Literature DB >> 27838748

Effects of the benzodiazepine inverse agonist FG7142 on the structure of anxiety-related behavior of male Wistar rats tested in hole board.

Maurizio Casarrubea1,2, Fabiana Faulisi1, Massimiliano Pensabene1,3, Claudio Mendola1,3, Riccardo Dell'Utri1, Maurizio Cardaci3,2, Andrea Santangelo1,4, Giuseppe Crescimanno5,6.   

Abstract

RATIONALE: Little is known about the structural characteristics of the behavior of rats with enhanced anxiety level. To fill this gap, a study was undertaken where effects of an anxiogenic drug were examined on behavioral structure of rats tested in hole board.
OBJECTIVES: This study investigates effects of increased anxiety level on the structure of the behavior of rats tested in hole board
METHODS: Different doses of FG7142 (1, 4, 8 mg/kg IP), a potent anxiety-inducing drug, were administered to three groups of male Wistar rats. A further group was administered saline. Experiments were recorded through a digital camera. Quantitative and multivariate approaches were applied.
RESULTS: Percent distributions and durations showed increases of immobile sniffing, rearing, head dip, and edge sniff and a significant reduction of grooming activities and of walking. In addition, a decrease of head dip/edge sniff ratio was detected. Transition matrices evidenced that FG7142 provoked evident modifications of behavioral structure mainly of general exploration of environment and focused exploration of the hole. Finally, adjusted residuals showed a reduced effectiveness of FG7142 on transitions from head dip to edge sniff; on the contrary, transitions from edge sniff to head dip underwent evident dose-dependent changes.
CONCLUSIONS: Present study provides a useful tool to analyze behavioral responses to different anxiety conditions. Accordingly, it is demonstrated that a condition of increased anxiety deeply modifies the structure of male Wistar rat's behavior in hole board. In addition, our results suggest that evaluation of head dip/edge sniff ratio can be considered a reliable index to appraise effects of pharmacological manipulation of anxiety and related behavioral elements.

Entities:  

Keywords:  Adjusted residuals; Anxiety; Cluster analysis; Edge sniff; FG7142; Head dip; Hole board; Wistar rat

Mesh:

Substances:

Year:  2016        PMID: 27838748     DOI: 10.1007/s00213-016-4474-8

Source DB:  PubMed          Journal:  Psychopharmacology (Berl)        ISSN: 0033-3158            Impact factor:   4.530


  47 in total

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Review 2.  Neotic preferences in laboratory rodents: issues, assessment and substrates.

Authors:  Robert N Hughes
Journal:  Neurosci Biobehav Rev       Date:  2007-01-02       Impact factor: 8.989

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Journal:  Psychopharmacology (Berl)       Date:  1976-11-24       Impact factor: 4.530

5.  Learning influence on the behavioral structure of rat response to pain in hot-plate.

Authors:  Maurizio Casarrubea; Filippina Sorbera; Andrea Santangelo; Giuseppe Crescimanno
Journal:  Behav Brain Res       Date:  2011-07-20       Impact factor: 3.332

Review 6.  Pharmacology of the beta-carboline FG-7,142, a partial inverse agonist at the benzodiazepine allosteric site of the GABA A receptor: neurochemical, neurophysiological, and behavioral effects.

Authors:  Andrew K Evans; Christopher A Lowry
Journal:  CNS Drug Rev       Date:  2007

7.  Structure of rat behavior in hole-board: I) multivariate analysis of response to anxiety.

Authors:  Maurizio Casarrubea; Filippina Sorbera; Giuseppe Crescimanno
Journal:  Physiol Behav       Date:  2008-10-09

8.  Multivariate data handling in the study of rat behavior: an integrated approach.

Authors:  Maurizio Casarrubea; Filippina Sorbera; Giuseppe Crescimanno
Journal:  Behav Res Methods       Date:  2009-08

9.  Effect of the chronic ingestion of chlorimipramine and desipramine on the hole board response to acute stresses in male rats.

Authors:  E L Rodríguez Echandía; S T Broitman; M R Fóscolo
Journal:  Pharmacol Biochem Behav       Date:  1987-02       Impact factor: 3.533

10.  The exploratory behaviour of rats in the hole-board apparatus: is head-dipping a valid measure of neophilia?

Authors:  Gillian R Brown; Christopher Nemes
Journal:  Behav Processes       Date:  2008-03-12       Impact factor: 1.777

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5.  Combining Quantitative and Qualitative Data in the Study of Feeding Behavior in Male Wistar Rats.

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6.  Effects of Different Anxiety Levels on the Behavioral Patternings Investigated through T-pattern Analysis in Wistar Rats Tested in the Hole-Board Apparatus.

Authors:  Maurizio Casarrubea; Giuseppe Di Giovanni; Giuseppe Crescimanno
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7.  Effects of high fat or high sucrose diet on behavioral-response to social defeat stress in mice.

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8.  Different Representation Procedures Originated from Multivariate Temporal Pattern Analysis of the Behavioral Response to Pain in Wistar Rats Tested in a Hot-Plate under Morphine.

Authors:  Maurizio Casarrubea; Stefania Aiello; Andrea Santangelo; Giuseppe Di Giovanni; Giuseppe Crescimanno
Journal:  Brain Sci       Date:  2019-09-12
  8 in total

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