Antiviral Res       Date:  2009-04-14       Impact factor: 5.970

7.  Peginterferon-alpha2a and ribavirin combination therapy in chronic hepatitis C: a randomized study of treatment duration and ribavirin dose.

Authors:  Stephanos J Hadziyannis; Hoel Sette; Timothy R Morgan; Vijayan Balan; Moises Diago; Patrick Marcellin; Giuliano Ramadori; Henry Bodenheimer; David Bernstein; Mario Rizzetto; Stefan Zeuzem; Paul J Pockros; Amy Lin; Andrew M Ackrill
Journal:  Ann Intern Med       Date:  2004-03-02       Impact factor: 25.391

8.  Effectiveness and safety of daclatasvir plus asunaprevir for patients with hepatitis C virus genotype 1b aged 75 years and over with or without cirrhosis.

Authors:  Eiichi Ogawa; Norihiro Furusyo; Naoki Yamashita; Akira Kawano; Kazuhiro Takahashi; Kazufumi Dohmen; Makoto Nakamuta; Takeaki Satoh; Hideyuki Nomura; Koichi Azuma; Toshimasa Koyanagi; Kazuhiro Kotoh; Shinji Shimoda; Eiji Kajiwara; Jun Hayashi
Journal:  Hepatol Res       Date:  2016-06-10       Impact factor: 4.288

9.  Effectiveness of Sofosbuvir, Ledipasvir/Sofosbuvir, or Paritaprevir/Ritonavir/Ombitasvir and Dasabuvir Regimens for Treatment of Patients With Hepatitis C in the Veterans Affairs National Health Care System.

Authors:  George N Ioannou; Lauren A Beste; Michael F Chang; Pamela K Green; Elliott Lowy; Judith I Tsui; Feng Su; Kristin Berry
Journal:  Gastroenterology       Date:  2016-06-04       Impact factor: 22.682

10.  Ledipasvir and sofosbuvir for previously treated HCV genotype 1 infection.

Authors:  Nezam Afdhal; K Rajender Reddy; David R Nelson; Eric Lawitz; Stuart C Gordon; Eugene Schiff; Ronald Nahass; Reem Ghalib; Norman Gitlin; Robert Herring; Jacob Lalezari; Ziad H Younes; Paul J Pockros; Adrian M Di Bisceglie; Sanjeev Arora; G Mani Subramanian; Yanni Zhu; Hadas Dvory-Sobol; Jenny C Yang; Phillip S Pang; William T Symonds; John G McHutchison; Andrew J Muir; Mark Sulkowski; Paul Kwo
Journal:  N Engl J Med       Date:  2014-04-11       Impact factor: 91.245

View more
  21 in total

Review 1.  2017 KASL clinical practice guidelines management of hepatitis C: Treatment of chronic hepatitis C.

Authors: 
Journal:  Clin Mol Hepatol       Date:  2018-08-10

2.  Grazoprevir/elbasvir treatment for the relapse of HCV genotype 1b infection after ledipasvir/sofosbuvir: A case report.

Authors:  Tomoko Tadokoro; Asahiro Morishita; Kyoko Oura; Koji Fujita; Shima Mimura; Teppei Sakamoto; Takako Nomura; Joji Tani; Hirohito Yoneyama; Tsutomu Masaki
Journal:  Exp Ther Med       Date:  2018-05-23       Impact factor: 2.447

3.  Health-related quality of life on the clinical course of patients with chronic hepatitis C receiving daclatasvir/asunaprevir therapy: A prospective observational study comparing younger (<70) and elderly (≥70) patients.

Authors:  Kazuki Ohashi; Toru Ishikawa; Mitsuyuki Suzuki; Hiroko Abe; Fujiko Koyama; Tomomi Nakano; Aya Ueki; Hirohito Noguchi; Erina Hasegawa; Shiori Hirosawa; Miki Kobayashi; Hiroshi Hirosawa; Kaede Sato; Takako Fukazawa; Yuka Maruyama; Toshiaki Yoshida
Journal:  Exp Ther Med       Date:  2017-11-10       Impact factor: 2.447

4.  TLL1 variant associated with development of hepatocellular carcinoma after eradication of hepatitis C virus by interferon-free therapy.

Authors:  Etsuko Iio; Kentaro Matsuura; Noritomo Shimada; Masanori Atsukawa; Norio Itokawa; Hiroshi Abe; Keizo Kato; Koichi Takaguchi; Tomonori Senoh; Yuichiro Eguchi; Hideyuki Nomura; Kai Yoshizawa; Jong-Hon Kang; Takeshi Matsui; Noboru Hirashima; Atsunori Kusakabe; Tomokatsu Miyaki; Kei Fujiwara; Kayoko Matsunami; Susumu Tsutsumi; Katsuhiko Iwakiri; Yasuhito Tanaka
Journal:  J Gastroenterol       Date:  2018-10-31       Impact factor: 7.527

5.  Validation of Modified ALBI Grade for More Detailed Assessment of Hepatic Function in Hepatocellular Carcinoma Patients: A Multicenter Analysis.

