Literature DB >> 27748721

Precision Medicine and Pancreatic Cancer: A Gemcitabine Pathway Approach.

James J Farrell1, Jennifer Moughan, Jonathan L Wong, William F Regine, Paul Schaefer, Al B Benson, John S Macdonald, Xiyong Liu, Yun Yen, Raymond Lai, Zhong Zheng, Gerold Bepler, Chandan Guha, Hany Elsaleh.   

Abstract

OBJECTIVES: There is a need for validated predictive markers of gemcitabine response to guide precision medicine treatment in pancreatic cancer. We previously validated human equilibrative nucleoside transporter 1 as a predictive marker of gemcitabine treatment response using Radiation Therapy Oncology Group 9704. Controversy exists about the predictive value of gemcitabine metabolism pathway biomarkers: deoxycytidine kinase (DCK), ribonucleotide reductase 1 (RRM1), RRM2, and p53R2.
METHODS: Radiation Therapy Oncology Group 9704 prospectively randomized 538 patients after pancreatic resection to receive either 5-fluorouracil or gemcitabine. Tumor DCK, RRM1, RRM2, and p53R protein expressions were analyzed using a tissue microarray and immunohistochemistry and correlated with treatment outcome (overall survival and disease-free survival) by unconditional logistic regression analysis.
RESULTS: There were 229 patients eligible for analysis from both the 5-fluorouracil and gemcitabine arms. Only RRM2 protein expression, and not DCK, RRM1, or p53R2 protein expression, was associated with survival in the gemcitabine treatment arm.
CONCLUSIONS: Despite limited data from other nonrandomized treatment data, our data do not support the predictive value of DCK, RRM1, or p53R2. Efforts should focus on human equilibrative nucleoside transporter 1 and possibly RRM2 as valid predictive markers of the treatment response of gemcitabine in pancreatic cancer.

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Year:  2016        PMID: 27748721      PMCID: PMC5119656          DOI: 10.1097/MPA.0000000000000710

Source DB:  PubMed          Journal:  Pancreas        ISSN: 0885-3177            Impact factor:   3.327


  50 in total

1.  Human equilibrative nucleoside transporter 1 level does not predict prognosis in pancreatic cancer patients treated with neoadjuvant chemoradiation including gemcitabine.

Authors:  Natsuko Kawada; Hiroyuki Uehara; Kazuhiro Katayama; Satoaki Nakamura; Hidenori Takahashi; Hiroaki Ohigashi; Osamu Ishikawa; Shigenori Nagata; Yasuhiko Tomita
Journal:  J Hepatobiliary Pancreat Sci       Date:  2012-11       Impact factor: 7.027

2.  Predictive and prognostic roles of ribonucleotide reductase M1 in resectable pancreatic adenocarcinoma.

Authors:  Hao Xie; Wei Jiang; John Jiang; Yixin Wang; Richard Kim; Xiaobo Liu; Xiuli Liu
Journal:  Cancer       Date:  2012-06-26       Impact factor: 6.860

3.  Expression status of ribonucleotide reductase small subunits hRRM2/p53R2 as prognostic biomarkers in stage I and II non-small cell lung cancer.

Authors:  Nan-Yung Hsu; Jeng-Yuan Wu; Xiyong Liu; Yun Yen; Chih-Yi Chen; Ming-Chih Chou; Chun-Hsuan Lin; Huei Lee; Ya-Wen Cheng
Journal:  Anticancer Res       Date:  2011-10       Impact factor: 2.480

4.  ERCC1 and RRM1 gene expressions but not EGFR are predictive of shorter survival in advanced non-small-cell lung cancer treated with cisplatin and gemcitabine.

Authors:  P Ceppi; M Volante; S Novello; I Rapa; K D Danenberg; P V Danenberg; A Cambieri; G Selvaggi; S Saviozzi; R Calogero; M Papotti; G V Scagliotti
Journal:  Ann Oncol       Date:  2006-09-15       Impact factor: 32.976

5.  Transcription analysis of human equilibrative nucleoside transporter-1 predicts survival in pancreas cancer patients treated with gemcitabine.

Authors:  Elisa Giovannetti; Mario Del Tacca; Valentina Mey; Niccola Funel; Sara Nannizzi; Sergio Ricci; Cinzia Orlandini; Ugo Boggi; Daniela Campani; Marco Del Chiaro; Mauro Iannopollo; Generoso Bevilacqua; Franco Mosca; Romano Danesi
Journal:  Cancer Res       Date:  2006-04-01       Impact factor: 12.701

6.  Stable suppression of the R2 subunit of ribonucleotide reductase by R2-targeted short interference RNA sensitizes p53(-/-) HCT-116 colon cancer cells to DNA-damaging agents and ribonucleotide reductase inhibitors.