Authors:  Atsushi Hiraoka; Takashi Kumada; Kunihiko Tsuji; Koichi Takaguchi; Ei Itobayashi; Kazuya Kariyama; Hironori Ochi; Kazuto Tajiri; Masashi Hirooka; Noritomo Shimada; Toru Ishikawa; Yoshihiko Tachi; Toshifumi Tada; Hidenori Toyoda; Kazuhiro Nouso; Kouji Joko; Yoichi Hiasa; Kojiro Michitaka; Masatoshi Kudo
Journal:  Liver Cancer       Date:  2018-06-11       Impact factor: 11.740

6.  Real-world efficacy and safety of ledipasvir and sofosbuvir in patients with hepatitis C virus genotype 1 infection: a nationwide multicenter study by the Japanese Red Cross Liver Study Group.

Authors:  Keiji Tsuji; Masayuki Kurosaki; Jun Itakura; Nami Mori; Shintaro Takaki; Chitomi Hasebe; Takehiro Akahane; Kouji Joko; Hitoshi Yagisawa; Jirou Takezawa; Ryou Nakata; Atsunori Kusakabe; Yuji Kojima; Hiroyuki Kimura; Takashi Tamada; Haruhiko Kobashi; Akeri Mitsuda; Masahiko Kondou; Chikara Ogawa; Yasushi Uchida; Tetsuro Sohda; Ryouichi Narita; Namiki Izumi
Journal:  J Gastroenterol       Date:  2018-04-06       Impact factor: 6.772

7.  Efficacy and safety of sofosbuvir and ledipasvir in Japanese patients aged 75 years or over with hepatitis C genotype 1.

Authors:  Yoshinori Ozono; Kenji Nagata; Satoru Hasuike; Hisayoshi Iwakiri; Kenichi Nakamura; Mai Tsuchimochi; Yuri Yamada; Yuka Takaishi; Mitsue Sueta; Tadashi Miike; Yoshihiro Tahara; Shojiro Yamamoto; Kotaro Shide; Tomonori Hidaka; Yoko Kubuki; Kazunori Kusumoto; Toshimasa Ochiai; Junya Kato; Naoto Komada; Shuichi Hirono; Kazuo Kuroki; Masafumi Shigehira; Kazuya Shimoda
Journal:  World J Hepatol       Date:  2017-12-28

8.  Integrated Resistance Analysis of CERTAIN-1 and CERTAIN-2 Studies in Hepatitis C Virus-Infected Patients Receiving Glecaprevir and Pibrentasvir in Japan.

Authors:  Preethi Krishnan; Gretja Schnell; Rakesh Tripathi; Jill Beyer; Thomas Reisch; Tatyana Dekhtyar; Michelle Irvin; Wangang Xie; Bo Fu; Margaret Burroughs; Rebecca Redman; Hiromitsu Kumada; Kazuaki Chayama; Christine Collins; Tami Pilot-Matias
Journal:  Antimicrob Agents Chemother       Date:  2018-01-25       Impact factor: 5.191

9.  Long-Term Outcomes and Evaluation of Hepatocellular Carcinoma Recurrence after Hepatitis C Virus Eradication by Direct-Acting Antiviral Treatment: All Kagawa Liver Disease Group (AKLDG) Study.

Authors:  Joji Tani; Tomonori Senoh; Akio Moriya; Chikara Ogawa; Akihiro Deguchi; Teppei Sakamoto; Kei Takuma; Mai Nakahara; Kyoko Oura; Tomoko Tadokoro; Shima Mimura; Koji Fujita; Hirohito Yoneyama; Hideki Kobara; Asahiro Morishita; Takashi Himoto; Akemi Tsutsui; Takuya Nagano; Koichi Takaguchi; Tsutomu Masaki
Journal:  Cancers (Basel)       Date:  2021-05-08       Impact factor: 6.639

10.  Real-world virological efficacy and safety of elbasvir and grazoprevir in patients with chronic hepatitis C virus genotype 1 infection in Japan.

Authors:  Hidenori Toyoda; Masanori Atsukawa; Koichi Takaguchi; Tomonori Senoh; Kojiro Michitaka; Atsushi Hiraoka; Shinichi Fujioka; Chisa Kondo; Tomomi Okubo; Haruki Uojima; Toshifumi Tada; Hirohito Yoneyama; Tsunamasa Watanabe; Toru Asano; Toru Ishikawa; Hideyuki Tamai; Hiroshi Abe; Keizo Kato; Kunihiko Tsuji; Chikara Ogawa; Noritomo Shimada; Etsuko Iio; Akihiro Deguchi; Ei Itobayashi; Shigeru Mikami; Akio Moriya; Hironao Okubo; Joji Tani; Akihito Tsubota; Yasuhito Tanaka; Tsutomu Masaki; Katsuhiko Iwakiri; Takashi Kumada
Journal:  J Gastroenterol       Date:  2018-05-08       Impact factor: 6.772

View more

北京卡尤迪生物科技股份有限公司 © 2022-2023.