Authors:  Z Ping Lin; Michael F Belcourt; Joseph G Cory; Alan C Sartorelli
Journal:  J Biol Chem       Date:  2004-04-19       Impact factor: 5.157

7.  An analysis of human equilibrative nucleoside transporter-1, ribonucleoside reductase subunit M1, ribonucleoside reductase subunit M2, and excision repair cross-complementing gene-1 expression in patients with resected pancreas adenocarcinoma: implications for adjuvant treatment.

Authors:  Sarah B Fisher; Sameer H Patel; Pelin Bagci; David A Kooby; Bassel F El-Rayes; Charles A Staley; N Volkan Adsay; Shishir K Maithel
Journal:  Cancer       Date:  2012-05-08       Impact factor: 6.860

8.  Gemcitabine chemoresistance and molecular markers associated with gemcitabine transport and metabolism in human pancreatic cancer cells.

Authors:  Y Nakano; S Tanno; K Koizumi; T Nishikawa; K Nakamura; M Minoguchi; T Izawa; Y Mizukami; T Okumura; Y Kohgo
Journal:  Br J Cancer       Date:  2007-01-16       Impact factor: 7.640

9.  Human equilibrative nucleoside transporter 1 and Notch3 can predict gemcitabine effects in patients with unresectable pancreatic cancer.

Authors:  K Eto; H Kawakami; M Kuwatani; T Kudo; Y Abe; S Kawahata; A Takasawa; M Fukuoka; Y Matsuno; M Asaka; N Sakamoto
Journal:  Br J Cancer       Date:  2013-03-14       Impact factor: 7.640

10.  Randomized, multicenter, phase II study of CO-101 versus gemcitabine in patients with metastatic pancreatic ductal adenocarcinoma: including a prospective evaluation of the role of hENT1 in gemcitabine or CO-101 sensitivity.

Authors:  Elizabeth Poplin; Harpreet Wasan; Lindsey Rolfe; Mitch Raponi; Tone Ikdahl; Ihor Bondarenko; Irina Davidenko; Volodymyr Bondar; August Garin; Stefan Boeck; Steffen Ormanns; Volker Heinemann; Claudio Bassi; T R Jeffrey Evans; Roland Andersson; Hejin Hahn; Vince Picozzi; Adam Dicker; Elaina Mann; Cynthia Voong; Paramjit Kaur; Jeff Isaacson; Andrew Allen
Journal:  J Clin Oncol       Date:  2013-11-12       Impact factor: 44.544

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  6 in total

Review 1.  Biomarker-Based Therapy in Pancreatic Ductal Adenocarcinoma: An Emerging Reality?

Authors:  Benjamin A Krantz; Eileen M O'Reilly
Journal:  Clin Cancer Res       Date:  2017-12-21       Impact factor: 12.531

2.  Gambogic acid sensitizes gemcitabine efficacy in pancreatic cancer by reducing the expression of ribonucleotide reductase subunit-M2 (RRM2).

Authors:  Guanggai Xia; Hongcheng Wang; Ziliang Song; Qingcai Meng; Xiuyan Huang; Xinyu Huang
Journal:  J Exp Clin Cancer Res       Date:  2017-08-10

3.  Enhancing Drug Efficacy and Therapeutic Index through Cheminformatics-Based Selection of Small Molecule Binary Weapons That Improve Transporter-Mediated Targeting: A Cytotoxicity System Based on Gemcitabine.

Authors:  Justine M Grixti; Steve O'Hagan; Philip J Day; Douglas B Kell
Journal:  Front Pharmacol       Date:  2017-03-27       Impact factor: 5.810

4.  Human equilibrative nucleoside transporter-1 (hENT1) and ribonucleotide reductase regulatory subunit M1 (RRM1) expression; do they have survival impact to pancreatic cancer?

Authors:  Dae Wook Hwang; Eun Shin; Jai Young Cho; Ho-Seong Han; Yoo-Seok Yoon
Journal:  Ann Hepatobiliary Pancreat Surg       Date:  2020-05-31

5.  Expression of CHPF modulates cell proliferation and invasion in lung cancer.

Authors:  Chengsong Cao; Yong Liu; Qun Wang; Jing Zhao; Ming Shi; Junnian Zheng
Journal:  Braz J Med Biol Res       Date:  2020-04-27       Impact factor: 2.590

6.  Super-Enhancer-Associated Hub Genes In Chronic Myeloid Leukemia Identified Using Weighted Gene Co-Expression Network Analysis.

Authors:  Hongying Ma; Jian Qu; Jian Luo; Tingting Qi; Huanmiao Tan; Zhaohui Jiang; Haiwen Zhang; Qiang Qu
Journal:  Cancer Manag Res       Date:  2019-12-23       Impact factor: 3.989

  6 in total

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